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Nervous System
CNS Brain & spinal cord
Acetyl choline
Dopamine
Serotonin
Norepinephrine
GABA
Glutamate
Opioids
Somatic Neuromuscular junction Nicotinic (ACh)
PNS
PSNS Organs, glands Muscarinic (ACh)
SNS CV & lung smooth muscle
Alpha (NE)
Beta (NE) Enteric Many
neurotransmitters
PSNS
Muscarinic
Bethanechol
Pilocarpine
Donepezil
Neostigmine
Anti Muscarinic
Atropine
Scopolamine
1st Generation antihistamines
Tricyclic antidepressants
CNS
Acetyl choline
Anti-‐Alzheimer's, Smoking cessation, Antiemetics
Dopamine Anti Parkinson's, Anti EPS, Antipsychotics, ADHD,
Antiemetics
GABA AEDs, Sedatives, Hypnotics, General anesthetics
Glutamate Ketamine, Memantine
Norepinephrine Antidepressants, Antipsychotics, Antihypertensive
Opioids Sedation, Analgesia, Addiction, Antitussive, Antidiarrheal
Serotonin Antidepressants, Antipsychotics, Antiemetics, Antimigraine
SNS
Alpha
Antagonists
Alpha 1
Doxazosin
Tamsulosin
Mixed
Phentolamine
Agonists
Alpha 2
Clonidine
Mixed
Ephedrine
Oxymetazoline
Phenylephrine
Pseudoephedrine
Mixed Alpha and Beta
Agonists
Dobutamine
Catecholamines
Antagonists
Labetalol
Beta
Agonists
Albuterol
Isoproterenol
Salmeterol
Terbutaline
Antagonists
Atenolol
Metoprolol
Propranolol