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1996 amino acids, peptides amino acids, peptides U 0400 07 - 246 Coupling of N-Trifluoroacetyl Amino Acids under ”Neutral” Condi- tions. Silylation of the title amino acids before coupling under classical conditions is found to produce higher yields of peptides with concomitant essential decrease of racemization (1-4% d,l product). — (BENOUARGHA, A.; VERDUCCI, J.; JACQUIER, R.; Bull. Soc. Chim. Fr. 132 (1995) 8, 824-828; CNRS, Aminoacides Pept., Univ. Montpellier II, F-34095 Montpellier, Fr.; FR) 1

ChemInform Abstract: Coupling of N-Trifluoroacetyl Amino Acids under “Neutral” Conditions

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1996 amino acids, peptides

amino acids, peptidesU 0400

07 - 246Coupling of N-Trifluoroacetyl Amino Acids under ”Neutral” Condi-tions. — Silylation of the title amino acids before coupling under classicalconditions is found to produce higher yields of peptides with concomitantessential decrease of racemization (1-4% d,l product). — (BENOUARGHA,A.; VERDUCCI, J.; JACQUIER, R.; Bull. Soc. Chim. Fr. 132 (1995) 8,824-828; CNRS, Aminoacides Pept., Univ. Montpellier II, F-34095 Montpellier,Fr.; FR)

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