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2003-2004GI Diseases Review
April 18, 202305:44 PM
Activated charcoal
Antidote
Alosetron
IBS treatment
5HT3 receptor antagonist
Aluminum hydroxide
Antiulcer
Antacid
Amoxicillin
Penicillin antibioticCell wall synthesis inhibitor
Antiulcer
Amino penicillinInhibits peptidoglycan cross-
linking
Ampicillin
Penicillin antibioticCell wall synthesis inhibitor
Amino penicillinInhibits peptidoglycan cross-
linking
Anthraquinonescascara segrada, danthron, senna
Contact cathartics
Aprepitant dimenhydrinate
Antiemetic
Neurokinin 1 receptor antagonist
Atropine
Anticholinergic
AntimuscarinicTreatment for bradycardia,
diarrhea, cholinesterase poisoning
Azithromycin
Macrolide antibioticBacteriostatic protein synthesis
inhibitor
50S ribosome Inhibits translocation
Balsalazide
NSAID (salicylate)
Treatment of IBD
Bisacodyl
Contact cathartic
Bismuth subsalicylate
AntiulcerAntidiarrheal
Budesonide
AdrenocorticosteroidGlucocorticoid
Anti-inflammatory steroidInhaled OR treatment of IBD
Calcium carbonate
Antiulcer
Antacid
Cascara sagrada
Contact cathartic
Anthraquinone derivative
Castor Oil
Contact cathartic
Cimetidine
AntihistamineAntiulcer
H2 receptor antagonist
Cisapride
Prokinetic agent
5HT4 agonist
Clarithromycin
Macrolide antibioticBacteriostatic protein synthesis
inhibitor Antiulcer
50S ribosomeInhibits translocation
Danthron
Contact cathartic
Anthraquinone derivative
Dexamethasone
AdrenocorticosteroidGlucocorticoidAntineoplastic
Antiemetic
Anti-inflammatory steroidNot by inhalation
Dimenhydrinate
AntihistamineAntiemetic
H1 receptor antagonist
Diphenhydramine
Classical antihistamineAntiemetic
H1 antagonist
Diphenoxylate docusate
Antidiarrheal
Opiate
Docusates
Lubricating laxatives
Stool softeners
Doxycycline
Tetracycline antibioticBacteriostatic protein synthesis
inhibitor
30S ribosomePrevents aminoacyl tRNA attachment
Dronabinol
Antiemetic
Cannabinoid
Droperidol
Antiemetic
D2 receptor antagonist
Erythromycin
Macrolide antibioticBacteriostatic protein synthesis
inhibitor
50S ribosomeInhibits translocation
Granisetron
Antiemetic
5HT3 receptor antagonist
Infliximab
TNF inhibitor
Anti-TNF monoclonal antibody Treatment of IBD
Ipecac
Emetic
Kaolin
Antidiarrheal
Lactulose
Saline (osmotic) cathartic
Lansoprazole
Antiulcer
H+/K+ ATPase inhibitor
Loperamide
Antidiarrheal
Opiate
Magnesium hydroxide
AntiulcerSaline (osmotic) cathartic
Antacid
Meclizine
AntihistamineAntiemetic
H1 receptor antagonist
Mesalamine(5-ASA)
NSAID (salicylate)
Treatment of IBD
Methylcellulose
Bulk laxative
Metoclopramide
Prokinetic agentAntiemetic
D2 antagonist
Metronidazole
AntibioticAntiparasitic
Antiulcer
AnaerobesReduction leads to intermediates
that damage DNA
Mineral oil
Lubricating laxative
Stool softener
Minocycline
Tetracycline antibioticBacteriostatic protein synthesis
inhibitor
30S ribosomePrevents aminoacyl tRNA attachment
Misoprostol
ProstaglandinAntiulcer
Olsalazine
NSAID (salicylate)
Treatment of IBD
Omeprazole/esomeprazole
Antiulcer
H+/K+ ATPase inhibitor
Ondansetron
Antiemetic
5HT3 receptor antagonist
Oxytetracycline
Tetracycline antibioticBacteriostatic protein synthesis
inhibitor
30S ribosomePrevents aminoacyl tRNA attachment
Pantoprazole
Antiulcer
H+/K+ ATPase inhibitor
Pectin
Antidiarrheal
Polyethylene glycol- electolyte solution
AntidoteCathartic
Procarbazine
Antineoplastic
MiscellaneousProbably acts as alkylating
agent
Prochlorperazine
Antiemetic
D2 receptor antagonistPhenothiazine
Promethazine
Classical antihistamineAntipsychotic
Antiemetic
H1 antagonist
Rabeprazole
Antiulcer
H+/K+ ATPase inhibitor
Ranitidine
AntihistamineAntiulcer
H2 receptor antagonist
Rebamipide
Antiulcer
Senna
Contact cathartic
Anthraquinone derivative
Scopolamine
AnticholinergicAntiemetic
Muscarinic receptor antagonist
Simethicone
Anti-flatulent
Sodium bicarbonate
AntiulcerAntidote
AntacidAlkalinization of urine to treat drug toxicity (esp. barbiturates, salicylates,
methanol)
Sodium phosphate
Saline (osmotic) cathartic
Sucralfate
Antiulcer
Sulfasalazine
Disease modifyinganti-rheumatic drug (DMARD)
Metabolized to sulfonamide+ salicylate (NSAID) Treatment of IBD
Tegaserod
Antiemetic
5HT4 receptor agonist
Tetracycline
AntibioticBacteriostatic protein synthesis
inhibitor Antiulcer
30S ribosomePrevents aminoacyl tRNA attachment