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ChemInform 2010, 41, issue 29 © 2010 Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim www.cheminform.wiley-vch.de Tetrazole derivatives R 0310 DOI: 10.1002/chin.201029156 A Mild and General One-Pot Preparation of Cyanoethyl-Protected Tetrazoles. — The procedure for the synthesis of title compounds possessing acid-sensitive func- tionalities employs pyridine to mitigate the negative effects of HCl generated during the formation of imidoyl chlorides from amides (III) and PCl5. — (KENNEDY, L.; Tetrahedron Lett. 51 (2010) 15, 2010-2013; Metab. Dis. Chem., Bristol-Myers Squibb, Princeton, NJ 08543, USA; Eng.) — Mais 29- 156

ChemInform Abstract: A Mild and General One-Pot Preparation of Cyanoethyl-Protected Tetrazoles

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Tetrazole derivativesR 0310 DOI: 10.1002/chin.201029156

A Mild and General One-Pot Preparation of Cyanoethyl-Protected Tetrazoles. — The procedure for the synthesis of title compounds possessing acid-sensitive func-tionalities employs pyridine to mitigate the negative effects of HCl generated during the formation of imidoyl chlorides from amides (III) and PCl5. — (KENNEDY, L.; Tetrahedron Lett. 51 (2010) 15, 2010-2013; Metab. Dis. Chem., Bristol-Myers Squibb, Princeton, NJ 08543, USA; Eng.) — Mais

29- 156

ChemInform 2010, 41, issue 29 © 2010 Wiley-VCH Verlag GmbH & Co. KGaA, Weinheim