BIO-DATA OF M - Maharaja Sayajirao University of … · Web viewBIO-DATA OF M.R.YADAV Name : Dr. M. R. Yadav PERSONAL Address : Official Residential Pharmacy Department, Faculty of

BIO-DATA OF M.R.YADAV

Name : Dr. M. R. Yadav

PERSONALAddress :Official ResidentialPharmacy Department, Faculty of Technology and Engineering, The M. S. University of Baroda,Vadodara– 390 001, Gujarat

B-1, Kalyan Nagar (Opp. Anant Park, Near Sabari School) Vasna Road, Vadodara-390 015Gujarat

Date of Birth : 21st September 1954E-mail address : [email protected], [email protected] No. : (O): 0265-2434187

FAX: 0265-2418927, 2423898 (M): 09426721112

EDUCATIONALEducational Qualifications :

Degree Institution Field /Subject(s) Year Positions

B. Pharmacy University of Delhi, Delhi Pharmacy 1976 IInd Rank

M. Pharmacy B.H.U., Varanasi Pharmaceutical Chemistry 1982 Ist Rank

Ph. D. Panjab University, Chandigarh Pharmaceutical Chemistry 1986 -

PRESENT POSITION

PROFESSOR & HEAD OF THE DEPARTMENTPharmacy Department, Faculty of Technology, Kalabhavan,The M. S. University of Baroda, Vadodara- 390 001

SPECIAL RECOGNITION Organized Graduate Pharmacy Aptitude Test for Pharmacy Graduates [GPAT-2010

Examination (AICTE, New Delhi)] as Co-ordinator, for the FIRST TIME in INDIA. Organized GPAT-2011 & GPAT-2012 Examinations, an All India level examination

organized under the aegis of AICTE, New Delhi, for Pharmacy Graduates consecutively for THREE years, wherein about forty five thousand students appeared each year.

REPRESENTATION IN NATIONAL BODIES1

mailto:[email protected]

Member, Scientific Body, National Pharmacopoeia Commission, Ministry of Health & Family Welfare, Govt. of India

Chairman, Pharmacy Accreditation Evaluation Committee of National Board of Accreditation, New Delhi for a period of three years from 31st May 2010.

Chairman, National Advisory/Monitoring Committee for GPAT, AICTE, New Delhi from Nov 2009 –Oct 2011

Coordinator, National Monitoring Committee-GPAT, AICTE, New Delhi from Nov 2010 to June 2012.

Expert Member, Project Evaluation Committee, UGC, New Delhi Member, Executive Committee of National Board of Accreditation for empanelment of

Chairpersons/Experts in the field of Pharmacy, NBA, New Delhi Member National Board of Accreditation (NBA), AICTE, New Delhi from May 2010 for

three years. Member of South Central Regional Committee, AICTE, Hyderabad, from May 2010 for

three years. Member of All India Board for Pharmacy Education (AIB-PE), AICTE, New Delhi from June

2006-May 2009. Member of Sectoral Committee, National Board of Accreditation (NBA) for Management

and Pharmacy, AICTE, New Delhi from Aug 2006-July 2009. Member, Scientific Services Committee, IPC, from 2004-2006

AWARDS RECEIVED ‘Pharmacy Teacher of the Year – 2010 Award’ of Association of Pharmacy Teachers of

India Ranbaxy Laboratories’ Silver Medal in B. Pharmacy at University of Delhi, 1976 Best Paper prize in oral session of Medicinal Chemistry at 57 th IPC, Hyderabad, December

2005 Subhash C. Verma Memorial Prize for Best Research Paper presented in the oral scientific

session of 18th All Gujarat Annual Meeting of Indian Pharmacological Society held at Anand Pharmacy college, Anand, January 2004

EMPLOYMENTPRESENT POSITION:

PROFESSOR & HEAD, Pharmacy Department, Faculty of Technology and Engineering, The M.S. University of Baroda, Vadodara-390 001 From 27th February 2010 till date

POSITIONS HELD ACADEMIC:1. Lecturer at Dept. of Pharm. Sciences (Currently, University Institute of Pharmaceutical

Sciences), Panjab University, Chandigarh-160 014 From 20th November 1985 to 31st January 1992

2. Assistant Professor at College of Pharmacy (Currently, DIPSAR, Delhi Institute of Pharmaceutical Sciences and Research), Government of National Capital Territory of Delhi, Pushp Vihar, Phase-III, New Delhi-110 017

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From 2nd Feb. 1992 to 30th June 19963. Professor of Pharmacy (Pharmaceutical Chemistry), Pharmacy Department, Faculty of

Tech. & Engg., Kalabhavan, The M.S. University of Baroda, Vadodara-390 001 From 1st July 1996 till date

INDUSTRIAL:1. Approved Manufacturing Chemist at M/S Tribhavan Injectables, Kirti Nagar Industrial Area, New Delhi

From 1st Aug. 1976 to 31st July 1980

ADMINISTRATIVE:1. Head, Pharmacy Department, Faculty of Tech. & Engg., The M. S. University of Baroda,

Vadodara From February 27th 2010 till date.

2. Principal Coordinator, Q.I.P. (Pharmacy), AICTE at Pharmacy Department From March 2012 to June 2013.

3. Co-ordinator, Quality Improvement programme in Pharmacy (AICTE), Pharmacy Department, The M.S. University of Baroda, Vadodara.

From May 2003 to July 20054. Co-ordinator, Centre for Post graduate Studies and Research at Shri G.H. Patel Pharmacy

Building, Pharmacy Department, The M.S. University of Baroda, Vadodara. From 1st Aug. 2005 to 31st July 2007

5. Co-ordinator, IPR Cell, The M. S. University of Baroda, Vadodara 6. Head, Department of Pharmaceutical Chemistry, College of Pharmacy (currently DIPSAR)

New Delhi. From Jan. 1994 to June 1996

RESEARCH CONTRIBUTIONRESEARCH INTERESTS: Designing and Synthesis of Medicinal Agents belonging to the following categories:

Selective COX-II inhibitors Steroidal Aromatase inhibitors TACE inhibitors Newer anti-hypertensive agents using dual targeted approach Protease inhibitors as Antimalarial agents Diaryl diazepines as potential anticancer agents Development of Non-Nucleoside Reverse Transcriptase Inhibitors (NNRTI) as antiviral agents Preparation of metal complexes of some known antibiotics as H .pylori

Inhibitors ACAT inhibitors as antihyperlipidemic agents Virtual screening of chemical databases for anticancer and

antimalarial leads Computational studies on selective COX-2, Farnesyltransferase, TACE, HIV

integrase, Telomerase Inhibitors

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RESEARCH PROJECTS HANDLED:

1. DSA Phase-I program of UGC, New Delhi as Co-ordinator, Marh 2013 to Feb 2018, Rs. 98 Lakhs

2. AICTE-MODROB project entitled, “Evaluation of serotinergic and dopaminergic potential of some novel ligands”, March 2013 to March 2014, Rs. 15.0 Lacs.

3. “FIST Program of DST on Molecular Modeling”, March 2011, Rs. 48 Lacs, Continuing from June 2011

4. “Design and Development of Novel Steroidal Aromatase Inhibitors”, RPS (AICTE) Project From April 2008 to March 2010, Rs. 19.5 Lacs

5. “Design and Development of New Specific COX-II Inhibitors”, UGC, New Delhi, Major Research Project from April 2002 to Mar. 2005, Rs. 5.83 Lacs

6. “Development of Protease Inhibitors as Antimalarial Drugs using Computer Aided Drug Design”, TAPTEC Research Project supported by AICTE, New DelhiFrom April 2003 to Mar. 2007, Rs. 14.0 Lacs

7. “Design and Development of New Drugs with Potential Applications in Inflammatory Disorders”, TAPTEC Research Project supported by AICTE, New DelhiFrom April 1998 to Mar. 2000, Rs. 10.0 Lacs

8. “Studies in Neuromuscular Blocking Agents Azasteroids”, UGC (Minor) Research ProjectFrom June 1993 to May 1995, Rs. 38,000/-

ACADEMIC ACHIEVEMENTS:Research Supervision:

Ph. D. : Awarded 19Thesis submitted 01

Synopsis submitted 01Presently Registered 08

M. Pharm (Dessertation) : Supervised 39Under Guidance 03

Ph.D. Examiner at Universities:

Chhatrapati Shahu Ji Maharaj University, Kanpur University of Delhi, Delhi University of Pune, Pune Panjab University, Chandigarh Kakatiya Univeristy, Warangal Hemchandracharya North Gujarat University, Gujarat Swami Ramanad Teerth Marathwada University, Nanded, Maharashtra Devi Ahilya Vishwavidyalaya, Indore Guru Jambheshwar University, Hissar North Maharashtra University, Jalgoan Banaras Hindu University, Varanasi Dr H.S. Gaur Vishwavidyalaya, Sagar Mumbai University, Mumbai Rajiv Gandhi Prodyogiki Vishwavidyalaya, Bhopal Hamdard University (Jamia Hamdard), New Delhi

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Bharti Vidyapeeth Deemed University, Pune

AFFILIATION TO PROFESSIONAL/ACADEMIC/SCIENTIFIC BODIESEXPERT MEMBER OF VARIOUS STATUTATIORY BODIES

Expert member, UGC, New Delhi for evaluation of projects. All India Council for Technical Education, New Delhi, for Approval/Renewal of Various

Pharmacy Courses of Colleges throughout India Pharmacy Council of India, New Delhi, for Approval/Renewal of Degree/Diploma in

Pharmacy courses as PCI Inspector. Expert member of Local Inspection Committee of Gujarat University, Ahmadabad and

Hemchandracharya North Gujarat University, Patan for Affiliation of Colleges to the concern Universities.

REPRESENTATION INBOARDS/COMMITTEES OF THE M.S. UNIVERSITY OF BARODA Member, Finance and Establishment Standing Committee Member, Purchase Committee, The M.S. University of Baroda, Vadodara Chairman, Board of Studies (Pharmacy), The M. S. University of Baroda, Vadodara, 2011-

14 Chairman, Board of Studies (Pharmacy), The M.S. University of Baroda, Vadodara, 2010 Member, Board of Studies (Pharmacy), The M.S. University of Baroda, Vadodara, 1997 -

2009

UNIVERSITY BOARDS Member, Board of Studies in Pharmaceutical Chemistry, Lachoo Memorial College of

Science and Technology (Autonomous), Jodhpur, Rajasthan, 1st July 2012 to 30th June 2014

Member, Faculty of Pharmacy, Ganpat University, Ganpat Vidyanagar, Kherva, Mehsana, Gujarat, 1st March 2012 to 7th Jan 2015

Member, Board of Studies (Pharmacy), Kakatiya University, Warangal, A.P., Jan 2012 to Dec 2014

Member, Board of Studies (Pharmacy), Saurashtra University, Rajkot, 2011 onwards Member, Board of Studies, Ganpat University, Ganpatnagar, Mehsana, 2009-2012 Member, Board of Studies (Pharmacy), Devi Ahilya Vishwavidyalaya, Indore, 2010-2013 Member, Board of Studies, NMIMS, Mumbai, 2007 – 2009 Member, Subject Area Committee, Nirma University, Ahmedabad

EXPERT MEMBER OF SELECTION COMMITTEES

1. Acted as Expert member of Selection Committee in Subject field Biopharmacology for selection of candidates for the Award of DAAD Fellowship, Ministry of Human Resource Development, Government of India, New Delhi.

2. Expert Member Selection Committee for the Posts of Professors/Readers/Lecturers at : Kakatiya University, Warangal, A.P. Jivaji University, Gwalior, M.P. Guru Gobind Singh Indraprashta University, Delhi Shri G.S. Institute of Technology and Science, Indore

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Birla Institute of Technology, Ranchi NMIMS, School of Pharmacy, Mumbai Panjab University, Chandigarh Jamia Hamdard (Deemed University), New Delhi Sardar Patel University, Vallabh Vidya Nagar Gujarat University, Ahmedabad J. N. Vyas University, Jodhpur

CHAIRMAN/C0-CHAIRMAN OF SCIENTIFIC SESSIONS Chairperson, two day National conference on ‘Particle technology with special emphasis

on nanotechnology’ organized by Parul Institute of Pharmacy, Vadodara, 22nd-23rd April 2011

Acted as Chairman, Plenary lecture in IPA Convention 2011, Indore, hosted by IPA M.P. State Branch, Indore (M.P.) held on 19th & 20th Feb 2011.

Acted as Chairman of Medicinal Chemistry Session at Indian Pharmaceutical Congress held at Pune (2002), Chennai (2003), Hyderabad (2005), Mumbai (2006), Varanasi (2007), New Delhi (2008) and Ahmedabad (2009)

Acted a Co-Chairman of Medicinal Chemistry section at Indore (1999), Hyderabad (2000) and New Delhi (2001).

JUDGING OF SCIENTIFIC PRESENTATIONS Acted as a Judge for the Scientific Poster Presentation “Radiotracers in Drug

Development”, XXIV Annual Conference of Indian Association of Biomedical Scientists organised by Institute of Nuclear Medicine and Allied Sciences, DRDO, New Delhi.

ORGANIZING OF SCIENTIFIC/PROFESSIONAL EVENTS Organized two-days AICTE sponsored National Seminar on “Approached in drug discovery” at

Pharmacy Department, The M. S. University of Baroda., Vadodara, on 26 – 27 Feb 2013. Organized UGC sponsored Two days National Seminar on ‘Statistical Analysis in Drug

Development and Discovery’, at Pharmacy Department, The M. S. University of Baroda, Vadodara, on 20th and 21st Jan 2012

Dy. Co-odinator, National seminar on ‘Neutraceuticals and plants in human health’, Department of Botany, The M. S. University of Baroda, Vadodara, Dec 10-11, 2011.

Organized one week AICTE sponsored QIP Staff Development Programme on “Glimpses of Current Advances in The Field of Pharmaceutical Sciences”, at Pharmacy Department, The M. S. University of Baroda from 2nd - 8th June 2010 as Convener.

Organized two days regional seminar on “Intellectual Property and Innovation Management in Knowledge Era” held on 26th and 27th August 2009 at The M. S. University of Baroda, Vadodara as Co-ordinator.

Organised Two weeks ISTE Sponsored Summer School on “Trends in Developments of Drugs & Delivery Systems-A Futuristic Approach” as Co-ordinator at Pharmacy Department, The M.S. University of Baroda, Vadodara From 19th to 31st May 1997.

TRAINING PROGRAMMES ATTENDED

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Workshop cum Retreat on “IP Management in Public Private partnership” organized by INDO-US SCIENCE AND TECHNOLOGY FORUM, TIFAC-DST, Govt. of India at National Center for biological sciences (NCBS), Bangalore, from February 8-10, 2006

“Internet Training Programme”, organized by Computer Center, The M.S.University of Baroda, Vadodara, 11-17th Jan 2000

“Computer Aided Drug Design’, Summer school organised by National Institute of Pharmaceutical Education and Research, S.A.S.Nagar, Punjab, 15 -19th June 1998

ISTE Sponsored Summer Schoold on “Quality Control of Drugs and Pharmaceuticals by Modern Instruments” organized by L.M.College of Pharmacy, Ahmedabad, 8 -21st May 1995.

Post Graduate Teachers Workshop in Medicinal & Analytical Chemistry, organized by K.L.E. College of Pharmacy, Belgaum, 5 -6th June 1993

UGC/DSA Supported Certificate “Course Course-cum-Workshop on QSAR”, organized by Department of Chemical Technology, Matunga, Bombay, Feb 6-8, 1992

ISTE Sponsored course on “ Application of Computer Programming in Pharmaceutial Sciences” organized by L.M.College of Pharmacy, Ahmedabad, 8 -28th May 1988.

EDITORIAL ADVISORY BOARD

Member, Editorial Board, ‘International Journal of Pharmaceutical Sciences and Nanotechnology’, Pharma Book Syndicate, Hyderabad

Member of Editorial Advisory Board of ‘The Open Drug Discovery Journal’ ISSN: 1877 3818, Bentham Open.

Member, Advisory Board for Rajeev Gandhi University of Health Sciences Journal of Pharmaceutical Sciences, Bangalore

JOURNAL REFEREE Bio-organic Medicinal Chemistry (Science Direct) European Journal of Medicinal Chemistry (Science Direct) Journal of Molecular Structure (Science Direct) Immunology and Cell Biology (Nature Publishing Group) Computer-Aided Molecular Design (Springer Link) Journal of Heterocyclic Chemistry (Wiley Interscience) Chemical Biology and Drug Design (Wiley Interscience) Molecular Informatics (Wiley Interscience) Current Medicinal Chemistry (Bentham Science) Medicinal Chemistry (Bentham Science) Medicinal Chemistry Research (Bentham Science) Letters in Drug Design and Discovery (Bentham Science) Mini Reviews in Medicinal Chemistry (Bentham Science)

PROFESSIONAL BODIES IPA Vadodara Branch: President since June 2012 for two years. Life Member of:

Society of Pharmaceutical Education and Research (SPER/LM/GU/009) Indian Society of Technical Education (LM-4312) Indian Pharmaceutical Association (DEL/LM/101)

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India Pharmacy Graduate Association (LM-363) Indian Pharmacological Society (GULM-519) Association of Pharmacy Teachers of India (GU/LM-060)

SPECIAL LECTURE/TALK DELIVERED ABROAD AS RESOURCE PERSON 1. Scientific talk entitled, ‘Dual α1- and AT-1 inhibitors as potential antihypertensive agents’

delivered in Indo-Russian Seminar at National Medical University, Volgograd, Russia held during 8th to 10th Sept 2011

SPECIAL LECTURES/TALKS DELIVERED AS RESOURCE PERSON (NATIONAL)1. Invited lecture entitled, “Strategies for structure elucidation using UV, IR, NMR & MS spectral data”,

organized by Sardar Patel College of Pharmacy, Bakrlol, Anand, Gujarat, in the GUJCOST SPONSORED one day National seminar on “Structural analysis by various spectroscopic techniques” on 1 st Oct 2013

2. Invited lecture entitled, ‘Modeling techniques in drug discovery’ delivered at B.N. Institute of Pharmaceutical Sciences, Udaipur, AICTE sponsored Faculty Development Programme on “ An approach to develop new models in the field of medicinal chemistry” from 16 th 28th Sept 2013 on 16th

Sept 2013. 3. Invited lecture entitled, ‘Refurbishing the image of pharmacy education in the changing scenario’

delivered at Sigma Institute of Pharmacy, Vadodara in AICTE sponsored National level Pharma Carnival on Road map for strengthening pharmacy education in changing scenario (17 th 18th Aug 2013) on 17th August 2013.

4. Invited lecture entitled, ‘High resolution mass spectrometery in drug research’, delivered at Babaria Institute of Pharmacy, Vadodara in AICTE sponsored National Seminar on Quality assurance issues in drug discovery and formulation development, on 27th July 2013.

5. Invited lecture entitled, Targets for cancer chemotherapy’, delivered at Pune District Education Association’s Seth Govind Raghunath sable College of Pharmacy, Saswad, Pune in AICTE sponsored National Seminar on Frontiers in cancer chemotherapy, on 26th July 2013.

6. Invited lecture entitled, ‘Exploring QSAR for lead optimization’ delivered at B.V. Patel PERD Center, Ahmedabad, on 14th May 2013.

7. Expert lecture entitled, ‘Selectivity in mono, di and tri-alkylation of 3-benzazepine scaffold’ at Gujarat Technological University, Ahmedabad on 9th April in “Research week 2013” during April 3-16, 2013.

8. Invited lecture entitled, ‘Plants as a source of lead molecules in drug discovery’, delivered at Shree S.K. Patel College of Pharmaceutical Sciences and Research, Ganpat University, Ganpat Vidyanagar, Mehsana, in AICTE sponsored two days National seminar on “Recent advances in drug discovery from natural resources” on 29th March 2013.

9. Invited lecture entitled, ‘Design and development of multi-targeted 6,7-dimethoxyquinazoline analogs as dual α1- and AII-receptor antagonists’, delivered at Bombay College of Pharmacy, Kalina, Santacruz, Mumbai on 28th Feb 2013 in AICTE sponsored Faculty development programme on “New facets of medicinal chemistry in drug discovery” during 18th Feb to 2nd March 2013.

10. Invited lecture entitled, ‘Changing paradigm in drug discovery’, delivered at Pharmacy Department, The M.S.University of Baroda, Vadodara in AICTE sponsored two-days National Seminar on “Approached in drug discovery” during 26 – 27 Feb 2013 on 27th Feb 2013

11. Invited lecture entitled, ‘Design and development of multi-targeted 6,7-dimethoxyquinazoline analogs as dual α1- and AII-receptor antagonists’, delivered at Pharmacy Department, The M.S.University of Baroda, Vadodara in AICTE sponsored two-days National Seminar on “Approached in drug discovery” during 26 – 27 Feb 2013 on 26th Feb 2013

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12. Invited lecture entitled, ‘Facing GPAT Examination made easy’, in Continuing Pharmacy Education programme of Indian Pharmacy Association, Vadodara branch on 25th Feb 2013

13. Invited lecture entitled, ‘Design and synthesis of some multi-targeted ligands as anti-hypertensive agents’, delivered at Department of Pharmacy, Sumandeep Vidyapeeth Waghodia Distt, Vadodara, in a Two-days National Seminar on “Pharma Rendezous” during 22 – 23 Feb 2013, on 23rd Feb 2013

14. Invited lecture entitled, ‘LC-MS: A versatile technique for pharmaceutical Analysis’ in one day National seminar on “Advanced in analysis of pharmaceuticals dosage forms by chromatography” sponsored by GUJCOST, organized by Shankarsinh Vaghela Bapu Institute of Pharmacy, Gandhinagar-Mansa Road, Vasan, Gandhinagar on 16th Feb 2013

15. Invited lecture entitled, ‘Alternative methods and techniques in pharmaceutical analysis’ in State level seminar on “Justification for selection of Pharmaceutical analytical techniques” organized by Atmiya Pharmacy College, Ankodiya, Vadodara on 4th Feb 2013

16. Invited lecture entitled, ‘Virtual screening for the discovery of new drugs’ delivered during the training school on ‘Computer aided drug design: Hands on workshop’(from 28 th January to 9th

February 2013) at UGC Networking Resource Center, University Institute of Pharmaceutical Sciences, Panjab University, Chandigarh on 29th Jan 2013

17. Invited lecture entitled, ‘Exploring QSAR for lead optimization’ delivered during the training school on ‘Computer aided drug design: Hands on workshop’(from 28th January to 9th February 2013) at UGC Networking Resource Center, University Institute of Pharmaceutical Sciences, Panjab University, Chandigarh on 28th Jan 2013.

18. Invited lecture entitled, ‘Virtual screening – A versatile tool for new drug discovery process’ in two day CSIR Sponsored workshop on Hands on training on software related to computer aided drug design, at Nirma Institute of Pharmacy, Ahmedabad on 22nd Jan 2013

19. Invited talk entitled, ‘Accreditation- NBA perspective’ on 9th Dec 2012 at 64th Indian Pharmaceutical Congress, SRM University, Chennai, organized by Indian Pharmaceutical Congress Association during 7th to 9th Dec 2012

20. Invited talk entitled, ‘Design and development of steroidal aromatase inhibitors as potential drugs for breast cancer’, on 24th Nov 2012 at International conference on recent advances in pharmaceutical sciences RAPS-2012’ at University College of Pharmaceutical Sciences, Kakatiya University, Warangal-506009, Andhra Pradesh, from 22nd -24th Nov 2012

21. Invited talk entitled, Do we need regulatory bodies for the growth of higher education?’ delivered on 13th Oct 2012 at NAAC sponsored National Level Seminar on ‘Higher education: Excellence towards quality management and assurance’, organized by Anand Pharmacy College, Anand, Gujarat on 12 th

and 13th Oct 201222. Invited talk as mentor scientist entitled, ‘Wonders of Pharmaceutical Analysis’, delivered in the

science camp on 4th Oct 2012 on ‘Innovation in science pursuit for inspired research internship 2012’ from 1st Oct to 6th Oct 2012 at SPP School of Pharmacy & Technology Management, NMIMS, Mumbai

23. Invited talk on ‘NMR Spectroscopy’ under the “CPE Programme” of Indian Pharmaceutical Association, Vadodara Branch on 24th Aug 2012 at Faculty of Technology Auditorium, The M.S.University of Baroda, Vadodara

24. Invited talk on ‘New Steroidal aromatase inhibitors as potential anticancer agents in breast cancer, at Shri Sarvajanik College of Pharmacy, Mehsana, Gujarat on 21st July 2012.

25. Invited lecture on ‘Design and development of site specific chemical delivery systems for anti-arthritic agents’, delivered at Pioneer Pharmacy Degree College, Vadodara, in a One day state level seminar & poster competition on ‘Advances and emerging trends in pharmaceutical Sciences’ on 7th April 2012

26. Invited lecture on ‘Dual α1- and AT-1 inhibitors as potential antihypertensive agents’, delivered at Shri B.M. Shah College of Pharmaceutical Education & Research, Modasa, during GUJCOST sponsored National Seminar on “Pharmaceutical Education: Need of Academia and Industry Harmonization” on March 3, 2012

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27. Invited lecture on ‘Rrelevance of different analytical technique in pharmaceutical analysis – current perspectives’ delivered at Pharmacy Department, The M. S. University of Baroda, under Ms. Kanan Ishwar Mehta Memorial Annual lectures on 27th Sept 2011.

28. Invited lecture on ‘Application of Spectroscopy in Pharmacy Field’ delivered in one day symposium on “Novel technologies to expedite drug discovery and development”, organized by Saraswati Institute of Pharmaceutical Sciences, Gandhinagar on 24th Sept 2011.

29. Invited talk on ‘New Steroidal aromatase inhibitors as potential anticancer agents in breast cancer, at Al-Ameen College of Pharmacy, Bangalore, on 20th Sept 2011

30. Invited talk on ‘Simulation techniques in drug design and development’ at Department of Chemistry, Faculty of Science, The M. S. University of Baroda, Vadodara in a Five day Winter School of Bio-inorganic Chemistry from 8th -12th March 2011, under UGC-CAS Program, on 10th March 2011.

31. Invited talk on ‘Interpretation of NMR spectra and identification of organic compounds by spectroscopy’ at Saraswathi Vidya Bhavan’s College of Pharmacy, Dombivli (E), in two days National workshop on ‘NMR & Co-relation spectroscopy’, on 4th & 5th February 2011.

32. Invited talk on ‘Structural elucidation of organic compounds’ delivered at Sinhgad College of Pharmacy, Pune, under University of Pune sponsored seminar grant, 18th -20th Jan 2011.

33. Invited talk ‘Steroidal aromatase inhibitors as potential drugs for breast carcinoma’ delivered in International conference on Recent Advances in Pharmaceutical sciences- 2010, organized by Department of Pharmaceutics, IT-BHU, Varanasi, 22-23rd Dec 2010.

34. Invited talk on ‘Spectroscopic techniques- Recent developments’, delivered at Ravishankar College of Pharmacy, Bhopal, on 18th Dec 2010.

35. Invited talk on ‘Structure elucidation using spectroscopic techniques’ delivered in National Seminar on ‘Quality assurance issues in drug discovery & formulation development’ at Babaria Institute of Pharmacy, Vadodara, on 3rd - 4th December 2010.

36. Invited talk on ‘New aromatase inhibitors: Steroids as potential therapeutics for breast cancer’, delivered in ‘6th International symposium on Innovations in pharmaceutical sciences and technology’ organized by B. V. Patel Education Trust and B. V. Patel PERD Centre, Ahmedabad, Gujarat from 26-28th Nov 2010.

37. Invited talk on ‘Discovery of some novel TACE inhibitors: A journey through desktop to benchtop’ delivered in ‘International conference on Recent Advances in Drug Discovery’ organized by the University College of Pharmaceutical Sciences, Kakatiya University, Warangal, A.P. from 22nd to 24th Oct 2010.

38. Invited talk on ‘Theoretical principles of NMR Spectroscopy’ delivered at Parul College of Pharmacy, Gujarat, under the SDP on the topic, on 4th Sept 2010.

39. Invited talk on Interpretation of NMR spectra for structure elucidation in "Structural elucidation of organic compounds through spectroscopic data” on 28th and 29th June, 2010 organized by Satara College of Pharmacy, Satara, Maharashtra, 29th June, 2010.

40. Invited talk on ‘QSAR and Molecular Modelling’ in AICTE sponsored Quality Improvement Programme 2010 on ‘Glimpses of current Advances in the Field of Pharmaceutical Sciences’ on June 7th, 2010, organized by Pharmacy Department, The M. S. University of Baroda, Vadodara, 7th to 12th June 2010.

41. Invited talk on ‘Research Methodology in synthetic Medicinal Chemistry’ in AICTE sponsored Quality Improvement Programme 2010 on ‘Glimpses of current Advances in the Field of Pharmaceutical Sciences’ on June 7th, 2010, organized by Pharmacy Department, The M. S. University of Baroda, Vadodara, 7th to 12th June 2010.

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42. Invited talk on ‘Peptidomimetics in Drug Discovery’ at University Institute of Pharmaceutical Sciences, Panjab University, Chandigarh on 1st June 2010 in UGC Networking Resource Centre under the theme of ‘Emerging Trends in Drug Discovery’ and Development from 31st May to 12th June 2010.

43. Invited talk on ‘Indian Patent and PCT Applications’ at The M. S. University of Baroda in UGC sponsored Symposium on ‘Patent awareness and Scientific writing’, 27th March 2009

44. Invited talk delivered on “High Throughput Screening in Drug Discovery” at Poona College of Pharmacy, Pune, Maharashtra under AICTE sponsored staff development programme for Pharmacy teachers on 27th Feb 2009.

45. Invited talk delivered on “CoMFA and CoMSIA techniques in Drug Design and Discovery” at R.C.Patel Institute of Pharmaceutical Education and Research, Shirpur, Maharashtra under AICTE sponsored staff development programme for Pharmacy teachers on 13th Feb 2009.

46. Invited talk entitled, ‘Stereochemistry’ delivered at STE’s Sinhgad College of Pharmacy, Vadgaon, Pune on 10th Feb 2009.

47. Invited lecture delivered on the topic “Spectrophotometric techniques” at Baroda college of Pharmacy, Vadodara on 8th Sept. 2008.

48. Lecture Delivered on “Peptides in Drug Design” in PCI Sponsored State level Orientation Programme for Pharmacy Teachers” held at Shri Sarvajanic Pharmacy College, Mehasana, Gujarat, 1st Feb. 2008.

49. Invited Talk entitled, “Pharmacy Education - Current Scenario and Future Directions”, delivered at Annual Convention of APTI organised by UIPS, Panjab University, Chandigarh, 25th Oct. 2007.

50. Invited Talk on “3D-QSAR and Docking Studies in Drug Design” delivered at National Seminar and Workshop of Pharmacoinformatics organised by PSG College of Pharmacy, Coimbatore, 23rd March 2007.

51. Guest Lecture at Shri Sarvajanic Pharmacy College, Mehsana, on the topic “3D-QSAR and Docking Studies in Drug Design” on 23rd Oct. 2007.

52. Invited Lecture in AICTE Sponsored Two Weeks Staff Development Programme entitled, “3D-QSAR and Docking Studies in Drug Design” organized by S.K. Patel College of Pharmaceutical Education and Research, Ganpat University, Kherva, Mehsana from 13th to 27th April 2007.

53. Invited lecture in AICTE Sponsored Two Weeks Staff Development Programme entitled, “Advances in Characterization of Phytochemical Constituents” organized by S.K. Patel College of Pharmaceutical Education and Research, Ganpat University, Kherva, Mehsana from Jan. 29th to 11th Feb. 2007.

54. Invited Lecture under Continuing Pharmacy Education Programme of Indian Pharmaceutical Association, Vadodara Branch on “Licensing of Intellectual Property Rights” on 14 th Oct. 2006.

55. Invited Lecture in Workshop on “Contemporary Topics in Pharmaceutical Sciences on “Peptidomimetics in Drug Discovery” organized by QIP Centre AICTE and TIFAC Centre of Relevance and Excellence in New Drug Delivery System at Pharmacy Department, The M.S. University of Baroda on 21st June 2006.

56. Invited Lecture entitled “Protease Inhibitors as Potential Drugs” delivered at C.U. Shah College of Pharmacy, SNDT Women’s University, Mumbai on 16th Feb 2006 during their Silver Jubilee Celebrations.

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57. Special Lecture entitled “Designing of Peptidomemetics as Potential Drugs” delivered at Shri Sarvajanic Pharmacy College, Mehsana, Gujarat, during National Pharmacy Week on 26th Oct. 2005.

58. Invited Lecture entitled, “Computer Assisted Drug Design” on a One day Workshop on “Computer Assisted Drug Design” organized by Prin. K.M. Kundanani College of Pharmacy, Mumbai on 15th Oct. 2005.

59. Guest lecture entitled, “Importance of Organic Chemistry in Pharmacy” delivered at S.B. College of Pharmacy, Sivakasi, TN, on the Annual Celebrations on 23rd March 2005.

60. Invited Lecture entitled, “QSAR in Dosage form Designing” delivered at AICTE-ISTE Sponsored Short Term Training Programme Organized by A.R. College of Pharmacy, Vallabh Vidyanagar, from 25th May to 5th June 2004.

61. Invited Lecture entitled, “Radiotracers in in vitro and Preclinical Studies” delivered in 24th

Annual Conference of Indian Association of Biomedical Scientist on the topic Radiotracers in Drug Development, organized by Institute of Nuclear Medicine and Allied Sciences, DRDO, New Delhi on 2nd Nov. 2003.

62. Invited Lecture entitled “Peptide Leads in New Drug Discovery” delivered at UGC Sponsored Refresher Course in Pharmaceutical Sciences on Current Concept in Drug Design and Formulation Development organized by Department of Pharm. Sciences, Guru Jambheshwar University Hisar from Oct. 1st to Oct. 21st 2003.

63. Invited Lecture entitled “Applications of Computers in Drug Discovery” delivered at UGC Sponsored Refresher Course in Pharmaceutical Sciences on Recent Advances in Pharmaceutical Technology and Computer Applications, organized by Department of Pharm. Sciences, Guru Jambheshwar University Hisar from Feb. 20th to March 12th 2003.

64. Invited Lecture entitled “Protease Inhibitors as New Drugs” delivered at UGC Sponsored Refresher Course in Pharmaceutical Sciences on Recent Advances in Pharmaceutical Technology and Computer Applications organized by Department of Pharm. Sciences, Guru Jambheshwar University, Hisar from Feb. 20th to March 12th 2003.

65. Invited Lecture entitled “Drug Discovery- In Retrospect” delivered at UGC Sponsored Refresher Course in Pharmaceutical Sciences organized by Department of Pharm. Sciences, Guru Jambheshwar University Hisar from Jan 30th to Feb.19th 2002.

66. Invited Lecture entitled “Molecular Modelling and Drug Designing” delivered at UGC Sponsored Refresher Course in Pharmaceutical Sciences organized by Department of Pharm. Sciences, Guru Jambheshwar University Hisar from Jan 30th to Feb.19th 2002.

67. Invited Lecture entitled “Computers and Drug Discovery” delivered at AICTE-ISTE Sponsored Short Term Training programme on Pharm. Sciences in the New Millennium- Emerging Trends & Challenges Ahead, organized by A.R. College of Pharmacy, Vallabh Vidyanagar, from 30th April 2001 to 12th May 2001.

68. Invited Lecture entitled “Basic Test for Common Medicines”, WHO Sponsored Professional Training Programme organized by Pharmacy Department, The M.S. University of Baroda on 23rd April 2001.

69. Invited Lecture delivered in AICTE Sponsored Short Term Training Programme organized by ISTE at Department of Pharm. Sciences, from 28th Feb. to 12th March 2000.

70. Invited Lecture delivered AICTE and ISTE Sponsored Short Term Training Programme on Recent Developments in Pharm. Sciences organized by A.R. College of Pharmacy, Vallabh Vidyanagar from 26th Oct. to 7th Nov. 1998.

12

71. Invited Lecture in ISTE Summer School on Trends in Development of Drugs and Delivery Systems-A Futuristic Approach organized by Pharmacy Department, The M.S. University of Baroda, Vadodara from 19th to 31st March 1997.

SCIENTIFIC PUBLICATIONSResearch Papers : 95Reviews : 22Book Chapters : 04 Patents : 16

List of Research Articles:

Sr. No.

Title of the Paper Author(s) Name of Journal, Vol. & Page No.

Year

1. Exploring Cytotoxic Potential of Some Novel 6,7-Dimethoxyquinazolines

M. R. Yadav, B. S. Chauhan, P. P. Naik and R. Giridhar

Eur. J. Med. Chem Communicated

2. Synthesis and SAR of substituted 3-benzazepines as potent and selective 5-HT2C receptor agonists

A.Verma, A.Sinha, N. Prajapati, R.Giridhar and M.R.Yadav

Curr. Med. Chem. Communicated

3. An HPTLC method for quantification of cholesteryl esters from human plasma and rat liver microsomes

Hardik Gandhi, Palash Pal, Rajani Giridhar, M.R.Yadav

Biomedical Chromatography.

In Press

4. Molecular Modeling Studies of Some Triazine Derivatives as G-quadruplex binders for inhibition of telomerase enzyme

Vishal P Zambre, Rajani Giridhar and Mange Ram Yadav

Med. Chem. Res., 22, 4685-4699

2013

5. Synthesis of novel 4,6-diaryl-aminopyrimidines as potential antiplasmodial agents

R. Giridhar, R.S. Tamboli, D.G.Prajapati, S. Soni, S. Gupta and M.R.Yadav

Med. Chem. Res., 2013

6. Design and synthesis of 6,7-dimethoxyquinazoline analogs as multi-targeted ligands for <alpha>1- and AII-receptors antagonism

P. Naik, H. Gandhi, B.S. Chauhan, R. Giridhar, M.R.Yadav

Bio-org. Med. Chem. Lett., 23, 3959-3966

2013

7. Microwave Assisted Palladium Catalyzed Intermolecular α-Arylation of Copper-Amide

Amit Verma, N. Prajapati,S. Salecha,R. Giridhar, M.R. Yadav

Tet. Lett., 54, 2029 - 2032

2013

13

Enolate.of Benzazepine8. Novel 2-aminobenzamides as

potential orally active antithrombotic agents

Verma, Amit; Giridhar, Rajani; Modh, Pratik; Yadav, Mange Ram

Med. Chem. Lett., 4, 32-36

2013

9. Pyrido[1,2-a]pyrimidin-4-ones as potential plasmodial falcipain-2 inhibitors

M. R. Yadav, U. R. Mane, R. Giridhar, H. Li, J. Huang, R. C. Gupta, S. S. Nadkani, C. Dutt, V. Chouthaiwale and P. P. Naik

Bio-org. Med. Chem. 20, 6296 - 6304

2012

10. A facile IL-DMSO assisted synthesis of benzo annelated five-, six- and seven- membered heterocycles

Amit Verma, R.Giridhar and M. R. Yadav

Tet. Lett., 53, 2954 -2958

2012

11. Assessment of antiplatelet activity of 2-aminopyrimidines

Rajani Giridhar, Riyaj S. Tamboli, R. Ramajayam, Dhaval G. Prajapati and M.R.Yadav

Eur. J. Med. Chem., 50, 428-432

2012

12. Steroidal carbonitriles as Potential aromatase inhibitor

Mange Ram Yadav, Prafulla M. Sabale, Rajani Giridhar, Christina Zimmer and Rolf W. Hartmann

Steroids, 77, 850 - 857

2012

13. Cytotoxic potential of novel 6,7-dimethoxyquinazolines

M. R. Yadav, Fedora Grande ; Bishram S Chouhan ; Prashant P Naik ; Rajani Giridhar ; Antonio Garofalo; Nouri Neamati

Eur. J. Med. Chem., 48, 231 -247

2012

14. Revelation on the potency of α1-blockers – Parallel blockade of Angiotensin II receptor: A new finding

M. R. Yadav, H. P. Gandhi, P. P. Naik and R. Giridhar

Pharm. Biol., 50, 439 -442

2012

15. Improved percutaneous delivery of some NSAIDs for the treatment of arthritis

R. Thosani, V. Pawar, R. Giridhar and M.R.Yadav

J. Pharm. Bioallied Sciences, 4(S), S12-3

2012

16. Cartilage tartgeted chemical delivery of naproxen and ibuprofen for the treatment of arthritis

V.Pawar, V. Gohil, R.Tamboli, R.Giridhar and M.R.Yadav

J. Pharm. Bioallied Sciences, 4(S), S10-1

2012

17. Synthesis, preliminary biological evaluation and molecular modeling of some new heterocyclic inhibitors of TACE

P. Sengupta, C. S. Puri, H. A. Chokshi, C. K. Sheth,A. S. Midha, T. Rao C., Rajamannar T., P. R. Murumkar and M.R. Yadav

Eur. J. Med. Chem., 46, 5549-55

2011

14

18. Synthesis and Preliminary Screening of Novel A- and D-Ring Modified Steroids as Aromatase Inhibitors

M. R. Yadav, Prafulla M. Sabale, Rajani Giridhar, Dharmendra Baria, Christina Zimmer and Rolf W. Hartmann

Let. Drug Des. Dis., 8,

2011

19. Determining of Structural Requirements of Influenza Neuraminidase Type A Inhibitors and Binding Interaction Analysis with the Active Site of A/H1N1 by 3D-QSAR CoMFA and CoMSIA Modeling

Murumkar P. , Le Ly, Truong Thanh and M.R.Yadav

Med. Chem. Commun., 2, 710-719

2011

20. Synthesis of Some Novel Androstanes as Potential Aromatase Inhibitors

M. R. Yadav, P. M. Sabale, R. Giridhar,C. Zimmer and R. W. Hartmann

Steroids, 76, 464-70

2011

21. 3D-QSAR studies of 4-quinolone derivatives as high-affinity ligands at the benzodiazepine site of brain GABAA receptors

A. Gaurav, M.R.Yadav, R. Giridhar, V. Gautam, R. Singh

Medicinal Chemistry Research, 20, 192-97 2011

22. Development of highly predictive 3D-QSAR CoMSIA models for anthraquinone and acridone derivatives as telomerase inhibitors which target G-quadruplex DNA telomere

V.P. Zambre, P.R. Murumkar, R. Giridhar, M. R. Yadav

Journal of Molecular Graphics and Modelling, 29, 229-239

2010

23. Development of predictive pharmacophore model for in silico screening, and 3D QSAR CoMFA and CoMSIA studies for lead optimization, for designing of potent tumor necrosis factor alpha converting enzyme inhibitors

Murumkar, P.R., Zambre, V.P., Yadav, M.R.

Journal of Computer-Aided Molecular Design 24 (2), pp. 143-156 2010

24. Synthesis and anti-HIV-1 integrase activitiy of cyano pyrimidinones

Ramajayam, R., Mahera, N.B., Neamati, N., Yadav, M.R., Giridhar, R.

Archiv der Pharmazie 342 (12), 710-715

2009

25. QSAR studies on 4-quinolone derivatives as high-affinity ligands at the benzodiazepine site of brain GABAA receptors

Gaurav, A., Yadav, M.R., Giridhar, R., Gautam, V., Singh, R.

Medicinal Chemistry 5 (4), 353-358 2009

15

26. Metalloantibiotics: synthesis, characterization and antimicrobial evaluation of bismuth-fluoroquinolone antibiotic complexes against Helicobacter pylori

Anwar Shaikh, Rajani Giridhar, Francis Mgraud and M.R.Yadav

Acta Pharm. 59 (3), pp. 259-271

2009

27. Studies on novel 2-imidazolidinones and tetrahydropyrimidin-2(1H)-ones as potential TACE inhibitors: Design, synthesis, molecular modeling, and preliminary biological evaluation

Shirshendu DasGupta, Prashant R Murumkar, Rajani Giridhar and M. R. Yadav

Bio-org. Med. Chem., 17, 3604-17

2009

28. Structural investigation of acridine derivatives by CoMFA and CoMSIA reveals novel insight towards DNA G-quadruplex mediated telomerase inhibition and offer a highly predictive 3D-model for substituted acridines

Vishal P Zambre, Prashant R Murumkar, Rajani Giridhar and M. R. Yadav

J. Chem. Info. Mod. 49,5, 1298-1311

2009

29. Design, synthesis and preliminary screening of some new conformationally constrained Falcipain-2 inhibitors as potential antimalerial agents

A. K. Shinde, B. S. Chauhan, S. D. Gupta, R. Giridhar, P. Rosenthal, J. Gut and M.R.Yadav

Letters in Drug Design & Discovery, 6 (4), 258-267

2009

30. Development of predictive 3D-QSAR CoMFA and CoMSIA Models for β-Aminohydroxamic Acid-Derived Tumor Necrosis-α Converting Enzyme Inhibitors

Prashant R. Murumkar, Vishal P. Zambre, Rajani Giridhar and M. R. Yadav

Chem. Biol. Drug Des., 73, 97-107

2009

31. Synthesis, antileukemic and antiplatelet activities of 2,3-diaryl-6,7-dihydro-5H-1,4-diazepines

R.Ramajayam, R.Giridhar, M.R.Yadav, R.Balraman, H.Djaballah, D.Shum and C.Rady

Eu. J. Med. Chem., 43, 2004-2010

2008

32. Site specific chemical delivery of NSAIDs to inflamed joints: Synthesis, biological activity and γ-imaging studies of quaternary ammonium salts of tropinol esters of some NSAIDs

M.R. Yadav, Vijay Pawar, P.K. Halen, R. Giridhar

Bio-org. Med. Chem., 16(21) 9443-9449

2008

16

33. Peptidomimetics 2-Cyanopyrrolidine as Potential Selective Cathepsin L Inhibitors

M.R.Yadav, A.K. Shinde, B.S. Chauhan, R. Giridhar, Robert Menard

J. Enz. Inh. Med. Chem., 23(2), 190-197

2008

34. 3D-Quantitative Structure-Activity Relationship Studies on Benzothiadiazapine Hydroxamates as Inhibitors of Tumor Necrosis Factor-α Converting Enzyme

Prashant R. Murumkar, R.Giridhar and Mange Ram Yadav


2008

35. Studies on crystal forms of Pefloxacine: Preparation, Characterization and Dissolution Profile

M.R.Yadav, Anwar Shaikh, V. Ganesan, Rajani Giridhar, Renu C.

J. Pharm. Sci., 2637-2648

2008

36. Synthesis antiproliferative activity of some diaryldiazepines and diarylpyrimidines

R. Ramajayam, R. Giridhar, M.R.Yadav, H.Djaballah, D.Shun and C.Radu

J. Enz. Inhib. Med. Chem., 22(6), 716-721

2007

37. Combining antocholinergic and anti-inflammatory activities into a single moiety: A novel approach to reduce gastrointestinal toxicity of ibuprofen and ketoprofen

P.K Halen, K.K. Chagti, R.Giridhar, M.R.Yadav


2007

38. Substituted aminoalcohol ester analogs of indomethacin with reduced toxic effects

P.K Halen, K.K. Chagti, R.Giridhar, M.R.Yadav

Med. Chem. Res., 16, 101-111

2007

39. Insights into the structural requirements of farnesyltransferase inhibitors as potential anti-tumor agents based on 3D QSAR CoMFA and CoMSIA models

D. S. Puntambekar, R. Giridhar, M. R. Yadav

Eur. J. Med. Chem., 41 (11) 1279-1292

2007

40. Bismuth -norfloxacin complex: Synthesis, physicochemical and antimicrobial evaluation

A.R. Shaikh, R. Giridhar, M.R. Yadav

Int. J. Pharmaceutics, 332 , 24–30

2007

41. Studies in 3,4-diaryl-1,2,5-oxadiazoles and their N-oxides: Search for better COX-2 inhibitors

M. R.Yadav, S.T. Shirude, D. S. Puntambekar, P.J. Patel, H.B. Prajapati, A. Parmar R. Balaraman, R. Giridhar

Acta Pharm. 57, 13–30

2007

17

42. Synthesis and Evaluation of some Gastrointestinal sparing anti-inflammatory amino ethyl ester derivatives and naphthalene-based NSAIDs

P.K.Halen, Manisha Rawal, K.K. Chagti, R. Giridhar, M.R. Yadav

Arch. Pharm. Chem. LifeSci.340, 88-94

2007

43. Synthesis and Pharmacological Investigation of Novel 1-Alkyl-4-(4-substituted aryl/heteroaryl)-1,2,4-triazolo[4,3-a]quinazolin-5(4H)-ones as a New Class of H1-Antihistaminic Agents

V.Alagarsamy, M.R.Yadav and R. Giridhar

Arznein.-Forsch., 56 (12), 834-841 2006

44. Synthesis of new chemical entities from paracetamol and NSAIDs with improved pharmacodynamics profile

P.K.Halen, S.T. Shirode, R. Giridhar, M.R. Yadav

Biorg. & Med. Chem., 14, 8701-8706

2006

45. Anti-HIV, Antibacterial, Antifungal activities of some novel 1, 4-disubstituted 1,2,4-triazolo[4,3-a] Quinazolin-5(4H)-ones

V. Alagarsamy, R. Giridhar, M. R.Yadav, R. Revathi, E. deCercq, K. Rukmani

Indian J. Pharm. Sci., 68, 532-535

2006

46. Synthesis of new chemical entities from paracetamol and NSAIDS with improved pharmacodynamic profile

M.R.Yadav, D.M. Brahamkshatriya, S.T. Shirude, A. Parmar, R. Balaraman and R. Giridhar

Biorg. Med. Chem., 14, 8701-8706

2006

47. Synthesis and pharmacological evaluation of some dual acting aminoalcohol esters derivatives of flubiprofen and biphenyl acetic acid

P.K. Halen, M. R. Yadav, K.K Chagti, and R. Giridhar

Chem. Biodiv., 3, 1238-1248

2006

48. Synthesis and Anti-Inflammatory activity of 2,3-Diaryl-4-(3H)quinazolinones

M.R.Yadav, S.T. Shirude, A. Parmar, R. Balaraman and R. Giridhar

Khim. Geterotsikl. Soedin., 42, 1198-1205

2006

49. Understanding the Antitumor activity of tricyclicpiperazinyl derivatives as farnesyltransferase inhibitors using CoMFA and CoMSIA

D.S. Puntambekar, R. Giridhar and M.R.Yadav

Eur. J. Med. Chem., 41, 1279–1292

2006

18

50. Synthesis of Novel substituted diaryl 1,4-Diazepines

R.Ramajayam, R. Giridhar and M.R.Yadav

Chemistry of Heterocyclic Compounds, 42 (7), 901-906

2006

51. An efficient and time saving microwave-assisted selenium dioxide oxidation of 1,2-diarylethanones

S.T. Shirude, P. Patel, R. Giridhar and M.R.Yadav

Indian J. Chem., 45B, 1080-1085

2006

52. 3D-QSAR studies of farnesyl transferase inhibitors: A comparative molecular field analysis study

D.S. Puntambekar, R. Giridhar and M.R. Yadav

Biorg. Med. Chem. Lett. 16, 1821-1827

2006

53. 3D QSAR CoMFA/CoMSIA studies on 5-aryl-2,2-dialkyl-4-phenyl-3H)furanone derivatives as selective COX-II inhibitors

D.S. Puntambekar, R. Giridhar and M.R. Yadav

Acta Pharm. 56, 157 2006

54. Synthesis and evaluation of dual acting esters of aspirin and ketorolac

P.K. Halen, M.R. Yadav, K.K Chagti, C.S. Reshmi,R. Giridhar

Ars. Pharm., 47, 61-79

2006

55. Synthesis and pharmacological investigation of novel 1-substituted 4-(methoxyphenyl)-1,2,4-triazolo[4,3-a] Quinazolin-5(4H)-ones as a new class of H1-antihisttaminic agents

V Alagarsamy , R. Giridhar, M.R. Yadav

J Pharm. Pharmacol., 58, 1249- 1255

2006

56. Identification of novel non-Nucleoside reverse transcriptase inhibitors using fragment-based lead generation

R .Ramajayam, R. Giridhar, M.R.Yadav, E. deClercq, C. Pannecouque and G.P. Dhaval

Med. Chem. Res, 14, 475-487

2005

57. QSAR studies of diarylimidazoles as selective COX-2 inhibitors

M.R.Yadav, D.S.Puntambekar, K.P.Sarathy, S. Vengurlekar, R. Giridhar

Indian J. Chem., 45B, 475-482

2005

58. A novel approach towards therapeutic optimization of diclofenac

M.R.Yadav, P.Halen, K. Chagti, B. Hemalatha R.Giridhar

ARS Pharma., 46, 263-267

2005

59. Synthesis and pharmacological V. Alagarsamy, R. Giridhar, Bioorganic Med. 2005

19

investigation of novel 1-substituted-4-phenyl-1,2,4-triazolo[4,3-a]quinazolin-5(4H)-ones as a new class of H1-antihistaminic agents

M.R.Yadav Chem. Lett., 15, 1877-1880

60. Effect of bis[Curcumino] oxovanadium complex on non-diabetic and Streptozotocin-induced Diabetic Rats

J.B.Majithia, R.Balaraman, R. Giridhar, M.R.Yadav

J.Trace Elem. Med. Biol., 18, 211-217

2005

61. Synthesis and H1-antihistaminic activity of some novel 1-substituted-4-(3-methylphenyl)-1,2,4-triazolo [4,3-a]quinazolin-5(4H)-ones.

Alagarsamy V, Giridhar R, Yadav M.R.

Biol. Pharm. Bull., 28 (8), 1531-34

2005

62. Studies on the Development of Taste Masked Suspension of Chloroquine

V.Chandibhamar, M.R.Yadav and R.S.R. Murthy

Bull. Chim. Farmac., 143, 377-382

2004

63. Synthesis of 3-Oxo-4-aza-5-System from (25R)-3-oxo-A-norspristone

M.R.Yadav, M.M.Ganesh, R.Giridhar, M.Kumar

Asian J. Chem., 16(2), 1027-1033

2004

64. QSAR Study by Fujita-Ban of Some Substituted α,β-Diaryl Five Membered Heterocyclic as COX-1/COX-2 Inhibitors

K.P.Sarathy, R.Giridhar and M.R.Yadav

Indian Drugs, 40(1), 9-18

2003

65. New Azasteroidal Neuromuscular Blocking Agent Possessing Acetylcholine-like Moiety in Ring A

M.R.Yadav, R.Giridhar, S.P.Rathod, M.Mahatma and P.M.Sabale

Indian J. Chem., 40B, 1177-1185

2001

66. Crystal Forms of Nimesulide-A Sulfonanilide(NSAID)

A.Kapoor, D.K.Majumdar and M.R.Yadav


1998

67. Phosphite Deoxygenation of Steroidal[3,4-c] and [16,17-c] furazan N-oxides

D.P.Jindal, R.Gupta, I.B.Singh, J.S.R.A.Sharma and M.R.Yadav


1997

68. Chemical and Pharmacological Studies on Fixed Oil of Ocimum sanctum

S.Singh, D.K.Majumdar and M.R.Yadav

Indian J. Exp. Biol.,34, 1212-1215

1996

69. Synthesis of some Novel Hetrocyclic Steroids by Beckmann Rearrangement

D.P.Jindal, R.Gupta, R.Kaushal, I.B.Singh and M.R.Yadav


1996

70. Naproxen-L-Phenylalanine alkyl ester prodrugs: Synthesis

V.K.Sharma, M.R.Yadav and S.Singh

Inflamm. Res.,44, S287-S287

1995

20

http://www.ncbi.nlm.nih.gov/pubmed?term=Yadav%20MR%5BAuthor%5D&cauthor=true&cauthor_uid=16079509

http://www.ncbi.nlm.nih.gov/pubmed?term=Giridhar%20R%5BAuthor%5D&cauthor=true&cauthor_uid=16079509

http://www.ncbi.nlm.nih.gov/pubmed?term=Giridhar%20R%5BAuthor%5D&cauthor=true&cauthor_uid=16079509

http://www.ncbi.nlm.nih.gov/pubmed?term=Alagarsamy%20V%5BAuthor%5D&cauthor=true&cauthor_uid=16079509

and Biological Evaluation71. Synthesis and Biological

Activity of [16,17-c]furaxano-5α/β-androstano[3,4-c]furazans

D.P.Jindal, R.Gupta, I.B.Singh, N.Sharma and M.R.Yadav


1995

72. Synthesis and Biological Activity of Steroidal[3,4-d]triazoles

A.K.Verma, R.Gupta, M.R.Yadav and D.P.Jindal


1995

73. Wolf-Kishner reduction Studies on Steroidal hydrazoneoximes

A.K.Verma, N.Sharma, M.R.Yadav D.P.Jindal

J. Indian Chem. Soc.,71, 283-284

1994

74. Studies in Synthesis of Some Potential Neuromuscular Blocking Azasteroids

M.R.Yadav Indian J. Chem., 32B, 746-753

1993

75. Studies in 17a-Azasteroidal[3,2-c]furoxans

D.P. Jindal, J. Abraham and M.R. Yadav


1992

76. 17-methyl-3β-pyrrilidino-17-aza-D-homo-5-androstene dimethiodide

M.R.Yadav Indian J. Chem., 31B, 1-2

1992

77. Certain Steroidal[3,4-c]-1’,2’,5’ oxadiazoles

M.R.Yadav and D.P.Jindal Indian J. Chem., 30B, 473-476

1991

78. 5 α-Androstano[3,4-c][16,17-c]bisfuroxan

D.P.Jindal and M.R.Yadav Indian J. Chem., 30B, 515-516

1991

79. Hetroaromatic-ring fused steroids

M.R.Yadav and D.P.Jindal Indian J. Pharm. Sci., 52, 42-42

1990

80. Synthesis and Study of Azatriterpenes

M.S.Y.Khan, S.Ahmed, M.R.Yadav and D.P.Jindal

J. Indian Chem. Soc.,67, 330-331

1990

81. Novel Camphorimideoximes and Camphorquinone dioxime

V.K.Kapoor, K.K.Chagti, M.R.Yadav and D.P.Jindal


1990

82. Studies in Steroidal[3,4-c]-1’,2’,5’ oxadiazoles

M.R.Yadav, J.Abraham and D.P.Jindal


1990

83. Synthesis and Study of Heterocyclic Oxadiazoles

D.P.Jindal, I.B.Singh and M.R.Yadav


1989

84. 5-Pregneno[3,4-c]-1’,2’,5’ oxadiazoles

M.R.Yadav, D.P.Jindal and H.Singh


1988

85. 2’-Phenyl;-5 α-pregnano[3,4-c]-1’,2’,5’-triazole-20-one

D.P.Jindal, N.Sharma and M.R.Yadav


1987

86. Synthesis and Anti-inflammatory Activity of Some Camphor Analogues

V.K.Kapoor, K.K.Chagti, M.R.Yadav and D.P.Jindal


1987

21

87. 17-Oxo-17a-aza-D-homo-5 α-androstano[3,4-c]-1’,2’,5’ oxadiazole N-oxide

D.P.Jindal, J.Abraham and M.R.Yadav


1987

88. Pregneno[3,4-c]-1’,2’,5’ oxadiazol-20-ones

D.P.Jindal, M.R.Yadav, R.K.Sharma,V.R.Agrawal and H.Singh


1987

89. 17α-preg-20-yno[3,4-c]-1’,2’,5’ oxadiazol-17-ols

H.Singh, M.R.Yadav and D.P.Jindal


1987

90. Steroidal 5-eno[3,4-c]-1’,2’,5’ oxadiazoles

D. Paul, M.R.Yadav and H.Singh

Inian J. Pharm. Sci., 48, 108-108

1986

91. 5-Pregnenol[3,4-c]-1’,2’,5’ oxadiazoles

H.Singh, D. Paul, M.R.Yadav R.K.Sharma and V.R.Agrawal

Inian J. Pharm. Sci., 47, 55-55

1985

92. Substituted thiocarbonimidic diamide Derivatives and Their Antihistaminic properties

S.N.Pandya, M.R.Yadav and K.Gupta

Eastern Phamacist,28, 211-212

1985

93. 17 Hydroxy-5ξ,17α-preg-20-yno[3,4-c]-1’,2’,5’ oxadiazoles

H.Singh, M.R.Yadav and D. Paul


1985

94. Steroidal [3,4-c]-1’,2’,5’ oxadiazoles

H.Singh, M.R.Yadav, S.P.Garg, R.K.Sharma and D. Paul

Heterocycles,23, 2929-2938

1985

95. 5ξ-Pregnanol[3,4-c]-1’,2’,5’ oxadiazoles

D. Paul, M.R.Yadav, R.K.Sharma, V.R.Agrawal and H.Singh

Indian J. Chem, 24B, 1-1

1985

List of Reviews:

Sr. No. Title of the Review Author(s)Name of Journal, Vol.

& Page No.Year

1.

Management of Hypertension – Journey from Single Drug Therapy to Multitargeted Ligand Therapy: A Clinical Overview

Prashant P. Naik. Vijay A. Pawar, Rajani Giridhar, Mange Ram Yadav

Current Clinical Pharmacology

In Press

2. Nitrogen containing privileged structures and their solid phase combinatorial synthesis

Amit Verma, M.R.Yadav, Rajani Giridhar, Navnit

Combi. Chem. High Thrpt. Screen., 16,

2013

22

Prajapati, Avinash C. Tripathi and Shailendra K. Saraf

3.

Falcipain-2 inhibitors as potential therapeutics for resistant strains of malaria: a patent review

Uttam Mane and M.R.Yadav

Expert Opinion on Therapeutic Patents In Press

4.

Novel methods and strategies in the discovery of TACE Inhibitors

Prashant Murumkar, R. Giridhar and M.R.Yadav

Expert Opinion on Drug Discovery, In Press

5.

ACAT Inhibitors: The Search for Novel Cholesterol Lowering Agents

Palash Pal, Hardik Gandhi, Rajani Giridhar and Mange Ram Yadav

Mini-Reviews in Med. Chem., 13, 1195-1219

2013

6.

Novel TACE inhibitors in drug discovery: A review of patented compounds

Murumkar, P.R., DasGupta, S., Chandani, S.R., Giridhar, R. M.R. Yadav

Expert Opinion on Therapeutic Patents 20 (1), pp. 31-57 2010

7.

Gemini Amphiphiles: A Novel Class ofNonviral Gene Delivery Vectors

Mukesh Kumar, Kaustub Jinturkar, M.R. Yadav,& A.N. Misra

Critical Reviews™ in Therapeutic Drug Carrier Systems, 27(3), 237-278

2010

8.

Angiotensin II Receptor Type 1 (AT1) Selective Nonpeptidic Antagonists - A Perspective

Prashant Naik, Prashant Murumkar, Rajani Giridhar and M. R. Yadav

Bioorganic and Medicinal Chemistry, 18, pp. 8418-56.

2010

9.

Prodrug Designing of NSAIDS

P.K. Halen, P.R. Murumkar, R. Giridhar and M. R. Yadav

Mini-Reviews in Med. Chem., (9), 124-139

2009

10.

Current perspective of TACE inhibitors: A review

DasGupta, S Murumkar, P. R., Giridhar, R., M.R. Yadav

Bioorganic and Medicinal Chemistry Chem. (17) 444-459

2009

11.The search for potent, small molecule NNRTIs: A review

Prajapati, D.G., Ramajayam, R., M.R. Yadav, Giridhar, R.

Bioorganic and Medicinal Chemistry 17 (16), pp. 5744-5762

2009

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12.

Recent Advances in Selective α1-Adrenoreceptor Antagonists as Antihypertensive Agents

K. S. Jain, J. B Bariwal, M. Kathiravan, M. S Phoujdar,R. S Sahne, B. S Chauhan, A. K Shah, M. R. Yadav

Bio-org. Med. Chem., (16) 4759-4800

2008

13.

Inhibition of farnesyltransferase: A rational approach to treat cancer?

D.S. Puntambekar, R.Giridhar, M.R. Yadav

J. Enz. Inh. Med. Chem.,22, 127-40 2007

14.

Current Scenario of 1,4-Diazepines as potent biomolecules- A mini review

R .Ramajayam, R. Giridhar, M.R.Yadav

Mini-Reviews in Med. Chem., 7 (8) 793-812 2007

15.Protease Inhibitors as Potential Drugs

M.R.YadavChronicle Pharmabiz, March 21, 65-68

2006

16.Intellectual Property- Related Issues

M.R.YadavPharma Glimpses, 15-17

2006

17.

The Multifaceted Profile of Cox-2 Enzyme and Emerging Therapeutic Uses of Cox-2 Inhibitors

Hetal B. Prajapati, R. Giridhar and M.R.Yadav

Indian J. Pharm. Sci. 65, 557-564

2003

18.Some Interesting Facets of Chiral Drugs

Halen P.K., Giridhar R. and Yadav M.R

Indian Drugs, 39, 457-464

2002

19.Industry- Academy Interaction- Need of the Hour

Mange Ram YadavAssoc. Pharm. Technocrt., 73-74 1994

20.RU-486: A Multifaceted Antihormonal Drug

Mange Ram Yadav and Manoj Kumar

Indian Drugs, 29, 387-394

1992

21.Antimicrobial Agents in Pharmaceutical Products

Dharam Paul Jindal and Mange Ram Yadav

Eastern Pharmacist, 29, 47-60 1986

22.Role of Antioxidants in Pharmaceutical Products

Dharam Paul Jindal and Mange Ram Yadav

Indian Drugs, 22, 1-17 1985

Patents:

Sr. No.

Title of the Patent Author(s)Registration/Application No., Year

24

1.

Gemini amphiphile based formulations and their method of preparation for polynucleotide delivery

Yadav M.R., Kumar M. and Misra A.N.

Indian patent, Appl./1828/MUM/2013

2.

Benzimidazolyl, benzoxazolyl and 2-pyridylimidazolyl derivatives as potential anticancer agents and the process for their preparation

Yadav M.R., Srinivasan B.P., Yogishkumar H. and Pawar V.A.

Indian patent, Appl./192/MUM/2013

3.

Piperazinylalkyl esters and the salts of some NSAIDs for improved percutaneous delivery and the process for their preparation

Yadav M.R. and Pawar V.A.

Indian patent, Appl.//MUM/2012

4.

Quaternary ammonium 8-methyl-8azabicyclo[3.2.1]octan-3-yl esters as muscarinic receptor antagonists and their method of preparation

Yadav M.R. Pawar V.A. and Huchanna Y.K.

Indian patent, Appl.//MUM/2012

5.

4-Amino-2-piperazinoquinazoline derivatives as potential antihypertensive agents and their method of preparation

M.R.Yadav, P.R.Naik and R.Giridhar

Indian Patent, Appl./253/MUM/2012

6.

2-Substituted 4-amino-6,7-dimethoxyquinazolines as dual acting antihypertensive agents and the process for their preparation

M.R.Yadav, R.Giridhar and Prashant P. Naik

Indian Patent,Appl./3412/MUM/2011

7.Benzazepine derivatives and the process for their preparation

R. Giridhar, M.R.Yadav and A. Verma

Indian Patent, Appl./3480/MUM/2010

8.

4-(Arylthia)-16 –cyano-17-oxo-4-androsten-3-ones, reduced derivatives 17–ols and the process for their preparation

M.R.Yadav, P.M. Sabale, P.R.Murumkar and R.Giridhar

Indian patent,Appl./ 3309/Mum/2010

9.Some polar diquaternary Gemini amphiphiles and the process for their preparation

M.R.Yadav, M. Kumar and A.N.Misra


10.

1-Aryl-2-imidazolidinones as potential TACE Inhibitors and the process for their preparation

M.R.Yadav,Shirshendu DasGupta and R.Giridhar


11. Trisciprofloxacinatobismuth and the Process for its Preparation

M.R.Yadav, Anwar R. Shaikh

Indian Patent,Appl./1449/Mum/2007

25

and R. Giridhar

12.

A Process for the preparation of 3-[o-m-p Mono/Disubbstituted phenyl]-4-[o/p-substituted phenyl] Furazans and Furoxans’.

M.R.Yadav, R.Giridhar and Hetal B. Prajapati


13.A Process for the Preparation of Biscurcumino-oxvanadium(iv)

M.R.Yadav, R.Balaraman and R.Giridhar


14.

A Process for the Preparation of 17α-Methyl-4-oxo-5α-androstano[2,3-d]pyrazol-17-ol

D.P.Jindal and M.R.Yadav

Indian Patent,Appl.1041/Del/94, Chem.Abstr.,124,1996,9095W

15.A process for the Preparation of 4,17β-Dihydroxy-3-oxo-4-androstene-2ξ-carbonitrile17-acetate


Indian Patent,Appl.1041/Del/88

16.A Process for the Preparation of 17α-Methyl-4-androstano[3,2-c]isoxazol-4,17-diol


Indian Patent,166480,1986, Appl.999/Del/86

BOOK/ BOOK CHAPTER1. Mange Ram Yadav, Prashant R. Murumkar and Vishal Zambre, “Advances in Studies on

Collagenase Inhibitors”, Advances in Studies on Matrix Metalloproteinase Inhibitors (Springer Basel AG), Experientia Supplementum Volume 103, 2012, pp 83-135.

2. Mange Ram Yadav, Shirshendu Das Gupta, Prashant R. Murumkar and Rajani Giridhar, “Small Molecule Selective TACE Inhibitors: Potential Therapeutic Agents”, NOVA international publication, Volume 3, USA, 2010,

3. Kanchan Kohli and Mange Ram Yadav, Pharmaceutical Chemistry-II, Piyush Publications, Delhi, 1995.

4. Harkishan Singh, Dharam Paul Jindal, Mange Ram Yadav and Manoj Kumar, “Heterosteroids in Drug Research” in Progress in Medicinal Chemistry, G.P. Ellis and G.B. West, Eds., Elsevier/ North-Holland Biomedical Press, Amsterdam, Vol. 28, 1991.

SCIENTIFIC PAPER PRESENTATIONSInternational Presentations:

1. Vishal P Zambre, Prashant R. Murumkar, Rajani Giridhar and Mange Ram Yadav DNA G-quadruplex ligands – anthraquinones and acridones: 3D - QSAR studies for a quantitative prediction of the telomerase inhibitory activity based on comparative molecular similarity indices analysis, 239th ACS Annual National Meeting, 2009 San Francisco, CA, USA.

2. Vishal P Zambre, Prashant Murumkar, Rajani Giridhar and Mange Ram Yadav, “3DQSAR studies on DNA G-quadruplex interactive agents as telomerase inhibitors” 17th European

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Symposium on QSAR in “Omics” and Systems Biology during 21-26 Sept. 2008 at Uppsala, Sweden.

3. Prashant R. Murumkar, Rajani Giridhar and Mange Ram Yadav Identification of ligand feature essential for TACE inhibitors by pharmacophore modeling. 237th ACS Annual National Meeting, 2009, Salt lake City, Utah, USA.

4. Vishal P Zambre Prashant R. Murumkar, Rajani Giridhar and Mange Ram Yadav, Ligand-based molecular modeling study on DNA G-quadruplex mediated telomerase inhibitors: A 3D-QSAR CoMFA, CoMSIA approach. 237th ACS Annual National Meeting, 2009, Salt lake City, Utah, USA.

5. Prashant R. Murumkar, Rajani Giridhar and Mange Ram Yadav 3D-QSAR studies on Benzodiazepine Hydroxamates as Tumor Necrosis Factor- alpha Converting Enzyme Inhibitors, 235th ACS Annual National Meeting, 2008, New Orleans, LA, USA.

6. Bishram Singh Chouhan, Rajani Giridhar and Mange Ram Yadav, Microwave Assisted Synthesis of Substituted 4-Quinazolones, Medchem. India, 2007, Select Biosciences (UK), Hyderabad, India.

7. R.Ramajayam, Rajani Giridhar and Mange Ram Yadav Design, Synthesis and Evaluation of 2,3-diaryl-1-4-diazepinesas Potential Anti-Proliferative Agents, 230th ACS Annual National Meeting, Washington DC,USA.

8. Devendra Puntambekar, Rajani Giridhar and Mange Ram Yadav, Development of Predictive CoMFA and CoMSIA Models for Alkoxylated and Hydroxylated Chalcones as Anti-Malarial Agents, 230th ACS Annual National Meeting, Washington DC, USA.

9. Devendra Puntambekar, Rajani Giridhar and Mange Ram Yadav, Insight into the Structural Requirements of Farnesyltransferase Inhibitors as Potential Anti-tumor Agents Based on 3D-QSAR, CoMSIA and CoMFA models, 233th ACS Annual National Meeting, Chicago, USA.

10. Bishram Singh Chouhan, Rajani Giridhar and Mange Ram Yadav Design and Synthesis of Some Multitargeted Ligand as Potential Anti-hypertensive Agents, 234th ACS Annual National Meeting, Boston, USA.

11. Vijay Kumar Sharma, Mange Ram Yadav and Surender Singh, Naproxen-L-phenylalanine Alkyl Ester Prodrugs: Synthesis and biologicsl evaluation, Second World Congress on Inflammation, Brighton, U.K., Sept. 17-22, 1995, Abstract No. W19/5.

12. Anjali Bhasin, D.K. Majumdar and Mange Ram Yadav, Dissolution characteristics of diclofenac crystals obtained from various solvents, International Symposium on Recent Trends in Pharmaceutical Sciences, Ootacamund, Feb 18-20, 1995, Abstract No. D27.

13. S. Bhatia, Mange Ram Yadav, M. S. Y. Khan, A. Kar and S. Singh, Synthesis and CNS Profile of some 2-phenylindole derivatives, International Symposium on Recent Trends in Pharmaceutical Sciences, Ootacamund, Feb 18-20, 1995, Abstract No. B43.

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14. Harkishan Singh, Mange Ram Yadav and Dharam Paul, Steroidal [3,4-c]-1’,2’,5’-Oxadiazoles as potential bioactive molecules, in 10th International Congress of Heterocyclic Chemistry, University, University of Waterloo, Canada, 11-16th Aug. 1985, Abstract No. P9-284.

National:1. P. P. Naik, B. S. Chouhan, R. Giridhar and Mange Ram Yadav, Synthesis and cytotoxic

activity of a series of novel 2-substitutedaryl 4-amino- 6,7-dimethoxyquinazolines, 61st Indian Pharmaceutical Congress, Ahmedabad, Dec. 2009 Abstract No. B-259

2. D.G. Prajapati, A. V. Mantri, R. Giridhar, and Mange Ram Yadav, Synthesis of Allyloxy Substituted 4,6-diarylpyrimidines as Potential HIV Reverse Transcriptase Inhibitors, 61st Indian Pharmaceutical Congress, Ahmedabad, Dec. 2009 Abstract No. B-253

3. Dharmendrasinh A. Baria, Prafulla M. Sable, Rajani Giridhar, Mange Ram Yadav, D-ring modified hetero-steroids as potential aromatase inhibitors, 61st Indian Pharmaceutical Congress, Ahmedabad, Dec. 2009. Abstract No. B-232

4. D.G. Prajapati, R. S. Tamboli, R. Giridhar, and Mange Ram Yadav, Assessment of Anti-platelet activity of 2-aminopyrimidines, 61st Indian Pharmaceutical Congres Ahmedabad, Dec, 2009. Abstract No. B-215

5. Prafulla M. Sabale, Umang Shah, Rajani Giridhar and Mange Ram Yadav Design and Synthesis of Novel Steroidal Aromatase Inhibitors, 61st Indian Pharmaceutical Congress, Ahmedabad, Dec. 2009. Abstract No. B-205

6. Prashant R Murumkar, Sneha R Chandani, Rajani Giridhar and Mange Ram Yadav, “Pharmacophore alignment based CoMFA and CoMSIA studies for Tumor Necrosis Factor Alpha Converting Enzyme Inhibitors” presented in 61st Indian Pharmaceutical Sciences to be held at Ahmedabad in 2009. Abstract No. B-59

7. Vishal P Zambre Prashant R. Murumkar, Rajani Giridhar and Mange Ram Yadav, “Comparative Molecular Similarity Indices Analysis of DNA G-Quadruplex Mediating Telomerase Inhibitors, 61st Indian Pharmaceutical Congress, Ahmedabad, Dec. 2009 Abstract No. B-58

8. Prashant R. Murumkar, Vishal P. Zambre, Rajani Giridhar, Mange Ram Yadav, “Structure Guided 3D-QSAR: A Useful Approach for Designing of TACE Inhibitors” in 60th Indian Pharmaceutical Sciences at New Delhi in Dec. 2008

9. Prashant R. Murumkar, Rajani Giridhar, Mange Ram Yadav “Development of predictive 3D-QSAR CoMFA and CoMSIA Models for-aminohydoxamic acid-derived TNF-converting enzyme inhibitors” in 59th Indian Pharmaceutical Sciences at Varanasi on 21st Dec. 2007.

10. Ramajayam R, Rajani Giridhar and Mange Ram Yadav, ‘2,3-substituted diaryl-6,7-dihydro-5H-1,4-diazepine as potential medicinal agents’ 57th Indian Pharmaceutical Congress, Hyderabad, Dec. 02 to 04 2005, Abstract no. BP-54

28

11. A.K.Shinde, Rajani Giridhar, Robert Menard, Mange Ram Yadav, ‘Synthesis and Evaluation of dipeptide nitrites as selective cathepsin-L inhibitors.’ 57th Indian Pharmaceutical Congress, Hyderabad, Dec. 02 to 04 2005, Abstract no. B-16

12. Mange Ram Yadav, D.S.Puntambekar, K.P. Sarathi, S. vengurlekar and Rajani Giridhar, ‘Quantitative Structure Activity Relationship studies of diarylimidazoles as selective COX-II inhibitors’ 56th Indian Pharmaceutical Congress, Kolkata, Dec. 03 to 05 2004, Abstract no. BP-39

13. V. Alagarsami, Rajani Giridhar and Mange Ram Yadav, ‘Synthesis and Pharmacological investigation of some novel 1,2,4-triazoloquinazoline-5(4H)-ones as antihistaminic agents’ 56th Indian Pharmaceutical Congress, Kolkata, Dec. 03 to 05 2004, Abstract no. B-11

14. H.B. Prajapati, Shrikant T. Shirude, Rajani Giridhar, R.Balaraman, A. Parmar and Mange Ram Yadav, ‘Synthesis and evaluation of 3,4-diaryl-1,2,5-oxadiazoles and corresponding N-Oxides as selective COX-II inhibitors’ 56th Indian Pharmaceutical Congress, Kolkata, Dec. 03 to 05 2004, Abstract no. B-5

15. A.K.Shinde, Rajani Giridhar and Mange Ram Yadav, ‘Cysteine protease inhibitors as potential anti-malarial drugs.’ 56th Indian Pharmaceutical Congress, Kolkata, Dec. 03 to 05 2004, Abstract no. B-3

16. Dharmendra G. Patel, Rajani Giridhar and Mange Ram Yadav, ‘Fujita Ban modified De-Novo studies on triazolinone-based balanced AT1-AT2 receptor antagonists.’ 55th Indian Pharmaceutical Congress, Chennai, Dec. 19 to 21 2003, Abstract no. BP-43

17. Datta M. Nimekar, Pathik S Brahmhkshatria, Rajani Giridhar and Mange Ram Yadav, p-aminophenol and acetylated phenol derivatives of certain commonly available NSAIDs as more COX-II selective inhibitors, 55th Indian Pharmaceutical Congress, Chennai, Dec. 19 to 21 2003, Abstract no. BP-42

18. Shitesh R. Patel, M.M.Ganesh, R.Ramajayam, Rajani Giridhar and Mange Ram Yadav, ‘16ξ-dimethylamine-3-pyrrolidino-5-androstane dimethiodide as a potential neuromuscular blocking agents’ 55th Indian Pharmaceutical Congress, Chennai, Dec. 19 to 21 2003, Abstract no. BP-41

19. P.K.Halen, K.K.Chagti, Rajani Giridhar and Mange Ram Yadav, ‘Synthesis and evaluation of certain ketorolac analogs with an improved therapeutic profile’ 55th Indian Pharmaceutical Congress, Chennai, Dec. 19 to 21 2003, Abstract no. BP-40

20. Sudha Vengurlekar, K.P.Sarathi, Rajani Giridhar and Mange Ram Yadav, ‘Structural requirements for 1,2-diarylimidazole as COX-II inhibitors: Hansch Analysis.’ 55th Indian Pharmaceutical Congress, Chennai, Dec. 19 to 21 2003, Abstract no. BP-39

21. K.K.Chagti, P.K.Halen, Rajani Giridhar and Mange Ram Yadav, ‘Indomethacin Derivatives with a better pharmacokinetics and pharmacodynamic profile’ 55th Indian Pharmaceutical Congress, Chennai, Dec. 19 to 21 2003, Abstract no. B-36

29

22. K.K.Chagti, P.K.Halen, Rajani Giridhar and Mange Ram Yadav, ‘Synthesis, Pharmacokinetics and Pharmacodynamic Profile of beta-amino ester derivatives of Ketoprofen’ 54th Indian Pharmaceutical Congress, Pune, Dec. 13 to 15 2002, Abstract no. BP-46

23. P.K.Halen, K.K.Chagti, Rajani Giridhar and Mange Ram Yadav, ‘Synthesis and Evaluation of certain Diclofenac analogues with therapeutic advantage over the parent drug.’ 54th Indian Pharmaceutical Congress, Pune, Dec. 13 to 15 2002, Abstract no. B-33

24. J.B. Majethia, R. Balaraman, Rajani Giridhar, Mange Ram Yadav, ‘Effect of vanadium and its complex on the blood glucose and lipid profile of Strptozocin induced diabetic rats’ 53nd Indian Pharmaceutical Congress, New Delhi, Dec. 21 to 23 2001, Abstract no. E-23

25. K.P.Sarathi, Rajani Giridhar and Mange Ram Yadav, ‘Structural Requirements for COX-1 and COX-II activity in 3,4-diaryl five membered ring system: Fujita Ban QSAR Approach Combined with Hansch Analysis ’ 53nd Indian Pharmaceutical Congress, New Delhi, Dec. 21 to 23 2001, Abstract no. B-36

26. P.K.Halen, K.K.Chagti, R.Giridhar and Mange Ram Yadav, ‘Synthesis and Evaluation of Some Naproxen analogues as dual acting potential drugs.’ 53nd Indian Pharmaceutical Congress, New Delhi, Dec. 21 to 23 2001, Abstract no. B-22

27. V. Ganeshan, Rajani Giridhar, Hetal Prajapati and Mange Ram Yadav, ‘Polymorphism in Sparfloxacine: Characterization and Dissolution studies.’ 53nd Indian Pharmaceutical Congress, New Delhi, Dec. 21 to 23 2001, Abstract no. A-72

28. Revathi R, Rajani Giridhar and Mange Ram Yadav, ‘Studies on some metal complexes of curcumin’ 52nd Indian Pharmaceutical Congress, Hyderabad, Dec. 1 to 3 2000, Abstract no. BP-34

29. Reshmi C.S, Kewal K. Chagti, Rajani Giridhar and Mange Ram Yadav, ‘A New Approach in the Direction of Therapeutic optimization of NSAIDs- A Study in the Synthesis and Kinetics of Some NSAIDs Derivatives’ 52nd Indian Pharmaceutical Congress, Hyderabad, Dec. 1 to 3 2000, Abstract no. BP-26

30. Hemalatha B, Rajani Giridhar and Mange Ram Yadav, ‘Synthesis and biological activity of Gastroprotective analogues of some NSAIDs.’ 52nd Indian Pharmaceutical Congress, Hyderabad, Dec. 1 to 3 2000, Abstract no. B-11

31. M.M. Ganesh, Hetal B. Prajapati, Rajani Giridhar and Mange Ram Yadav, ‘COX-1 Vs COX-II selectivity: A Molecular Modeling and QSAR study on 7-tertialrybutyl-2,3-dihydro-3,3-dimethylbenzofuran derivatives.’ 52nd Indian Pharmaceutical Congress, Hyderabad, Dec. 1 to 3 2000, Abstract no. B-6

32. Mange Ram Yadav, Rajani Giridhar, Mukesh Mahatma and Prafulla M.Sabale, 4ξ-acetoxy-17A, methyl-3ξ-pyrrolidino-17A-aza-D-homo 5α-androstene-dimethiodide: A new neuromuscular blocking agent. 17th Asian Congress of Pharmaceutical Sciences, Mumbai, Dec. 10 to 13 1998, Abstract No. IBP-23

30

33. Anjali Kapoor, D.K.Majumdar and Mange Ram Yadav, Dissolution Characteristics of various physical forms of Nimesulide. 48th Indian Pharmaceutical Congress, Chennai, Dec. 25th to 27th 1996, Abstract No. AP-25.

34. Nirmal Sharma, Sharda Sushil, A.K. Sharma, Mange Ram Yadav, Sumitra Yadav, Sangeeta Bhatia, S. Singh, R. Verma and V.K. Sharma, Teaching and reasearch- oriented to team work, 46th Indian Pharmaceutical Congress, Chandigarh, Dec 28-30, 1994.

35. Surendra N. Pandeya, and Mange Ram Yadav, Synthesis and Biological Activity of α,α'-Thiobisformamidine (Amidine) Salts, 46th Indian Pharmaceutical Congress, Chandigarh, Dec 28-30, 1994, Abstract No. B-41.

36. Mange Ram Yadav and Dharam Paul Jindal, 17-Substituted Steroidal [3,4-c]-1',2',5'-oxadiazole, 42th Indian Pharmaceutical Congress, Manipal, Dec 28-30, 1990, Abstract No. A20.

37. Mange Ram Yadav and Dharam Paul Jindal, Heteroaromatic Ring- fused Steroids, 41th

Indian Pharmaceutical Congress, Bombay, Dec 16-18, 1989, Abstract No. A19.

38. Jojy Abraham, Mange Ram Yadav and Dharam Paul Jindal, Certain Heterocycle- fused Azasteroids, 41th Indian Pharmaceutical Congress, Bombay, Dec 16-18, 1989, Abstract No. A7.

39. Dharam Paul Jindal, Inder Bir Singh and Mange Ram Yadav, Synthesis and Study of Heterocyclic Steroids, 40th Indian Pharmaceutical Congress, Calcutta, Dec 26-28 , 1988, Abstract No. A16.

40. Dharam Paul Jindal, Jojy Abraham and Mange Ram Yadav, 17a-methyl-17a-aza-D-homo-5α-androstano[3,4-c]-1',2',5'-oxadiazole, 39th Indian Pharmaceutical Congress, Madras, Dec 27-29 , 1986, Abstract No. A15.

41. Dharam Paul Jindal, J.S.R.A. Sharma and Mange Ram Yadav, Synthesis and Study of Steroidal [3,4-c]-1',2',5'-oxadiazole N-oxide, 39th Indian Pharmaceutical Congress, Madras, Dec 27-29 , 1986, Abstract No. A14.

42. Vijay K. Kapoor, Kewal Krishan, Mange Ram Yadav and Dharam Paul Jindal Synthesis and Anti-inflamatory activity of some camphor analouges, 38th Indian Pharmaceutical Congress, Ahmedabad, Dec 21-23, 1986, Abstract No. A15.

43. Dharam Paul Jindal, Neeta Sharma, and Mange Ram Yadav, 2'-Phenyl-5α-pregnano [3,4-c]-1',2',3'-triazol-20-one, 38th Indian Pharmaceutical Congress, Ahmedabad, Dec 21-23, 1986, Abstract No. A16.

44. Dharam Paul Jindal, Jojy Abraham and Mange Ram Yadav, 17-oxo-17a-aza-D-homo-5α-androstano[3,4-c]-1',2',5'-oxadiazole N-oxide, 38th Indian Pharmaceutical Congress, Ahmedabad, Dec 21-23, 1986, Abstract No. A5.

31

45. Dharam Paul, Mange Ram Yadav, and Harkishan Singh, Studies in the Synthesis of Steroidal 5-eno [3,4-c]-1',2',5'-oxadiazole, 37th Indian Pharmaceutical Congress, New Delhi, Dec 26-28, 1985, Abstract No. A10.

46. Harkishan Singh, Mange Ram Yadav, and Dharam Paul, Steroidal [3,4-c]-1',2',5'-oxadiazoles a Potential Bioactive Molecules, 10th International Congress of Heterocyclic Chemistry. Aug 11-16, 1985, University Of Waterloo, Ontario, Canada, Abstract No. p-284.

47. Harkishan Singh, Dharam Paul, Mange Ram Yadav, Rakesh Kumar Sharma and Vijaykumar R. Agrawal, 5-Pregnano[3,4-c]-1',2',5'-oxadiazoles, 36th Indian Pharmaceutical Congress, Bangalore, Feb 9-11, 1985, Abstract No. A15.

48. Harkishan Singh, Mange Ram Yadav, Dharam Paul, Sat Paul Garg and Rakesh Kumar Sharma, Steroidal [3,4-c]-1',2',5'-oxadiazoles, 35th Indian Pharmaceutical Congress, Hyderabad, Dec 18-20,1983, Abstract No. A28.

(Dr M. R. Yadav)

*************

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BIO-DATA OF M - Maharaja Sayajirao University of … · Web viewBIO-DATA OF M.R.YADAV Name : Dr. M. R. Yadav PERSONAL Address : Official Residential Pharmacy Department, Faculty of