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8/18/2019 FARMACOCINETICA FARMACODINAMIA
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Para ácidos
pKa = log + pH
(Ácido ionizado)
Para bases
pKb
(Ácido no ionizado)
+ pH(Base no Ionizada)
(Base ionizada)
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TRANSPRT! !SP!"IA#I$A% %! &N S&STRAT(S) '!%IA% PR &N TRANSPRTA%R (T)
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ABSR"IN %! #S AR'A"S !N !#INT!STIN !N &N"IN %!# pKa
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ases del *eabolis*o
,epaicoár*aco ase - !nzi*as
.idaci/nRed0cci/nHidr/lisis%escarbo.ilaci/n
'eabolios ase 1!nzi*as
"on20gaci/n con3 Acido gl0cor/nico Acido S0l45rico Acido Ac6ico7l0a*ina7licocola
'eabolios
A"TI8 N P#AR A"TI8 'ÁS P#AR INA"TI8 P#AR
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AR'A"%INA'IAINT!RR!#A"IN
AR'A"9R!"!PTR
%rRo*ero B
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