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December 5-7, 2016 Dubai, UAE
International Conference onMedicinal and Pharmaceutical Chemistry
PharmaMed-2016
Media Partners
Day 1 - December 5, 2016 - Al Shaheen08:00-09:30 Registrations
09:30-10:00 Opening Ceremony
Keynote Forum
10:00-10:30Title: Key requirements for successful transnational drug discovery projects
Sheraz Gul, Fraunhofer Institute for Molecular Biology & Applied Ecology, Germany
10:30-11:00Title: Applications in pharmaceuticals and drug analysis of modifi ed carbon paste electrodes using different voltammetric techniques
Mahmoud Khodari, South Valley University, Egypt
Coffee Break: 11:00-11:15 @ Foyer B
Session 1: Novel Opportunities for Drug Discovery and Medicinal ChemistrySession Chairs: Raphael Stoll, Ruhr University of Bochum, Germany Rebamang A. Mosa, University of Zululand, Republic of South Africa
11:15-11:40Title: Ruthenium-conjugated synthetic fl avonoid derivatives as novel modulators of platelet function
Sakthivel Vaiyapuri, University of Reading, UK
11:40-12:05Title: Lead modifi cation approaches in the design, synthesis and evaluation of novel chemical entities for muscarinic acetylcholine receptors
Richie R. Bhandare, Ajman University of Science and Technology, UAE
12:05-12:30Title: Biological activity of nanocomposites consisting of TiO2 nanoparticles and antisense oligonucleotides
Asya S. Levina, Novosibirsk State University, Russia
12:30-12:55Title: Bisphenol an analogues bind to ras proteins and compete with guanine nucleotide exchange
Raphael Stoll, Ruhr University of Bochum, Germany
Lunch Break: 12:55-14:00 @ Restaurant
14:00-14:25Title: Toward the design of novel antimicrobials: Synthesis and biological evaluation of phosphate isosters of fosmidomycin and analogs
Catherine Grosdemange-Billiard, Université de Strasbourg/CNRS, France
14:25-14:50Title: Cardioprotective potential of a lanosteryltriterpene from Protorhuslongifolia
Rebamang A. Mosa, University of Zululand, Republic of South Africa
14:50-15:15Title: Structural modifi cations of kidney cystatin in renal cancers
Mohd Anas Shamsi, Aligarh Muslim University, India
15:15-15:40Title: The dual-acting AChEInhibitor and H3 receptor antagonist UW-MD-72 reverses amnesia induced byscopolamine or dizocilpinein passive avoidance paradigm in rats
Bassem Sadek, United Arab Emirates University, United Arab Emirates
15:40-16:05Title: Physicochemical analysis of antioxidant compounds in fresh juice from cactus cladodes
TALBI Meryeme, University Hassan 1er, Morocco
Coffee Break: 16:05-16:20 @ Foyer B
Day 2 - December 6, 2016 - Al ShaheenKeynote Forum
09:30-10:00Title: Biomolecular NMR spectroscopy in medicinal chemistry
Raphael Stoll, Ruhr University of Bochum, Germany
10:00-10:30Title: Protective effects of apricot againist ketamin ıncuduced hepatotoxicity in rats
Ismet Yilmaz, Inonu University, Turkey
Coffee Break: 10:30-10:45 @ Foyer B
Session 2: Antibiotics and Anti Cancer Drugs Molecular Modeling and Computer-Aided Drug Design Pharmaceutical Analysis: Analytical MethodsSession Chairs: Mahmoud Khodari, South Valley University, Egypt
10:45-11:10Title: Fluoroquinolone-associated toxicities: Tipping the risk-benefi t scale
Monique R. Bidell, Albany College of Pharmacy and Health Sciences, USA
11:10-11:35Title: Design, synthesis and biological characterization of chalcones and propanediones as inhibitors of histone methyl transferase against leukemia cell lines
C. S Ramaa, Bharati Vidyapeeth’s College of Pharmacy, India
11:35-12:00Title: Discovery and optimization of novel antagonists of the WDR5-MLL interaction
Rima Al-awar, University of Toronto, Canada
12:00-12:25Title: Homology modelling, structure- and ligand-based drug design of novel tubulin inhibitors and calcium channel blockers with anti- proliferative and leishmanicidal activities
Carlos Henrique Tomich de Paula da Silva, University of São Paulo, Brazil
12:25-12:50Title: Selective electrochemical determination of desipramine using a lipid modifi ed carbon paste electrode
Mahmoud Khodari, South Valley University, Egypt
Lunch Break: 12:50-13:35 @ Restaurant
Session 3: Drug Design, Discovery and Development Pharmaceutical Analysis: Analytical Methods Pharmacology and ToxicologySession Chairs: Usharani Pingali, Nizam’s Institute of Medical Sciences (NIMS), India Marcela Krečmerová, Czech Academy of Sciences, Czech Republic
13:35-14:00Title: Antiviral acyclic nucleoside phosphonates: New structures and prodrugs
Marcela Krečmerová, Czech Academy of Sciences, Czech Republic
14:00-14:25Title: Design and synthesis of benzoazoles incorporating fl uorine and piperazine moieties with potential biological activities
Raid Abdel-jalil, Sultan Qaboos University, Oman
14:25-14:50Title: A Study of highly standardized aqueous extract of Terminalia chebula 250mg, 500mg versus Placebo in modifying cardiovascular risk with special reference to Endothelial dysfunction in patients with Type2 Diabetes
Usharani Pingali, Nizam’s Institute of Medical Sciences (NIMS), India
14:50-15:15Title: Structure-affi nity and structure-kinetics relationship study: A new combination strategy in medicinal chemistry
Dong Guo, Xuzhou Medical University, China
15:15-15:40Title: Synthesis, anti-inflammatory, analgesic, molecular modeling and admet studies of diclofenylalanylhydrazide
Magda Hassan Abd El Lattif, Taif University, Kingdom of Saudi Arabia
15:40-16:05Title: Synthesis of zinc oxide doped- poly(8-anilino-1-napthlene sulphonic acid) (ZnO/PANSA) as conducting platforms for TB drug biosensors
Rachel Ajayi, University of the Western Cape, South Africa
Coffee Break: 16:05-16:15 @ Foyer B
Workshop
16:15-18:00Title: A critical evaluation of assays in pre-clinical drug discovery
Sheraz Gul, Fraunhofer Institute for Molecular Biology & Applied Ecology, Germany
Day 3 - December 7, 2016 - Al ShaheenPoster Presentations: 10:00-12:30 @ Foyer B
P1Title: Role of formyl peptide receptors in the regulation of thrombosis and haemostasis
Maryam Salamah, University of Reading, UK
P2Title: Cytotoxic effects of bioactive compounds isolated of Iris persica L. on human cancer cell lines
Faiq H. S. Hussain, University of Salahaddin, Iraq
P3Title: A practical and eco-friendly synthesis of oxo-bile acids
Hwayoung Yun, Pusan National University, Republic of Korea
P4Title: Synthesis and cellular uptake of nanocomposites containing oligonucleotides and their analogues immobilized on inorganic nanoparticles
Marina N. Repkova, Novosibirsk State University, Russia
P5Title: In-vitro antidiabetic activity of partially purifi ed fractions of Pithecellobium dulce fruit
Preethi S, VIT University, India
P6Title: Apoptosis versus autophagy in the molecular mechanism of action of plant derived chemotherapeutics against hepatocellular carcinoma cells
Greeshma Tom, Rajiv Gandhi Centre for Biotechnology, India
P7Title: Anti-infl ammatory action through inhibition of NF kB activation and translocation by band-2 isolated from Tinospora cordifolia(Thunb.) miers. in LPS stimulated RAW 264.7 cell lines
Sheena Philip, Rajiv Gandhi Centre for Biotechnology, India
P8Title: Identifi cation of structural elements of MCP chemokines and their shared receptor CCR2
Zil e Huma, Monash University, Australia
P9Title: Targeting bacterial stringent response
Dominik Rejman, Czech Academy of Sciences v.v.i., Czech Republic
P10Title: Characterization of nucleotide pool in bacterial cells
Eva Zborníková, Czech Academy of Sciences v.v.i., Czech Republic
P11Title: Design TiO2 nanoparticles for using in nanocomposites containing oligonucleotides and their analogues
Elena V Bessudnova, Novosibirsk State University, Russia
P12Title: Low dose irbesartan has a renoprotective effect as high dose ramipril in diabetic rats treated with insulin
Abdulelah A. Thigah, Umm Al-Qura university, Saudi Arabia
P13Title: Aspirin and blood glucose and insulin resistance
Abdullah A. Alshamrani, Umm Al-Qura university, Saudi Arabia
P14Title: Prevalence and preventive measures of infertility in male by kruger’s criteria, a randomized study in private and government health care hospitals
Huda Ashraf, Jinnah University for Women, Pakistan
P15Title: In silico pharmacokinetics and molecular docking of three leads isolated from Tarconanthus Camphoratus L
Amina I. Dirar, Medicinal and Aromatic Plants Research Institute, Sudan
P16Title: Zika virus NS5 protein potential inhibitors: An enhanced in silico approach in drug discovery
Pritika Ramharack, University of KwaZulu-Natal, South Africa
Coffee Break: 11:00-11:15 @ Foyer B
Award Ceremony