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ChemInform 2011, 42, issue 27 © 2011 Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim General R 0010 DOI: 10.1002/chin.201127103 Transformation of Anionically Activated Trifluoromethyl Groups to Heterocycles under Mild Aqueous Conditions. — A wide range of heterocyclic compounds is pre- pared in a one-pot one-step reaction without any organic solvent. Excellent functional group tolerance is shown. — (QIAO*, J. X.; WANG, T. C.; HU, C.; LI, J.; WEXLER, R. R.; LAM, P. Y. S.; Org. Lett. 13 (2011) 7, 1804-1807, http://dx.doi.org/10.1021/ol200326u ; Bristol-Myers Squibb Res. Dev., Princeton, NJ 08543, USA; Eng.) — R. Steudel 27- 103

ChemInform Abstract: Transformation of Anionically Activated Trifluoromethyl Groups to Heterocycles under Mild Aqueous Conditions

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Page 1: ChemInform Abstract: Transformation of Anionically Activated Trifluoromethyl Groups to Heterocycles under Mild Aqueous Conditions

GeneralR 0010 DOI: 10.1002/chin.201127103

Transformation of Anionically Activated Trifluoromethyl Groups to Heterocycles under Mild Aqueous Conditions. — A wide range of heterocyclic compounds is pre-pared in a one-pot one-step reaction without any organic solvent. Excellent functional group tolerance is shown. — (QIAO*, J. X.; WANG, T. C.; HU, C.; LI, J.; WEXLER, R. R.; LAM, P. Y. S.; Org. Lett. 13 (2011) 7, 1804-1807, http://dx.doi.org/10.1021/ol200326u ; Bristol-Myers Squibb Res. Dev., Princeton, NJ 08543, USA; Eng.) — R. Steudel

27- 103

ChemInform 2011, 42, issue 27 © 2011 Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim

Page 2: ChemInform Abstract: Transformation of Anionically Activated Trifluoromethyl Groups to Heterocycles under Mild Aqueous Conditions

ChemInform 2011, 42, issue 27 © 2011 Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim

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