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Chemistry Services for Drug Discovery The SP The SP 3 3 -Collection -Collection Designed for Medicinal Chemistry Research

TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

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Page 1: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

Chemistry Services for Drug Discovery

The SPThe SP33-Collection-CollectionDesigned for Medicinal Chemistry Research

Page 2: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

Welcome to our new catalogue for medicinal chemistry containing compounds chosen as examples to highlight the variety of structures in our diverse total collection of “30,000” available compounds which can be found on our website.

This catalogue focusses on ring structures containing sp3-hybridised carbon atoms which are generally considered to have a three-dimensional character. These compounds offer the possibility to access biological targets with more globular shapes. Research has shown that a higher proportion of sp3-hybridised carbon atoms in compounds is associated with increased solubility and successful progression though clinical testing. Moreover, increased hetero-aliphatic ring count in lead compounds correlates to the desirable properties of decreased lipophilicity, increased solubility, decreased albumin-binding and reduced cytochrome P450 inhibition.

The compounds are arranged for ease of browsing into structural categories. The availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation of physicochemical properties and enables the probing of binding sites. Fluorine can modify the metabolic stability and pKa of compounds. The incorporation of functional groups such as boronic acids, carboxylic acids, aldehydes, amino and alcohols enables expedient synthetic strategies.

Our compounds are in stock for express delivery at competitive prices.

The complete collection can be found and searched on our website:

www.activate-scientifi c.com

Dear Colleague,

Spirocyclic Rings ............................................................................................................... 3

Bicyclic Rings .................................................................................................................. 19

Cyclopropanes ................................................................................................................ 32

Oxetanes ........................................................................................................................ 34

Cyclobutanes .................................................................................................................. 36

Azetidines ....................................................................................................................... 44

Cyclopentanes ................................................................................................................. 46

Pyrrolidines ..................................................................................................................... 48

Tetrahydrofurans ............................................................................................................. 50

Cyclohexanes .................................................................................................................. 52

Piperidines ...................................................................................................................... 54

Tetrahydropyrans ............................................................................................................ 56

Piperazines ..................................................................................................................... 58

Morpholines .................................................................................................................... 60

Page 3: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

3

Chemistry Services for Drug Discovery www.activate-scientifi c.com

Activate Scientifi c · Am Mitterweg 12 · D-83209 Prien · Germany · Tel: +49 (0) 8051-965166021A The Maltings · Roydon Road · Stanstead Abbotts · Hertfordshire SG12 8HG · UK · Tel: +44 (0) 1279843244

www.activate-scientifi c.com · info@activate-scientifi c.com · info-uk@activate-scientifi c.com

Spiro Compounds [2.3]-[2.4]-[2.5]

Spiro[2.3]hexane-1-carboxylic acid

On Stock

381,00 € 250mg

AS56538

(E)-1-Oxaspiro[2.3]hexane-5-carbonitrile

On Stock

686,00 € 250mg

AS15001

1,1-Difl uoro-5-azaspiro[2.3]hexane HCl

On Stock

558,00 € 250mg

AS56004

5-Boc-1-amino-5-azaspiro[2.3]hexane

CALL

1380,00 € 1g

AS62930

5-Methyl-5-azaspiro[2.3]hexane-1-carboxylic acid

CALL

1380,00 € 1g

AS62931

4-Azaspiro[2.4]heptane oxalate

On Stock

695,00 € 250mg

AS17849

4-Azaspiro[2.4]heptan-5-one

On Stock

166,00 € 250mg

AS26819

5-Azaspiro[2.4]heptane HCl

On Stock

295,00 € 100mg

AS17887

1,1-Difl uoro-5-azaspiro[2.4]heptane HCl

On Stock

558,00 € 250mg

AS51653

5-Boc-5-azaspiro[2.4]heptane-1-methanol

On Stock

457,00 € 100mg

AS56061

5-Boc-5-azaspiro[2.4]heptane-1-carboxylic acid

On Stock

725,00 € 1g

AS55531

1-Amino-5-Boc-5-azaspiro[2.4]heptane

On Stock

341,00 € 100mg

AS18101

(R)-7-(Boc-amino)-5-azaspiro[2.4]heptane

On Stock

280,00 € 250mg

AS41145

(S)-7-(Boc-amino)-5-azaspiro[2.4]heptane

On Stock

250,00 € 250mg

AS17618

5-(Boc-amino)-5-azaspiro[2.4]heptane HCl

On Stock

558,00 € 250mg

AS56355

Spiro[2.5]octane-6-carboxylic acid

On Stock

367,00 € 250mg

AS37315

6-(Methylamino)spiro[2.5]octane-1-carboxylic acid

CALL

1380,00 € 1g

AS63412

6-Oxaspiro[2.5]octane-1-carboxylic acid

On Stock

269,00 € 250mg

AS55466

6-Thiaspiro[2.5]octane-1-amine

CALL

985,00 € 1g

AS63415

4-Azaspiro[2.5]octane HCl

CALL

1120,00 € 1g

AS51930

1,1-Difl uoro-5-azaspiro[2.5]octane HCl

On Stock

394,00 € 250mg

AS56003

5-Boc-5-azaspiro[2.5]octane-1-carboxylicacid

On Stock

419,00 € 250mg

AS56209

6-Azaspiro[2.5]octane HCl

On Stock

365,00 € 1g

AS17850

1,1-Difl uoro-6-azaspiro[2.5]octane HCl

On Stock

352,00 € 250mg

AS56002

Page 4: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

Chemistry Services for Drug Discovery www.activate-scientifi c.com

4

Standard Pack Sizes: 1-5-10-25g • Call for 100-250-1000g pilot plant scale up

Spiro Compounds [2.5]-[3.3]

6-Boc-6-azaspiro[2.5]octan-4-ol

On Stock

365,00 € 250mg

AS57919

6-Azaspiro[2.5]octane-1-methanol

CALL

1320,00 € 1g

AS16089

6-Boc-1-amino-6-azaspiro[2.5]octane HCl

On Stock

166,00 € 250mg

AS16084-B

6-Boc-1-(aminomethyl)-6-azaspiro[2.5]-octane

On Stock

254,00 € 250mg

AS39320

6-Methyl-6-azaspiro[2.5]octane-1-amine

CALL

1380,00 € 1g

AS63058

6-Boc-6-azaspiro[2.5]octane-1-carboxylicacid

On Stock

239,00 € 1g

AS28479

6-Methyl-6-azaspiro[2.5]octane-1-carboxylic acid

CALL

1360,00 € 1g

AS63057

7-Oxa-4-azaspiro[2.5]octane HCl

On Stock

689,00 € 250mg

AS64211

7-Oxa-4-azaspiro[2.5]octan-5-one

On Stock

1560,00 € 1g

AS64130

6-Boc-1-oxa-6-azaspiro[2.5]octane

On Stock

142,00 € 1g

AS15293

4-Oxa-7-azaspiro[2.5]octane HCl

On Stock

1265,00 € 1g

AS64207

4-Oxa-7-azaspiro[2.5]octan-6-one

On Stock

1293,00 € 1g

AS64206

5-Oxa-7-azaspiro[2.5]octan-6-one

On Stock

527,00 € 1g

AS78377

4,7-Diazaspiro[2.5]octane oxalate

On Stock

330,00 € 250mg

AS17626-C

4-Boc-4,7-diazaspiro[2.5]octane

On Stock

429,00 € 250mg

AS39068

7-Boc-4,7-diazaspiro[2.5]octane

On Stock

710,00 € 1g

AS32599

7-Boc-4,7-diazaspiro[2.5]octane-5-one

On Stock

467,00 € 1g

AS78195

5-Methyl-5,7-diazaspiro[2.5]octan-6-one

On Stock

527,00 € 1g

AS78378

1,6-Dioxaspiro[2.5]octane

On Stock

279,00 € 250mg

AS15270

Spiro[3.3]heptan-2-one

On Stock

284,00 € 250mg

AS55895

Spiro[3.3]heptan-2-ol

On Stock

189,00 € 100mg

AS57532

Spiro[3.3]heptane-2-carboxylic acid

On Stock

284,00 € 250mg

AS55483

Spiro[3.3]heptan-2-amine HCl

On Stock

365,00 € 250mg

AS56958

6,6-Difl uorospiro[3.3]heptan-2-amine HCl

On Stock

333,00 € 100mg

AS56916

Page 5: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

Activate Scientifi c · Am Mitterweg 12 · D-83209 Prien · Germany · Tel: +49 (0) 8051-965166021A The Maltings · Roydon Road · Stanstead Abbotts · Hertfordshire SG12 8HG · UK · Tel: +44 (0) 1279843244

www.activate-scientifi c.com · info@activate-scientifi c.com · info-uk@activate-scientifi c.com

5

Chemistry Services for Drug Discovery www.activate-scientifi c.com

Spiro Compounds [3.3]

6,6-Difl uorospiro[3.3]heptane-2-carboxylicacid

On Stock

405,00 € 250mg

AS55805

6-Oxospiro[3.3]heptane-2-carboxylic acid

On Stock

195,00 € 250mg

AS51897

Methyl 6-oxospiro[3.3]heptane-2-carboxylate

On Stock

290,00 € 250mg

AS17571

2-(Boc-amino)spiro[3.3]heptane-6-one

On Stock

284,00 € 250mg

AS51898

Methyl 6-aminospiro[3.3]heptane-2-carboxylate HCl

On Stock

437,00 € 250mg

AS56071

6-(Boc-amino)spiro[3.3]heptane-2-carboxylic acid

On Stock

405,00 € 250mg

AS51722

6-(Boc-amino)spiro[3.3]heptane-2-amine

On Stock

375,00 € 250mg

AS51671

1-Azaspiro[3.3]heptane oxalate

On Stock

308,00 € 100mg

AS17888

1-Boc-1-azaspiro[3.3]heptane-6-one

On Stock

564,00 € 100mg

AS56379

1-Boc-1-azaspiro[3.3]heptane-6-ol

On Stock

813,00 € 250mg

AS18217

1-Boc-1-azaspiro[3.3]heptane-6-carboxylicacid

On Stock

749,00 € 100mg

AS56399

2-Azaspiro[3.3]heptane hemioxalate

On Stock

165,00 € 1g

AS51674-C

2-Boc-2-azaspiro[3.3]heptane

On Stock

312,00 € 250mg

AS51667

5,5-Difl uoro-2-azaspiro[3.3]heptane TFA

On Stock

493,00 € 100mg

AS56413

2-Boc-2-azaspiro[3.3]heptane-5-one

On Stock

370,00 € 100mg

AS52021

2-Boc-2-azaspiro[3.3]heptane-5-ol

On Stock

594,00 € 100mg

AS18117

5-(Boc-amino)-2-azaspiro[3.3]heptane

On Stock

493,00 € 100mg

AS56199

6,6-Difl uoro-2-azaspiro[3.3]heptane TFA

On Stock

329,00 € 100mg

AS51956

2-Boc-6,6-difl uoro-2-azaspiro[3.3]heptane

On Stock

300,00 € 100mg

AS51790

2-Boc-2-azaspiro[3.3]heptane-6-one

On Stock

158,00 € 250mg

AS12047

2-Azaspiro[3.3]heptan-6-ol HCl

On Stock

284,00 € 250mg

AS56296-B

2-Boc-2-azaspiro[3.3]heptan-6-ol

On Stock

128,00 € 250mg

AS12048

2-Boc-2-azaspiro[3.3]heptane-6-methanol

On Stock

353,00 € 100mg

AS56274

2-Boc-2-azaspiro[3.3]heptane-6-carboxylicacid

On Stock

270,00 € 250mg

AS51092

Page 6: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

Chemistry Services for Drug Discovery www.activate-scientifi c.com

6

Standard Pack Sizes: 1-5-10-25g • Call for 100-250-1000g pilot plant scale up

SPIRO COMPOUNDS [3.3]

2-Azaspiro[3.3]heptane-6-carboxylic acidTFA

On Stock

419,00 € 250mg

AS51093

Methyl 2-Boc-2-azaspiro[3.3]heptane-6-carboxylate

On Stock

394,00 € 250mg

AS56479

2-Boc-6-amino-2-azaspiro[3.3]heptane

On Stock

240,00 € 250mg

AS12049

2-Boc-6-aminomethyl-2-azaspiro[3.3]-heptane

On Stock

482,00 € 100mg

AS56276

6-(Boc-amino)-2-azaspiro[3.3]heptane HCl

On Stock

490,00 € 250mg

AS3575-B

6-Amino-2-azaspiro[3.3]heptane-6-carboxylic acid

On Stock

938,00 € 250mg

AS3576

6-(Trifl uoromethyl)-2-azaspiro[3.3]-heptan-6-ol HCl

On Stock

298,00 € 100mg

AS57262

2-Oxaspiro[3.3]heptan-6-one

On Stock

363,00 € 250mg

AS12916

2-Oxaspiro[3.3]heptan-6-ol

On Stock

270,00 € 250mg

AS17397

2-Oxaspiro[3.3]heptane-6-methanol

On Stock

419,00 € 100mg

AS52038

6-Amino-2-oxaspiro[3.3]heptane HCl

On Stock

270,00 € 250mg

AS51949

2-Oxaspiro[3.3]heptane-6-methanamine

On Stock

688,00 € 100mg

AS56403

6-(Methylamino)-2-oxaspiro[3.3]heptane

On Stock

1323,00 € 250mg

AS52048

6-Bromo-2-oxaspiro[3.3]heptane

On Stock

621,00 € 250mg

AS56273

6-Iodo-2-oxaspiro[3.3]heptane

On Stock

248,00 € 100mg

AS52053

2,6-Dioxaspiro[3.3]heptane

On Stock

370,00 € 250mg

AS51988

1-Thia-6-azaspiro[3.3]heptane HCl

CALL

1008,00 € 250mg

AS52029

6-Boc-1-thia-6-azaspiro[3.3]heptane

CALL

820,00 € 250mg

AS52060

1-Thia-6-azaspiro[3.3]heptane-1,1-dioxide HCl

On Stock

991,00 € 250mg

AS52028

2-Thiaspiro[3.3]heptan-6-one

On Stock

375,00 € 100mg

AS55619

2-Thia-6-azaspiro[3.3]heptane-2,2-dioxideHCl

On Stock

370,00 € 100mg

AS51887

2-Thia-6-azaspiro[3.3]heptanehemioxalate

On Stock

464,00 € 250mg

AS9653-B

2-Boc-6-thia-2-azaspiro[3.3]heptane

CALL

1650,00 € 1g

AS51885

6-Oxa-1-azaspiro[3.3]heptane hemioxalate

On Stock

270,00 € 100mg

AS6088-B

Page 7: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

Activate Scientifi c · Am Mitterweg 12 · D-83209 Prien · Germany · Tel: +49 (0) 8051-965166021A The Maltings · Roydon Road · Stanstead Abbotts · Hertfordshire SG12 8HG · UK · Tel: +44 (0) 1279843244

www.activate-scientifi c.com · info@activate-scientifi c.com · info-uk@activate-scientifi c.com

7

Chemistry Services for Drug Discovery www.activate-scientifi c.com

SPIRO COMPOUNDS [3.3]-[3.4]

1-Boc-6-oxa-1-azaspiro[3.3]heptane

On Stock

185,00 € 100mg

AS6108

1-Oxa-6-azaspiro[3.3]heptane HCl

On Stock

189,00 € 100mg

AS12211-B

6-Boc-1-oxa-6-azaspiro[3.3]heptane

On Stock

334,00 € 250mg

AS51901

6-Boc-1-oxa-6-azaspiro[3.3]heptan-3-one

On Stock

1650,00 € 1g

AS52051

6-Boc-1-oxa-6-azaspiro[3.3]heptan-3-amine

On Stock

688,00 € 100mg

AS52050

2-Oxa-6-azaspiro[3.3]heptane hemioxalate

On Stock

125,00 € 1g

AS12178-B

6-Boc-2-Oxa-6-azaspiro[3.3]heptane

On Stock

265,00 € 1g

AS12977

1-Boc-1,6-diazaspiro[3.3]heptanehemioxalate

On Stock

290,00 € 100mg

AS16399

2,6-Diazaspiro[3.3]heptane diHCl

On Stock

388,00 € 250mg

AS12203-B

2-Boc-2,6-diazaspiro[3.3]heptanehemioxalate

On Stock

180,00 € 250mg

AS12111-C

6-Boc-3,6-diazaspiro[3.3]heptane oxalate

On Stock

220,00 € 100mg

AS51793

2-Azaspiro[3.4]octane hemioxalate

On Stock

352,00 € 250mg

AS56681

2-Boc-2-azaspiro[3.4]octane-5-one

On Stock

385,00 € 100mg

AS56578

2-Boc-2-azaspiro[3.4]octane-6-one

On Stock

200,00 € 100mg

AS18124

2-Boc-2-azaspiro[3.4]octan-6-ol

On Stock

350,00 € 100mg

AS18208

2-Boc-5-oxa-2-azaspiro[3.4]octane-7-one

On Stock

365,00 € 250mg

AS57648

6-Oxa-1-azaspiro[3.4]octane hemioxalate

On Stock

350,00 € 100mg

AS18175

5-Oxa-2-azaspiro[3.4]octane HCl

CALL

716,00 € 250mg

AS13128-B

6-Oxa-2-azaspiro[3.4]octane HCl

CALL

621,00 € 250mg

AS13129-B

2-Boc-6-thia-2-azaspiro[3.4]octan-8-ol

CALL

1750,00 € 1g

AS52064

5-Azaspiro[3.4]octane hemioxalate

On Stock

270,00 € 100mg

AS52044-B

2-Amino-5-Boc-5-azaspiro[3.4]octane

On Stock

649,00 € 100mg

AS56279

2-(Boc-amino)-5-azaspiro[3.4]octane

On Stock

621,00 € 100mg

AS56280

5-Azaspiro[3.4]octane-2-carboxylic acidHCl

On Stock

674,00 € 100mg

AS56364

Page 8: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

Chemistry Services for Drug Discovery www.activate-scientifi c.com

8

Standard Pack Sizes: 1-5-10-25g • Call for 100-250-1000g pilot plant scale up

SPIRO COMPOUNDS [3.4]

5-Boc-5-azaspiro[3.4]octane-2-carboxylicacid

On Stock

725,00 € 100mg

AS56277

2-Oxa-5-azaspiro[3.4]octane hemioxalate

On Stock

350,00 € 100mg

AS6091-B

5-Boc-2-oxa-5-azaspiro[3.4]octane

On Stock

416,00 € 250mg

AS6110

6-Azaspiro[3.4]octane hemioxalate

On Stock

250,00 € 250mg

AS17676-B

6-Boc-6-azaspiro[3.4]octane-2-one

On Stock

138,00 € 250mg

AS12917

6-Boc-6-azaspiro[3.4]octan-2-ol

On Stock

386,00 € 1g

AS39801

6-Azaspiro[3.4]octane-2-methanol

On Stock

446,00 € 100mg

AS56589

6-Boc-6-azaspiro[3.4]octane-2-methanol

On Stock

446,00 € 100mg

AS56275

6-Boc-6-azaspiro[3.4]octane-2-carboxylicacid

On Stock

558,00 € 500mg

AS52052

1-(Boc-amino)-6-azaspiro[3.4]octane HCl

On Stock

965,00 € 250mg

AS56200-B

6-Boc-2-amino-6-azaspiro[3.4]octane

On Stock

411,00 € 250mg

AS18056

2-(Boc-amino)-6-azaspiro[3.4]octane

On Stock

482,00 € 100mg

AS52031

1-Oxa-6-azaspiro[3.4]octane hemioxalate

On Stock

352,00 € 250mg

AS51842

6-Boc-1-oxa-6-azaspiro[3.4]octane

On Stock

260,00 € 100mg

AS51845

6-Boc-1-oxa-6-azaspiro[3.4]octane-3-one

CALL

2460,00 € 1g

AS52049

2-Oxa-6-azaspiro[3.4]octane hemioxalate

On Stock

230,00 € 250mg

AS6087-B

6-Boc-2-oxa-6-azaspiro[3.4]octane

On Stock

370,00 € 250mg

AS6111

2-Oxa-6-azaspiro[3.4]octan-7-one

On Stock

490,00 € 250mg

AS6030

7-Boc-7-azaspiro[3.4]octane-3-one

On Stock

410,00 € 100mg

AS52018

5-Oxa-7-azaspiro[3.4]octan-6-one

On Stock

305,00 € 100mg

AS55601

1-Boc-1,6-diazaspiro[3.4]octanehemioxalate

On Stock

320,00 € 100mg

AS55546

6-Boc-1,6-diazaspiro[3.4]octanehemioxalate

On Stock

254,00 € 100mg

AS51767-C

2-Boc-2,5-diazaspiro[3.4]octanehemioxalate

On Stock

312,00 € 100mg

AS13120

5-Boc-2,5-diazaspiro[3.4]octane

On Stock

248,00 € 100mg

AS51987

Page 9: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

Activate Scientifi c · Am Mitterweg 12 · D-83209 Prien · Germany · Tel: +49 (0) 8051-965166021A The Maltings · Roydon Road · Stanstead Abbotts · Hertfordshire SG12 8HG · UK · Tel: +44 (0) 1279843244

www.activate-scientifi c.com · info@activate-scientifi c.com · info-uk@activate-scientifi c.com

9

Chemistry Services for Drug Discovery www.activate-scientifi c.com

Spiro Compounds [3.4]-[3.5]

2,5-Diazaspiro[3.4]octan-6-one HCl

On Stock

375,00 € 100mg

AS55955

2,6-Diazaspiro[3.4]octane diHCl

On Stock

255,00 € 250mg

AS57589

2-Boc-2,6-diazaspiro[3.4]octane

On Stock

252,00 € 250mg

AS51115-A

6-Boc-2,6-diazaspiro[3.4]octane HCl

On Stock

219,00 € 250mg

AS12376-B

2,6-Diazaspiro[3.4]octan-5-one HCl

On Stock

254,00 € 100mg

AS57267

2-Methyl-2,6-diazaspiro[3.4]octane oxalate

On Stock

220,00 € 100mg

AS12455

2-Boc-2,6-diazaspiro[3.4]octane-5-one

On Stock

223,00 € 100mg

AS57122

2,6-Diazaspiro[3.4]octan-7-one oxalate

On Stock

560,00 € 250mg

AS13116-B

2-Boc-2,6-diazaspiro[3.4]octane-7-one

On Stock

138,00 € 250mg

AS51896

5,8-Dioxaspiro[3.4]octane-2-methanol

On Stock

265,00 € 1g

AS17067

Methyl 5,8-dioxaspiro[3.4]octane-2-carboxylate

On Stock

235,00 € 1g

AS17002

2-Bromo-5,8-dioxaspiro[3.4]octane

On Stock

725,00 € 1g

AS55491

2,5,7-Triazaspiro[3.4]octan-8-one HCl

CALL

965,00 € 1g

AS3334

2-Boc-2-azaspiro[3.5]nonan-7-one

On Stock

330,00 € 100mg

AS17972

2-Boc-2-azaspiro[3.5]nonan-7-ol

On Stock

320,00 € 100mg

AS17934

2-Boc-2-azaspiro[3.5]nonane-7-carboxylic acid

On Stock

480,00 € 100mg

AS18188

2-Boc-7-amino-2-azaspiro[3.5]nonane

On Stock

720,00 € 250mg

AS18439

2-Oxaspiro[3.5]nonan-7-one

On Stock

360,00 € 250mg

AS52039

2-Oxaspiro[3.5]nonane-7-methanol

On Stock

420,00 € 250mg

AS52042

2-Oxaspiro[3.5]nonane-7-carboxylic acid

On Stock

1150,00 € 250mg

AS52040

2-Oxaspiro[3.5]nonane-7-methanamine

On Stock

961,00 € 250mg

AS52041

2-Oxaspiro[3.5]nonane-6,8-dione

On Stock

446,00 € 100mg

AS56659

7-Oxaspiro[3.5]nonan-2-ylmethanamine

On Stock

950,00 € 250mg

AS56587

5-Oxa-2-azaspiro[3.5]nonane HCl

CALL

739,00 € 250mg

AS13130-B

Page 10: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

Chemistry Services for Drug Discovery www.activate-scientifi c.com

10

Standard Pack Sizes: 1-5-10-25g • Call for 100-250-1000g pilot plant scale up

Spiro Compounds [3.5]

6-Oxa-2-azaspiro[3.5]nonane hemioxalate

On Stock

320,00 € 100mg

AS17966-C

7-Oxa-2-azaspiro[3.5]nonane HCl

On Stock

132,00 € 250mg

AS17438-B

7-Thia-2-azaspiro[3.5]nonane hemioxalate

On Stock

420,00 € 100mg

AS18102

7-Thia-2-azaspiro[3.5]nonane 7,7-dioxidehemioxalate

On Stock

360,00 € 100mg

AS56340

5-Azaspiro[3.5]nonane HCl

On Stock

360,00 € 100mg

AS17718-B

5-Boc-5-azaspiro[3.5]nonane-2-one

On Stock

254,00 € 100mg

AS57073

5-Boc-5-azaspiro[3.5]nonane-8-one

On Stock

1298,00 € 1g

AS16993

2-Oxa-5-azaspiro[3.5]nonane hemioxalate

On Stock

340,00 € 100mg

AS6086-C

5-Boc-2-oxa-5-azaspiro[3.5]nonane

CALL

1385,00 € 1g

AS52047

2,8-Dioxa-5-azaspiro[3.5]nonanehemioxalate

On Stock

372,00 € 100mg

AS52034-B

5-Boc-2,8-dioxa-5-azaspiro[3.5]nonane

CALL

1337,00 € 250mg

AS52046

8-Oxa-5-azaspiro[3.5]nonane hemioxalate

On Stock

420,00 € 100mg

AS18215

8-Oxa-2-thia-5-azaspiro[3.5]nonaneoxalate

On Stock

791,00 € 250mg

AS12921

5-Boc-8-oxa-2-thia-5-azaspiro[3.5]nonane

CALL

1455,00 € 250mg

AS12922

6-Azaspiro[3.5]nonane HCl

On Stock

300,00 € 100mg

AS17884

6-Azaspiro[3.5]nonan-5-one

On Stock

371,00 € 1g

AS77813

6-Boc-6-azaspiro[3.5]nonane-2-one

On Stock

376,00 € 250mg

AS17940

6-Boc-6-azaspiro[3.5]nonan-2-ol

On Stock

420,00 € 250mg

AS55504

6-Boc-1-amino-6-azaspiro[3.5]nonane

On Stock

688,00 € 100mg

AS56201

6-Boc-2-amino-6-azaspiro[3.5]nonane

On Stock

385,00 € 100mg

AS57549

1-Oxa-6-azaspiro[3.5]nonane hemioxalate

On Stock

478,00 € 250mg

AS52025-B

6-Boc-2-oxa-6-azaspiro[3.5]nonane

On Stock

320,00 € 250mg

AS6109

6-Boc-2,9-dioxa-6-azaspiro[3.5]nonane

On Stock

420,00 € 250mg

AS51791

7-Azaspiro[3.5]nonane HCl

On Stock

220,00 € 100mg

AS17773

Page 11: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

Activate Scientifi c · Am Mitterweg 12 · D-83209 Prien · Germany · Tel: +49 (0) 8051-965166021A The Maltings · Roydon Road · Stanstead Abbotts · Hertfordshire SG12 8HG · UK · Tel: +44 (0) 1279843244

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11

Chemistry Services for Drug Discovery www.activate-scientifi c.com

Spiro Compounds [3.5]

7-Boc-7-azaspiro[3.5]nonane-1-one

On Stock

240,00 € 250mg

AS52017

7-Boc-7-azaspiro[3.5]nonan-1-ol

CALL

985,00 € 1g

AS16073

7-Boc-1-amino-7-azaspiro[3.5]nonane

On Stock

458,00 € 250mg

AS51091

2-Fluoro-7-azaspiro[3.5]nonane HCl

On Stock

288,00 € 100mg

AS57563

2,2-Difl uoro-7-azaspiro[3.5]nonane HCl

On Stock

370,00 € 250mg

AS18110

7-Azaspiro[3.5]nonan-2-one HCl

On Stock

426,00 € 250mg

AS42947

7-Azaspiro[3.5]nonan-2-ol HCl

On Stock

328,00 € 250mg

AS57372

7-Boc-7-azaspiro[3.5]nonane-2-one

On Stock

95,00 € 1g

AS3577

7-Boc-7-azaspiro[3.5]nonane-2-ol

On Stock

265,00 € 1g

AS16873

7-Boc-7-azaspiro[3.5]nonane-2-methanol

On Stock

200,00 € 250mg

AS18164

7-Boc-7-azaspiro[3.5]nonane-2-carboxylic acid

On Stock

288,00 € 1g

AS51715

7-Boc-2-amino-7-azaspiro[3.5]nonane

On Stock

200,00 € 250mg

AS51668

7-Boc-7-azaspiro[3.5]nonane-2-methanamine

On Stock

380,00 € 250mg

AS51669

2-(Boc-amino)-7-azaspiro[3.5]nonane

On Stock

252,00 € 250mg

AS37413

2-Methyl-7-azaspiro[3.5]nonan-2-ol HCl

On Stock

284,00 € 250mg

AS55994-B

2-Amino-7-methyl-7-azaspiro[3.5]nonane

On Stock

478,00 € 250mg

AS52035

7-Methyl-7-azaspiro[3.5]nonane-2-methanol

On Stock

296,00 € 1g

AS56065

1-Oxa-7-azaspiro[3.5]nonane oxalate

On Stock

235,00 € 1g

AS12226-B

7-Boc-1-oxa-7-azaspiro[3.5]nonane

On Stock

245,00 € 1g

AS51900

7-Boc-1-oxa-7-azaspiro[3.5]nonane-3-one

On Stock

480,00 € 100mg

AS52056

7-Boc-1-oxa-7-azaspiro[3.5]nonane-2-methanamine

CALL

2235,00 € 1g

AS52061

7-Boc-1-oxa-7-azaspiro[3.5]nonane-2-methanol

On Stock

695,00 € 1g

AS52062

2-Oxa-7-azaspiro[3.5]nonane hemioxalate

On Stock

176,00 € 250mg

AS6026-B

7-Boc-2-oxa-7-azaspiro[3.5]nonane

On Stock

240,00 € 250mg

AS51841

Page 12: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

Chemistry Services for Drug Discovery www.activate-scientifi c.com

12

Standard Pack Sizes: 1-5-10-25g • Call for 100-250-1000g pilot plant scale up

Spiro Compounds [3.5]

1-Boc-1,6-diazaspiro[3.5]nonane

On Stock

290,00 € 100mg

AS17935

6-Boc-1,6-diazaspiro[3.5]nonane

On Stock

350,00 € 100mg

AS51770-A

1-Boc-1,7-diazaspiro[3.5]nonane

On Stock

718,00 € 250mg

AS51989

7-Boc-1,7-diazaspiro[3.5]nonane

On Stock

250,00 € 250mg

AS51772-A

7-Boc-1,7-diazaspiro[3.5]nonane-2-one

On Stock

240,00 € 250mg

AS17920

2-Boc-2,5-diazaspiro[3.5]nonane

On Stock

352,00 € 250mg

AS13115

5-Boc-2,5-diazaspiro[3.5]nonane

CALL

592,00 € 250mg

AS51774

5-Boc-8-oxa-2,5-diazaspiro[3.5]nonaneoxalate

CALL

1455,00 € 250mg

AS12925

2-Boc-8-oxa-2,5-diazaspiro[3.5]nonaneoxalate

CALL

1455,00 € 250mg

AS12924

6-Boc-2,6-diazaspiro[3.5]nonane HCl

On Stock

307,00 € 250mg

AS51771-B

2-Boc-2,6-diazaspiro[3.5]nonanehemioxalate

On Stock

476,00 € 250mg

AS51784-C

2-Boc-2,6-diazaspiro[3.5]nonan-7,9-dione

On Stock

280,00 € 100mg

AS12744

2-Boc-2,7-diazaspiro[3.5]nonane

On Stock

265,00 € 1g

AS51111

2,7-Diazaspiro[3.5]nonan-1-one HCl

On Stock

241,00 € 250mg

AS56983

7-Boc-2,7-diazaspiro[3.5]nonane-1-one

On Stock

235,00 € 250mg

AS38709

2-Methyl-2,7-diazaspiro[3.5]nonane

On Stock

300,00 € 250mg

AS38846

7-Methyl-2,7-diazaspiro[3.5]nonane diHCl

On Stock

536,00 € 250mg

AS42401

2-Boc-5-oxa-2,8-diazaspiro[3.5]nonane

On Stock

765,00 € 250mg

AS9732

8-Boc-5-oxa-2,8-diazaspiro[3.5]nonane

On Stock

552,00 € 250mg

AS9733

5-Boc-5,8-diazaspiro[3.5]nonane

On Stock

592,00 € 250mg

AS55799

8-Boc-5,8-diazaspiro[3.5]nonane

On Stock

254,00 € 100mg

AS56910

8-Boc-2-oxa-5,8-diazaspiro[3.5]nonane

On Stock

542,00 € 100mg

AS52058

2-oxa-5,8-diaza-spiro[3.5]nonane diHCl

CALL

1150,00 € 250mg

AS52036

8-Boc-2-oxa-5,8-diazaspiro[3.5]nonane-6-one

CALL

1478,00 € 1g

AS9735

Page 13: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

Activate Scientifi c · Am Mitterweg 12 · D-83209 Prien · Germany · Tel: +49 (0) 8051-965166021A The Maltings · Roydon Road · Stanstead Abbotts · Hertfordshire SG12 8HG · UK · Tel: +44 (0) 1279843244

www.activate-scientifi c.com · info@activate-scientifi c.com · info-uk@activate-scientifi c.com

13

Chemistry Services for Drug Discovery www.activate-scientifi c.com

Spiro Compounds [4.4]-[4.5]

1-Oxaspiro[4.4]nonan-6-one

CALL

788,00 € 250mg

AS52027

1-Oxaspiro[4.4]nonan-6-amine HCl

CALL

1372,00 € 1g

AS52026

6-Bromo-1,4-dioxaspiro[4.4]nonane

CALL

1850,00 € 5g

AS51582

7-Oxa-1-azaspiro[4.4]nonane HCl

On Stock

227,00 € 100mg

AS43803

2-Azaspiro[4.4]nonane hemioxalate

On Stock

290,00 € 250mg

AS17565-C

2-Boc-2-azaspiro[4.4]nonane-7-one

On Stock

858,00 € 250mg

AS55811

2-Boc-7-amino-2-azaspiro[4.4]nonane

On Stock

1420,00 € 1g

AS63181

2-Boc-7-(aminomethyl)-2-azaspiro[4.4]nonane

CALL

1420,00 € 1g

AS63180

1-Oxa-7-azaspiro[4.4]nonane HCl

On Stock

206,00 € 100mg

AS56284-B

7-Boc-1-oxa-7-azaspiro[4.4]nonane-3-one

On Stock

352,00 € 250mg

AS51132

7-Boc-1-oxa-7-azaspiro[4.4]nonan-3-ol

On Stock

985,00 € 1g

AS55535

2-Oxa-7-azaspiro[4.4]nonane

On Stock

352,00 € 250mg

AS56677

1-Boc-1,7-diazaspiro[4.4]nonane

On Stock

290,00 € 100mg

AS51769

7-Boc-1,7-diazaspiro[4.4]nonane

On Stock

295,00 € 100mg

AS51768

1,7-Diazaspiro[4.4]nonan-2-one TFA

On Stock

420,00 € 100mg

AS55983

7-Boc-1,7-diazaspiro[4.4]nonane-2-one

On Stock

320,00 € 100mg

AS51717

6-Boc-2,6-diazaspiro[4.4]nonan-1-one

On Stock

243,00 € 250mg

AS13201

2-Boc-2,7-diazaspiro[4.4]nonane

On Stock

102,00 € 250mg

AS51106-A

2,7-Diazaspiro[4.4]nonan-1-one HCl

On Stock

352,00 € 250mg

AS55876

2,7-Diazaspiro[4.4]nonan-3-one HCl

On Stock

446,00 € 100mg

AS56678

2-Boc-2,7-diazaspiro[4.4]nonane-6-one

On Stock

380,00 € 250mg

AS16334

2-Boc-2,7-diazaspiro[4.4]nonane-8-one

On Stock

306,00 € 250mg

AS57015

2-Methyl-2,7-diazaspiro[4.4]nonane diHCl

On Stock

326,00 € 250mg

AS42267

1-Azaspiro[4.5]-decane-2,8-dione

On Stock

206,00 € 250mg

AS55814

Page 14: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

Chemistry Services for Drug Discovery www.activate-scientifi c.com

14

Standard Pack Sizes: 1-5-10-25g • Call for 100-250-1000g pilot plant scale up

Spiro Compounds [4.5]

1-Oxaspiro[4.5]decan-8-one

On Stock

785,00 € 1g

AS2869

2-Oxaspiro[4.5]decan-8-one

On Stock

464,00 € 100mg

AS56074

8-Oxa-1-azaspiro[4.5]decane

On Stock

300,00 € 100mg

AS17848

2-Azaspiro[4.5]decane

On Stock

527,00 € 1g

AS78323

2-Boc-2-azaspiro[4.5]decane-6-amine

On Stock

825,00 € 250mg

AS55667

2-Boc-2-azaspiro[4.5]decan-7-one

On Stock

420,00 € 100mg

AS55649

8,8-Difl uoro-2-azaspiro[4.5]decane HCl

On Stock

254,00 € 100mg

AS57945

2-Azaspiro[4.5]decane-8-carboxylic acid

CALL

1380,00 € 1g

AS63184

2-Azaspiro[4.5]decan-8-amine

CALL

1240,00 € 1g

AS63185

2-Boc-2-azaspiro[4.5]decan-8-one

On Stock

323,00 € 100mg

AS56283

2-Boc-2-azaspiro[4.5]decane-8-amine

On Stock

446,00 € 100mg

AS55542

2-Methyl-2-azaspiro[4.5]decan-8-amineHCl

CALL

1360,00 € 1g

AS63182

7-Oxa-2-azaspiro[4.5]decane hemioxalate

On Stock

365,00 € 250mg

AS57863

8-Oxa-2-azaspiro[4.5]decane HCl

On Stock

285,00 € 1g

AS51895-B

2-Boc-8-oxa-2-azaspiro[4.5]decane

On Stock

465,00 € 1g

AS63186

8-Oxa-2-azaspiro[4.5]decan-3-one

On Stock

385,00 € 1g

AS17290

7-Azaspiro[4.5]decane

On Stock

627,00 € 1g

AS78326

1,4-Dioxa-7-azaspiro[4.5]decane

On Stock

235,00 € 250mg

AS17359

7-Boc-1-oxa-7-azaspiro[4.5]decan-3-one

On Stock

420,00 € 250mg

AS16351

7-Boc-1-oxa-7-azaspiro[4.5]decane-3-ol

CALL

415,00 € 250mg

AS56512

7-Boc-1-oxa-7-azaspiro[4.5]decane-3-methanamine

On Stock

428,00 € 100mg

AS55770

2-Oxa-7-azaspiro[4.5]decane HCl

On Stock

456,00 € 250mg

AS39544

8-Boc-8-azaspiro[4.5]decan-1-one

On Stock

252,00 € 250mg

AS55772

8-Boc-8-azaspiro[4.5]decan-2-one

On Stock

254,00 € 100mg

AS56954

Page 15: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

Activate Scientifi c · Am Mitterweg 12 · D-83209 Prien · Germany · Tel: +49 (0) 8051-965166021A The Maltings · Roydon Road · Stanstead Abbotts · Hertfordshire SG12 8HG · UK · Tel: +44 (0) 1279843244

www.activate-scientifi c.com · info@activate-scientifi c.com · info-uk@activate-scientifi c.com

15

Chemistry Services for Drug Discovery www.activate-scientifi c.com

Spiro Compounds [4.5]

1,4-Dioxa-8-azaspiro[4.5]decane HCl

On Stock

39,00 € 5g

AS31782-B

1,4-Dioxa-8-azaspiro[4.5]decane-6-methanamine

On Stock

482,00 € 250mg

AS17630

1-Oxa-8-azaspiro[4.5]decane HCl

On Stock

158,00 € 250mg

AS51904

8-Boc-1-oxa-8-azaspiro[4.5]decan-2-one

On Stock

265,00 € 1g

AS55270

8-Boc-2-hydroxy-1-oxa-8-azaspiro[4.5]decane

On Stock

440,00 € 250mg

AS55493

8-Boc-2-(aminomethyl)-1-oxa-8-azaspiro[4.5]decane

On Stock

448,00 € 100mg

AS55640

1-Oxa-8-azaspiro[4.5]decan-3-one HCl

On Stock

184,00 € 250mg

AS38009

8-Boc-1-oxa-8-azaspiro[4.5]decan-3-one

On Stock

281,00 € 250mg

AS16350

8-Boc-1-oxa-8-azaspiro[4.5]decan-3-ol

On Stock

352,00 € 250mg

AS51808

2-Oxa-8-azaspiro[4.5]decane oxalate

On Stock

336,00 € 250mg

AS41042

8-Boc-2-oxa-8-azaspiro[4.5]decan-3-one

On Stock

255,00 € 250mg

AS57145

1,4-Dioxaspiro[4.5]decane

On Stock

136,00 € 1g

AS29155

1,4-Dioxaspiro[4.5]decan-7-one

On Stock

187,00 € 1g

AS74597

1,4-Dioxaspiro[4.5]decan-7-ol

On Stock

326,00 € 1g

AS74576

1,4-Dioxaspiro[4.5]decan-7-amine

CALL

619,00 € 1g

AS74756

1,4-Dioxaspiro[4.5]dec-7-en-7-boronicacid pinacol ester

On Stock

649,00 € 250mg

AS15332

7-Methyl-1,4-dioxaspiro[4.5]decan-8-one

On Stock

644,00 € 5g

AS29351

1,4-Dioxaspiro[4.5]decan-8-ol

On Stock

44,00 € 1g

AS39846

1,4-Dioxaspiro[4.5]decane-8-methanol

On Stock

325,00 € 1g

AS64159

1,4-Dioxaspiro[4,5]dec-7-en-8-boronicacid pinacol ester

On Stock

175,00 € 1g

AS31921

8-Amino-1,4-dioxaspiro[4.5]decane-8-carboxylic acid

On Stock

765,00 € 5g

AS24554

8-(Boc-amino)-1,4-dioxaspiro[4.5]decane-8-carboxylic acid

On Stock

324,00 € 1g

AS27567

6,10-Dioxaspiro[4.5]decane-7,9-dione

On Stock

202,00 € 250mg

AS44043

1-Boc-1,7-diazaspiro[4.5]decane

On Stock

444,00 € 250mg

AS52059

Page 16: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

Chemistry Services for Drug Discovery www.activate-scientifi c.com

16

Standard Pack Sizes: 1-5-10-25g • Call for 100-250-1000g pilot plant scale up

Spiro Compounds [4.5]

7-Boc-1,7-diazaspiro[4.5]decane

On Stock

558,00 € 250mg

AS51775

1-Boc-1,8-diazaspiro[4.5]decane HCl

On Stock

420,00 € 250mg

AS51785-B

8-Boc-1,8-diazaspiro[4.5]decane

On Stock

480,00 € 250mg

AS51773-A

8-Boc-1,8-diazaspiro[4.5]decan-2-one

On Stock

320,00 € 250mg

AS72061

2-Boc-2,6-diazaspiro[4.5]decane

On Stock

457,00 € 100mg

AS56282

6-Boc-2,6-diazaspiro[4.5]decane

On Stock

465,00 € 250mg

AS51779

2-Boc-8-oxa-2,6-diazaspiro[4.5]decan-7-one

On Stock

395,00 € 100mg

AS18073

2-Boc-2,7-diazaspiro[4.5]decane

On Stock

283,00 € 250mg

AS16339

7-Boc-2,7-diazaspiro[4.5]decane

On Stock

800,00 € 1g

AS51107

2-Boc-2,7-diazaspiro[4.5]decane oxalate

On Stock

352,00 € 250mg

AS17828

7-Boc-2,7-diazaspiro[4.5]decan-1-one

On Stock

332,00 € 250mg

AS13203

2,7-Diazaspiro[4.5]decan-1-one HCl

On Stock

359,00 € 1g

AS16335-B

2,7-Diazaspiro[4.5]decan-3-one

On Stock

335,00 € 250mg

AS41982

7-Boc-2,7-diazaspiro[4.5]decan-3-one

On Stock

525,00 € 250mg

AS42457

2-Boc-2,7-diazaspiro[4.5]decan-6-one

On Stock

424,00 € 250mg

AS16340

2-Boc-2,8-diazaspiro[4.5]decane

On Stock

237,00 € 250mg

AS51116

8-Boc-2,8-diazaspiro[4.5]decane

On Stock

235,00 € 250mg

AS21274-A

8-Boc-2,8-diazaspiro[4.5]decan-1-one

On Stock

269,00 € 1g

AS13147

2,8-Diazaspiro[4.5]decan-1-one HCl

On Stock

180,00 € 250mg

AS34519

2,8-Diazaspiro[4.5]decan-3-one

On Stock

224,00 € 250mg

AS51117

8-Boc-2,8-diazaspiro[4.5]decan-3-one

On Stock

192,00 € 250mg

AS51133

2,8-Diazaspiro[4.5]decane-1,3-dione HCl

On Stock

252,00 € 250mg

AS56528

9-Boc-6-oxa-2,9-diazaspiro[4.5]decane

On Stock

223,00 € 100mg

AS57050

7-Boc-2,4-dioxo-1-oxa-3,7-diazaspiro[4.5]decane

On Stock

332,00 € 100mg

AS57944

Page 17: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

Activate Scientifi c · Am Mitterweg 12 · D-83209 Prien · Germany · Tel: +49 (0) 8051-965166021A The Maltings · Roydon Road · Stanstead Abbotts · Hertfordshire SG12 8HG · UK · Tel: +44 (0) 1279843244

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17

Chemistry Services for Drug Discovery www.activate-scientifi c.com

Spiro Compounds [4.5]-[4.6]-[5.5]

7-Boc-2,4-Dioxo-1,3,7-triazaspiro[4.5]decane

On Stock

263,00 € 250mg

AS57922

1,3,8-Triazaspiro[4.5]decane-2,4-dione

On Stock

132,00 € 1g

AS22811

1-Methyl-1,3,8-triazaspiro[4.5]decan-4-one

On Stock

313,00 € 100mg

AS57568

8-Boc-2,4,8-triazaspiro[4.5]decane-1,3-dione

On Stock

105,00 € 1g

AS21695

2-Azaspiro[4.6]undecane

On Stock

278,00 € 250mg

AS18553

2-Azaspiro[4.6]undecan-3-one

On Stock

371,00 € 1g

AS77815

1-Boc-1-azaspiro[5.5]undecan-4-one

On Stock

250,00 € 250mg

AS28943

2-Boc-2-Azaspiro[5.5]undecane-9-one

On Stock

410,00 € 250mg

AS55648

9-Oxa-2-azaspiro[5.5]undecane HCl

On Stock

467,00 € 1g

AS78159

2-Boc-9-oxa-2-azaspiro[5.5]undecane

On Stock

638,00 € 250mg

AS51893

9-Oxa-2-azaspiro[5.5]undecan-1-one

On Stock

278,00 € 1g

AS78497

3-Azaspiro[5.5]undecane HCl

On Stock

276,00 € 250mg

AS40752

3-Boc-3-azaspiro[5.5]undecan-7-one

On Stock

572,00 € 250mg

AS55773

3-Boc-3-azaspiro[5.5]undecan-9-one

On Stock

260,00 € 250mg

AS18269

9-Amino-3-Boc-3-azaspiro[5.5]undecane

On Stock

621,00 € 250mg

AS56285

4-Boc-4-azaspiro[5.5]undecane-9-carboxylic acid

On Stock

393,00 € 100mg

AS51680

9-Boc-2-oxa-9-azaspiro[5.5]undecane

On Stock

638,00 € 250mg

AS51892

3-Oxa-9-azaspiro[5.5]undecane

On Stock

401,00 € 250mg

AS55806

9-Boc-3-oxa-9-azaspiro[5.5]undecane

On Stock

352,00 € 250mg

AS51891

1-Boc-1,8-diazaspiro[5.5]undecane

On Stock

243,00 € 250mg

AS51781

8-Boc-1,8-Diazaspiro[5.5]undecane

On Stock

361,00 € 100mg

AS51778

8-Boc-3-oxa-1,8-diazaspiro[5.5]undecane-2-one

On Stock

765,00 € 250mg

AS18059

1-Boc-4-oxa-1,8-diazaspiro[5.5]undecane

On Stock

867,00 € 250mg

AS9729

8-Boc-4-oxa-1,8-diazaspiro[5.5]undecane

CALL

652,00 € 250mg

AS9730

Page 18: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

Chemistry Services for Drug Discovery www.activate-scientifi c.com

18

Standard Pack Sizes: 1-5-10-25g • Call for 100-250-1000g pilot plant scale up

Spiro Compounds [5.5]

1-Boc-1,9-diazaspiro[5.5]undecane

On Stock

360,00 € 100mg

AS51780

9-Boc-1,9-diazaspiro[5.5]undecane

On Stock

290,00 € 100mg

AS51776

1,9-Diazaspiro[5.5]undecan-2-one HCl

On Stock

254,00 € 100mg

AS57547

9-Boc-4-oxa-1,9-diazaspiro[5.5]undecane

On Stock

592,00 € 250mg

AS55769

9-Boc-3-oxa-1,9-diazaspiro[5.5]undecane-2-one

On Stock

394,00 € 250mg

AS18209

7-Boc-2,7-diazaspiro[5.5]undecan-1-one

On Stock

294,00 € 250mg

AS13204

2-Boc-2,8-diazaspiro[5.5]undecane

On Stock

478,00 € 250mg

AS51109

2,8-Diazaspiro[5.5]undecane-1-one

On Stock

293,00 € 250mg

AS14825

8-Boc-2,8-diazaspiro[5.5]undecan-1-one

On Stock

249,00 € 250mg

AS13207

2-Boc-2,9-diazaspiro[5.5]undecane

On Stock

420,00 € 250mg

AS51777

9-Boc-2,9-diazaspiro[5.5]undecane

On Stock

290,00 € 250mg

AS3540

2,9-diBoc-2,9-diazaspiro[5.5]undecane

On Stock

433,00 € 1g

AS14575

2,9-Diazaspiro[5.5]undecan-1-one HCl

On Stock

222,00 € 250mg

AS13169

2-Boc-2,9-diazaspiro[5.5]undecan-1-one

On Stock

1650,00 € 1g

AS13172

9-Boc-2,9-diazaspiro[5.5]undecan-1-one

On Stock

266,00 € 250mg

AS16343

9-Boc-3-oxo-2,9-diazaspiro[5.5]undecane

On Stock

572,00 € 250mg

AS56514

9-Boc-2,9-diazaspiro[5.5]undecane-3,5-dione

On Stock

220,00 € 100mg

AS17703

9-Methyl-2,9-diazaspiro[5.5]undecane

On Stock

467,00 € 1g

AS78187

9-Methyl-2,9-diazaspiro[5.5]undecan-1-one

On Stock

371,00 € 1g

AS77849

3-Boc-3,9-diazaspiro[5.5]undecane HCl

On Stock

166,00 € 250mg

AS51108-B

1-Oxa-3,9-diazaspiro[5.5]undecan-2-oneHCl

On Stock

509,00 € 250mg

AS42576

9-Boc-1-oxa-3,9-diazaspiro[5.5]undecane-2-one

On Stock

456,00 € 250mg

AS42641

8-Boc-1-oxa-4,8-diazaspiro[5.5]undecane

On Stock

282,00 € 250mg

AS51894

4-Boc-1-oxa-4,9-diazaspiro[5.5]undecane

On Stock

807,00 € 250mg

AS18555

Page 19: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

Activate Scientifi c · Am Mitterweg 12 · D-83209 Prien · Germany · Tel: +49 (0) 8051-965166021A The Maltings · Roydon Road · Stanstead Abbotts · Hertfordshire SG12 8HG · UK · Tel: +44 (0) 1279843244

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19

Chemistry Services for Drug Discovery www.activate-scientifi c.com

Bicyclic Rings [1.1.1]-[2.2.1]

Bicyclo[1.1.1]pentan-1-amine HCl

On Stock

288,00 € 100mg

AS56976

1-(Boc-amino)-bicyclo[1.1.1]pentan-3-amine

On Stock

385,00 € 100mg

AS57291

1,1‘-(Bicyclo[1.1.1]pentane-1,3-diyl)-diethanone

On Stock

360,00 € 250mg

AS55665

Bicyclo[1.1.1]pentane-1,3-dicarboxylic acid

On Stock

206,00 € 250mg

AS55766

Dimethyl bicyclo[1.1.1]pentane-1,3-dicarboxylate

On Stock

284,00 € 250mg

AS55659

3-(Hydroxymethyl)bicyclo[1.1.1]pentane-1-carbonitrile

On Stock

314,00 € 100mg

AS56977

Methyl 3-(hydroxymethyl)bicyclo[1.1.1]pentane-1-carboxylate

On Stock

558,00 € 250mg

AS55923

3-(Methoxycarbonyl)bicyclo[1.1.1]pentane-1-carboxylic acid

On Stock

280,00 € 250mg

AS56052

Methyl 3-cyanobicyclo[1.1.1]pentane-1-carboxylate

On Stock

985,00 € 250mg

AS55926

Bicyclo[1.1.1]pentane-1,3-diamine diHCl

On Stock

635,00 € 100mg

AS56299

1,3-Bis(Cbz-amino)bicyclo[1.1.1]pentane

On Stock

467,00 € 100mg

AS55928

Methyl 3-aminobicyclo[1.1.1]pentane-1-carboxylate HCl

On Stock

360,00 € 100mg

AS55808

3-(Boc-amino)bicyclo[1.1.1]pentane-1-carboxylic acid

On Stock

864,00 € 250mg

AS55925

Methyl 3-(Boc-amino)bicyclo[1.1.1]pentane-1-carboxylate

On Stock

330,00 € 100mg

AS55924

N1,N3-dimethylbicyclo[1.1.1]pentane-1,3-diamine diHCl

On Stock

999,00 € 100mg

AS55927

2-Azabicyclo[2.1.1]hexane HCl

On Stock

1210,00 € 1g

AS55629

1,4-Diazabicyclo[2.1.1]hexane

On Stock

254,00 € 250mg

AS42565

(1R,4S,5S)-rel-2-Boc-2-azabicyclo[2.1.1]hexane-5-carboxylic acid

On Stock

1029,00 € 250mg

AS56532

(1R,4S,5S)-rel-2-Boc-2-azabicyclo[2.1.1]hexan-5-amine

On Stock

550,00 € 100mg

AS56533

Dimethyl bicyclo[2.2.1]heptane-1,4-dicarboxylate

On Stock

352,00 € 250mg

AS56006

Methyl 4-aminobicyclo[2.2.1]heptane-1-carboxylate

On Stock

298,00 € 100mg

AS57290

Bicyclo[2.2.1]heptane-1,4-diamine diHCl

On Stock

328,00 € 250mg

AS57368

2-Formylbicyclo[2.2.1]heptane

CALL

120,00 € 1g

AS34768

Ethyl (1R,2S,3R,4S)-rel-3-Aminobicyclo-[2.2.1]heptane-2-carboxylate

CALL

836,00 € 1g

AS27599

Page 20: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

Chemistry Services for Drug Discovery www.activate-scientifi c.com

20

Standard Pack Sizes: 1-5-10-25g • Call for 100-250-1000g pilot plant scale up

Bicyclic Rings [2.2.1]

5-Aminobicyclo[2.2.1]heptan-2-ol HCl

On Stock

288,00 € 100mg

AS57401

6-Aminobicyclo[2.2.1]heptan-2-ol HCl

On Stock

288,00 € 100mg

AS57748

2-Boc-bicyclo[2.2.1]hept-5-ene

On Stock

152,00 € 5g

AS23051

Bicyclo[2.2.1]hept-5-ene-2-carboxylic acid

On Stock

132,00 € 25g

AS40557

2-(Methylamine)-bicyclo[2.2.1]hept-5-ene

CALL

271,00 € 5g

AS28983

(1S,4S)-1,7,7-Trimethylbicyclo[2.2.1]heptan-2-one

On Stock

128,00 € 25g

AS27819-1S4S

2-Azabicyclo[2.2.1]heptane

On Stock

311,00 € 250mg

AS51925

2-Azabicyclo[2.2.1]hept-5-ene hemioxalate

On Stock

248,00 € 1g

AS56929

2-Boc-2-azabicyclo[2.2.1]hept-5-ene

On Stock

497,00 € 5g

AS29634

3-Oxo-2-azabicyclo[2.2.1]hept-5-ene

On Stock

28,00 € 5g

AS21031-RAC

(1R,4S)-3-Oxo-2-azabicyclo[2.2.1]hept-5-ene

On Stock

105,00 € 1g

AS21031-1R4S

(1S,4R)-3-Oxo-2-azabicyclo[2.2.1]hept-5-ene

On Stock

210,00 € 1g

AS21031-1S4R

2-Boc-3-oxo-2-azabicyclo[2.2.1]heptane

CALL

1360,00 € 1g

AS14342

2-Boc-2-azabicyclo[2.2.1]heptan-5-one

On Stock

254,00 € 250mg

AS44298

2-Azabicyclo[2.2.1]heptan-5-ol HCl

On Stock

288,00 € 100mg

AS56930

2-Boc-2-azabicyclo[2.2.1]heptan-5-ol

On Stock

255,00 € 250mg

AS56889

(1S,3S,4S,5S)-rel-2-Boc-5-hydroxy-2-aza-bicyclo[2.2.1]heptane-3-carboxylic acid

On Stock

1221,00 € 250mg

AS55970

2-Azabicyclo[2.2.1]heptan-6-ol HCl

On Stock

332,00 € 100mg

AS56931

2-Boc-2-azabicyclo[2.2.1]heptan-6-one

On Stock

328,00 € 250mg

AS57766

2-Boc-2-azabicyclo[2.2.1]heptan-6-ol

On Stock

255,00 € 250mg

AS57961

2-Boc-2-azabicyclo[2.2.1]heptan-7-amine

On Stock

248,00 € 100mg

AS55639

7-(Boc-amino)-2-azabicyclo[2.2.1]heptane

On Stock

546,00 € 100mg

AS55857

5-Azabicyclo[2.2.1]heptan-2-one

On Stock

476,00 € 1g

AS72029-ARAC

5-Boc-5-azabicyclo[2.2.1]heptan-2-one

On Stock

295,00 € 100mg

AS56145

Page 21: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

Activate Scientifi c · Am Mitterweg 12 · D-83209 Prien · Germany · Tel: +49 (0) 8051-965166021A The Maltings · Roydon Road · Stanstead Abbotts · Hertfordshire SG12 8HG · UK · Tel: +44 (0) 1279843244

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21

Chemistry Services for Drug Discovery www.activate-scientifi c.com

Bicyclic Rings [2.2.1]-[2.2.2]

7-Azabicyclo[2.2.1]heptane HCl

On Stock

232,00 € 250mg

AS12713

7-Boc-7-azabicyclo[2.2.1]heptan-2-one

On Stock

252,00 € 250mg

AS55789

(1R,2S,4S)-rel-7-Boc-7-azabicyclo[2.2.1]heptan-2-ol

CALL

558,00 € 250mg

AS55788

(1R,2R,4S)-rel-7-Boc-7-azabicyclo[2.2.1]heptan-2-ol

On Stock

301,00 € 100mg

AS56903

Ethyl 7-azabicyclo[2.2.1]heptane-2-carboxylate HCl

On Stock

564,00 € 100mg

AS55844

Methyl 7-Boc-7-azabicyclo[2.2.1]heptene-2-carboxylate

On Stock

521,00 € 250mg

AS14866

(1R,2R,4S)-rel-7-Boc-7-azabicyclo[2.2.1]heptan-2-amine

On Stock

518,00 € 100mg

AS55858

endo-7-Boc-7-azabicyclo[2.2.1]heptan-2-amine

On Stock

1640,00 € 1g

AS13389

2-Boc-2,5-diazabicyclo[2.2.1]heptane

On Stock

285,00 € 1g

AS51792

(1S,4S)-2-Boc-2,5-diazabicyclo[2.2.1]heptane

On Stock

95,00 € 1g

AS40006-1S4S

(1R,4R)-2-Methyl-2,5-diazabicyclo[2.2.1]heptane diHBr

On Stock

200,00 € 250mg

AS12918-1R4R

(1S,4S)-5-Methyl-2,5-diazabicyclo[2.2.1]heptane diHBr

On Stock

229,00 € 1g

AS12530

Bicyclo[2.2.2]octane-1-carboxylic acid

On Stock

220,00 € 100mg

AS39546

Ethyl 4-hydroxybicyclo[2.2.2]octane-1-carboxylate

On Stock

389,00 € 100mg

AS56729

Methyl 4-hydroxybicyclo[2.2.2]octane-1-carboxylate

On Stock

370,00 € 250mg

AS28192

Methyl 4-(hydroxymethyl)bicyclo[2.2.2]octane-1-carboxylate

On Stock

456,00 € 250mg

AS37659

4-Fluorobicyclo[2.2.2]octane-1-carboxylic acid

On Stock

724,00 € 100mg

AS56728

4-Fluorobicyclo[2.2.2]octan-1-amine

On Stock

1050,00 € 100mg

AS56005

4-Aminobicyclo[2.2.2]octane-1-carboxylicacid HCl

On Stock

367,00 € 250mg

AS41950

4-Aminobicyclo[2.2.2]octane-1-carbonitrileHCl

CALL

331,00 € 100mg

AS43437

Methyl 4-aminobicyclo[2.2.2]octane-1-carboxylate

On Stock

230,00 € 250mg

AS37136

4-(Boc-amino)-bicyclo[2.2.2]octane-1-carboxylic acid

On Stock

313,00 € 250mg

AS43438

Bicyclo[2.2.2]octane-1,4-dicarboxylic acid

On Stock

187,00 € 250mg

AS57289

Bicyclo[2.2.2]octane-1,4-diamine diHCl

On Stock

478,00 € 250mg

AS55972

Page 22: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

Chemistry Services for Drug Discovery www.activate-scientifi c.com

22

Standard Pack Sizes: 1-5-10-25g • Call for 100-250-1000g pilot plant scale up

Bicyclic Rings [2.2.2]

Bicyclo[2.2.2]oct-2-ene

CALL

601,00 € 250mg

AS9690

Bicyclo[2.2.2]octan-2-one

On Stock

219,00 € 250mg

AS42505

Bicyclo[2.2.2]octan-2-ol

On Stock

331,00 € 100mg

AS43959

Methyl trans-3-aminobicyclo[2.2.2]octane-2-carboxylate HCl

On Stock

490,00 € 250mg

AS56007

1-Azabicyclo[2.2.2]octane-4-carboxylicacid

On Stock

320,00 € 250mg

AS12182-A

1-Azabicyclo[2.2.2]octane-3-methanamine

On Stock

523,00 € 1g

AS17273

(1-Aza-bicyclo[2.2.2]oct-4-yl)methylamine

On Stock

350,00 € 250mg

AS18572

2-Azabicyclo[2.2.2]octane HCl

On Stock

284,00 € 250mg

AS51928

2-Azabicyclo[2.2.2]octan-3-one

On Stock

433,00 € 1g

AS55426

Methyl 3-oxo-2-azabicyclo[2.2.2]octane-1-carboxylate

CALL

418,00 € 100mg

AS66042

(3R)-2-Azabicyclo[2.2.2]octane-3-carboxylic acid

On Stock

410,00 € 100mg

AS56523

(3S)-2-Azabicyclo[2.2.2]octane-3-carboxylic acid

On Stock

300,00 € 100mg

AS57635

4-(Boc-amino)-1-formyl-2-oxabicyclo[2.2.2]octane

On Stock

385,00 € 100mg

AS57288

2-Boc-2-azabicyclo[2.2.2]octan-5-one

On Stock

290,00 € 250mg

AS51952

(1S,4S)-2-Boc-2-azabicyclo[2.2.2]octan-5-one

On Stock

385,00 € 100mg

AS57717-1S4S

(1R,4R)-2-Boc-2-azabicyclo[2.2.2]octan-5-one

On Stock

385,00 € 100mg

AS57718-1R4R

2-Boc-2-azabicyclo[2.2.2]octan-5-ol

On Stock

288,00 € 100mg

AS57343

2-Boc-2-azabicyclo[2.2.2]octane-6-one

On Stock

280,00 € 100mg

AS55603

2-Azabicyclo[2.2.2]octan-6-ol HCl

On Stock

248,00 € 100mg

AS55597

2-Boc-2-azabicyclo[2.2.2]octane-6-carboxylic acid

On Stock

564,00 € 100mg

AS55816

5-Azabicyclo[2.2.2]octan-2-onehemioxalate

On Stock

320,00 € 100mg

AS55661

2-Boc-(1R,4R)-2,5-diazabicyclo[2.2.2]octane

On Stock

2250,00 € 1g

AS3906-1R4R

2-Boc-(1S,4S)-2,5-diazabicyclo[2.2.2]octane

On Stock

2772,00 € 1g

AS3906-1S4S

2,5-Diazabicyclo[2.2.2]octane-3,6-dione

On Stock

310,00 € 250mg

AS26743

Page 23: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

Activate Scientifi c · Am Mitterweg 12 · D-83209 Prien · Germany · Tel: +49 (0) 8051-965166021A The Maltings · Roydon Road · Stanstead Abbotts · Hertfordshire SG12 8HG · UK · Tel: +44 (0) 1279843244

www.activate-scientifi c.com · info@activate-scientifi c.com · info-uk@activate-scientifi c.com

23

Chemistry Services for Drug Discovery www.activate-scientifi c.com

Bicyclic Rings [3.1.0]

2-(2,5-Diazabicyclo[2.2.2]octan-2-yl)-2-methylpropan-1-ol

On Stock

260,00 € 100mg

AS80359

(1R,3S,5R)-2-Boc-2-azabicyclo[3.1.0]hexane-3-carboxylic acid

On Stock

367,00 € 1g

AS44484

(1S,3S,5S)-2-azabicyclo[3.1.0]hexane-3-carboxylic acid TFA

On Stock

394,00 € 250mg

AS56206

(1S,3S,5S)-2-Boc-3-carbamoyl-2-azabicyclo[3.1.0]hexane

On Stock

151,00 € 250mg

AS38996

3-Azabicyclo[3.1.0]hexane HCl

On Stock

85,00 € 1g

AS12519

3-Azabicyclo[3.1.0]hexane-1-carboxylic acid HCl

On Stock

558,00 € 250mg

AS56204

3-Boc-3-azabicyclo[3.1.0]hexane-1-carboxylic acid

On Stock

200,00 € 250mg

AS56205

3-Azabicyclo[3.1.0]hexane-1-methanol HCl

On Stock

230,00 € 100mg

AS18415

1-(Boc-amino)-3-azabicyclo[3.1.0]hexane

On Stock

305,00 € 100mg

AS18076

1-Amino-3-Boc-3-azabicyclo[3.1.0]hexane

On Stock

240,00 € 100mg

AS56203

1-(Aminomethyl)-3-benzyl-3-aza-bicyclo[3.1.0]hexane

CALL

165,00 € 250mg

AS26357

(1R,2S,5S)-3-Azabicyclo[3.1.0]hexane-2-carboxylic acid

On Stock

565,00 € 250mg

AS3629

cis-(1S,2S,5R)-3-Azabicyclo[3.1.0]hexan-2-ylmethanol HCl

On Stock

333,00 € 100mg

AS57763-CIS

(1R,2S,5S)-3-Azabicyclo[3.1.0]hexane-2-methanol HCl

On Stock

290,00 € 100mg

AS3628

2-Cyano-3-azabicyclo[3.1.0]hexane

On Stock

220,00 € 100mg

AS17679

3-Oxabicyclo[3.1.0]hexane-2,4-dione

On Stock

39,00 € 1g

AS12902

6,6-Dimethyl-3-oxabicyclo[3.1.0]hexane-2,4-dione

On Stock

105,00 € 5g

AS24245

6-(Boc-amino)-3-azabicyclo[3.1.0]hexane

On Stock

395,00 € 250mg

AS34117

6,6-Difl uoro-3-azabicyclo[3.1.0]hexanehemioxalate

On Stock

248,00 € 100mg

AS51654

6,6-Dimethyl-3-azabicyclo[3.1.0]hexaneHCl

On Stock

355,00 € 1g

AS17342-B

6,6-Dimethyl-3-azabicyclo[3.1.0]hexane-2,4-dione

CALL

360,00 € 1g

AS19281

Ethyl 3-azabicyclo[3.1.0]hexane-6-carboxylate oxalate

On Stock

257,00 € 250mg

AS51944-BRAC

3-Boc-3-azabicyclo[3.1.0]hexane-6-carboxylic acid

On Stock

343,00 € 250mg

AS18475

endo-3-Boc-3-azabicyclo[3.1.0]hexane-6-carboxylic acid

On Stock

493,00 € 100mg

AS55771

Page 24: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

Chemistry Services for Drug Discovery www.activate-scientifi c.com

24

Standard Pack Sizes: 1-5-10-25g • Call for 100-250-1000g pilot plant scale up

Bicyclic Rings [3.1.0]-[3.1.1]

3-Azabicyclo[3.1.0]hexane-6-carboxamide

On Stock

494,00 € 250mg

AS17806

exo-3-Azabicyclo[3.1.0]hexan-6-ol HCl

On Stock

347,00 € 100mg

AS55655

exo-3-Azabicyclo[3.1.0]hexan-6-methanol

On Stock

254,00 € 250mg

AS3542

exo-3-Boc-3-azabicyclo[3.1.0]hexane-6-methanol

On Stock

295,00 € 250mg

AS12383

exo-6-Amino-3-Boc-3-azabicyclo[3.1.0]hexane

On Stock

294,00 € 1g

AS12411

exo-3-Boc-6-aminomethyl-3-azabicyclo[3.1.0]hexane

On Stock

276,00 € 250mg

AS12622

exo-3-Methyl-6-amino-3-azabicyclo[3.1.0]hexane

On Stock

856,00 € 250mg

AS12692

exo-6-(Boc-amino)-3-azabicyclo[3.1.0]hexane

On Stock

360,00 € 250mg

AS12404

exo-6-(Boc-aminomethyl)-3-azabicyclo[3.1.0]hexane

On Stock

380,00 € 250mg

AS12384

exo-3-Oxabicyclo[3.1.0]hexane-6-methanol

On Stock

284,00 € 250mg

AS55913

3-Oxabicyclo[3.1.0]hexane-6-carboxylicacid

On Stock

240,00 € 250mg

AS32068

exo-3-Oxabicyclo[3.1.0]hexane-6-carboxylic acid

On Stock

328,00 € 250mg

AS56967

trans-3-Oxabicyclo[3.1.0]hexane-6-aceticacid

On Stock

635,00 € 100mg

AS55949-TRANS

3-Boc-6-oxa-3-azabicyclo[3.1.0]hexane

On Stock

68,00 € 5g

AS40538

3-Boc-3,6-diazabicyclo[3.1.0]hexane

On Stock

374,00 € 250mg

AS38068

2-Azabicyclo[3.1.1]heptane-1-carboxylicacid HCl

On Stock

328,00 € 100mg

AS57693

2-Benzyl-2-azabicyclo[3.1.1]heptane-1-carboxylic acid

On Stock

467,00 € 100mg

AS56508

3-Azabicyclo[3.1.1]heptane

On Stock

2360,00 € 1g

AS18185

3-Azabicyclo[3.1.1]heptan-6-one HCl

On Stock

329,00 € 100mg

AS57099

3-Boc-3-azabicyclo[3.1.1]heptane-6-one

On Stock

484,00 € 250mg

AS17980

3-Benzyl-3-azabicyclo[3.1.1]heptan-6-one

CALL

625,00 € 250mg

AS17737

3-Cbz-3-azabicyclo[3.1.1]heptane-6-one

On Stock

1150,00 € 1g

AS55618

3-Azabicyclo[3.1.1]heptan-6-ol HCl

On Stock

320,00 € 100mg

AS17950

3-Boc-3-azabicyclo[3.1.1]heptane-6-ol

On Stock

290,00 € 100mg

AS17810

Page 25: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

Activate Scientifi c · Am Mitterweg 12 · D-83209 Prien · Germany · Tel: +49 (0) 8051-965166021A The Maltings · Roydon Road · Stanstead Abbotts · Hertfordshire SG12 8HG · UK · Tel: +44 (0) 1279843244

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25

Chemistry Services for Drug Discovery www.activate-scientifi c.com

Bicyclic Rings [3.1.1]-[3.2.0]

6-Hydroxymethyl-3-azabicyclo[3.1.1]

On Stock

563,00 € 250mg

AS18001

3-Benzyl-3-azabicyclo[3.1.1]heptan-6-amine

On Stock

360,00 € 100mg

AS55656

(3-Boc)-6-amino-3-azabicyclo[3.1.1]heptane

On Stock

360,00 € 100mg

AS18436

Endo-6-(boc-Amino)-3-azabicyclo[3.1.1]heptane

On Stock

485,00 € 100mg

AS57567

6-(Boc-amino)-3-azabicyclo[3.1.1]heptane

On Stock

482,00 € 100mg

AS56239

3-Boc-3-azabicyclo[3.1.1]heptane-6-carboxylic acid

On Stock

450,00 € 100mg

AS55138

Methyl 3-azabicyclo[3.1.1]heptane-6-carboxylate HCl

On Stock

845,00 € 250mg

AS18118

Methyl 3-Boc-3-azabicyclo[3.1.1]heptane-6-carboxylate

On Stock

380,00 € 100mg

AS18371

3-Boc-3-azabicyclo[3.1.1]heptane-6-carboxamide

On Stock

813,00 € 250mg

AS18211

6-Oxabicyclo[3.1.0]hex-3-ene

CALL

1063,00 € 1g

AS9127

6-Oxa-3-azabicyclo[3.1.1]heptane tosylate

On Stock

390,00 € 250mg

AS56537

6-Oxa-7-azabicyclo[3.1.1]heptane

On Stock

312,00 € 100mg

AS17946

3-Boc-3,6-diazabicyclo[3.1.1]heptane

On Stock

1365,00 € 1g

AS9769

3-Azabicyclo[3.2.0]heptane HCl

CALL

720,00 € 250mg

AS56480

3-Boc-3-azabicyclo[3.2.0]heptan-6-one

On Stock

220,00 € 100mg

AS17791

3-Tosyl-3-azabicyclo[3.2.0]heptan-6-one

On Stock

154,00 € 250mg

AS41410

(1S,5R)(3-Boc)-1,5-dimethyl-6-oxo-3-azabicyclo[3.2.0]heptane

On Stock

965,00 € 1g

AS16979-1S5R

3-Boc-3-azabicyclo[3.2.0]heptan-6-ol

On Stock

243,00 € 250mg

AS27713

3-Boc-3-azabicyclo[3.2.0]heptan-6-amine

On Stock

290,00 € 100mg

AS56337

6-Boc-6-azabicyclo[3.2.0]heptan-4-one

CALL

947,00 € 250mg

AS56096

cis-6-Azabicyclo[3.2.0]heptan-7-one

On Stock

255,00 € 1g

AS23705-CIS

exo-6-Boc-6-azabicyclo[3.2.0]heptan-4-ol

CALL

926,00 € 250mg

AS56097

endo-6-Boc-6-azabicyclo[3.2.0]heptan-4-ol

CALL

995,00 € 250mg

AS56095

2-Boc-2,6-diazabicyclo[3.2.0]heptane

On Stock

353,00 € 100mg

AS18205

Page 26: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

Chemistry Services for Drug Discovery www.activate-scientifi c.com

26

Standard Pack Sizes: 1-5-10-25g • Call for 100-250-1000g pilot plant scale up

Bicyclic Rings [3.2.0]-[3.2.1]

3-Cbz-3,6-diazabicyclo[3.2.0]heptane

On Stock

295,00 € 250mg

AS28512

3-Boc-3,6-diazabicyclo[3.2.0]heptane

On Stock

394,00 € 250mg

AS56288-RAC

(1R,5R)-3-Boc-3,6-diazabicyclo[3.2.0]heptane

On Stock

587,00 € 250mg

AS56288-1R5R

(1S,5S)-3-Boc-3,6-diazabicyclo[3.2.0]heptane

On Stock

558,00 € 250mg

AS56288-1S5S

6-Boc-3,6-diazabicyclo[3.2.0]heptane

On Stock

310,00 € 250mg

AS56092-RAC

(1R,5S)-6-Boc-3,6-diazabicyclo[3.2.0]heptane

On Stock

478,00 € 250mg

AS56092-1R5S

(1S,5R)-6-Boc-3,6-diazabicyclo[3.2.0]heptane

On Stock

478,00 € 250mg

AS56092-1S5R

3-benzyl 6-tert-butyl 3,6-diazabicyclo[3.2.0]heptane-3,6-dicarboxylate

On Stock

292,00 € 250mg

AS57761

Bicyclo[3.2.1]octan-3-one

On Stock

1150,00 € 1g

AS55636

Bicyclo[3.2.1]octan-3-amine HCl

On Stock

446,00 € 100mg

AS55870

exo-8-Methyl-azabicyclo[3.2.1]octan-3-amine

On Stock

225,00 € 250mg

AS12766

3-Benzyl-3-azabicyclo[3.2.1]octan-8-one

On Stock

230,00 € 1g

AS17069

3-Azabicyclo[3.2.1]octan-8-ol HCl

On Stock

326,00 € 250mg

AS17420

3-Boc-3-azabicyclo[3.2.1]octan-8-ol

On Stock

200,00 € 100mg

AS17799

3-Boc-3-azabicyclo[3.2.1]octane-8-carboxylic acid

On Stock

478,00 € 250mg

AS55517

Methyl 3-Boc-3-azabicyclo[3.2.1]octane-8-carboxylate

On Stock

200,00 € 100mg

AS17901

8-Fluoro-3-azabicyclo[3.2.1]octane HCl

CALL

2750,00 € 1g

AS56325

8,8-Difl uoro-3-azabicyclo[3.2.1]octane HCl

On Stock

298,00 € 100mg

AS57605

8-(Trifl uoromethyl)-3-azabicyclo[3.2.1]octan-8-ol

On Stock

288,00 € 100mg

AS57606

3-Boc-3-azabicyclo[3.2.1]octan-8-amine

On Stock

189,00 € 100mg

AS57604

8-Aminomethyl-3-Boc-3-azabicyclo[3.2.1]octane HCl

On Stock

552,00 € 250mg

AS18444

8-(Boc-amino)-3-azabicyclo[3.2.1]octane

On Stock

254,00 € 100mg

AS57607

8-Oxa-3-azabicyclo[3.2.1]octane

On Stock

443,00 € 1g

AS74385-A

8-Oxabicyclo[3.2.1]octan-3-one

On Stock

158,00 € 250mg

AS55813

Page 27: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

Activate Scientifi c · Am Mitterweg 12 · D-83209 Prien · Germany · Tel: +49 (0) 8051-965166021A The Maltings · Roydon Road · Stanstead Abbotts · Hertfordshire SG12 8HG · UK · Tel: +44 (0) 1279843244

www.activate-scientifi c.com · info@activate-scientifi c.com · info-uk@activate-scientifi c.com

27

Chemistry Services for Drug Discovery www.activate-scientifi c.com

Bicyclic Rings [3.2.1]

3-Oxo-8-oxabicyclo[3.2.1]oct-6-ene

On Stock

252,00 € 250mg

AS56719

8-Oxabicyclo[3.2.1]octane-3-carboxylicacid

On Stock

290,00 € 100mg

AS55630

8-Oxabicyclo[3.2.1]octane-3-carbonitrile

On Stock

535,00 € 100mg

AS56720

8-Oxabicyclo[3.2.1]octane-3-acetic acid

On Stock

535,00 € 100mg

AS56617

8-Azabicyclo[3.2.1]octane HCl

On Stock

290,00 € 250mg

AS17447

8-Boc-8-azabicyclo[3.2.1]octane-2-carboxylic acid

On Stock

300,00 € 100mg

AS17900

Methyl 8-Boc-8-azabicyclo[3.2.1]octane-2-carboxylate

On Stock

254,00 € 100mg

AS57259

8-Methyl-8-azabicyclo[3.2.1]octan-2-amine

On Stock

1186,00 € 250mg

AS18107

3-Oxa-8-azabicyclo[3.2.1]octane HCl

On Stock

139,00 € 1g

AS12052

exo-8-Azabicyclo[3.2.1]octane-3-ol HCl

On Stock

120,00 € 250mg

AS12980

8-Methyl-8-azabicyclo[3.2.1]oct-3-ene

On Stock

254,00 € 250mg

AS43864

exo-3-Fluoro-8-azabicyclo[3.2.1]octaneHCl

On Stock

333,00 € 100mg

AS56808

8-Boc-2-fl uoro-8-azabicyclo[3.2.1]octan-3-ol

On Stock

567,00 € 1g

AS14761

8-Boc-2-fl uoro-8-azabicyclo[3.2.1]octan-3-one

On Stock

283,00 € 1g

AS14556

3,3-Difl uoro-8-azabicyclo[3.2.1]octane HCl

On Stock

300,00 € 100mg

AS12698

3-exo-8-Boc-8-azabicyclo[3.2.1]octan-3-ol

On Stock

133,00 € 250mg

AS57390

exo-8-Azabicyclo[3.2.1]octane-3-methanolHCl

On Stock

352,00 € 250mg

AS51929

endo-8-Azabicyclo[3.2.1]octane-3-methanol HCl

On Stock

223,00 € 100mg

AS57700

exo-8-Boc-8-azabicyclo[3.2.1]octane-3-methanol

On Stock

275,00 € 250mg

AS55462

endo-8-Boc-8-azabicyclo[3.2.1]octane-3-methanol

On Stock

311,00 € 100mg

AS57746

endo-3-Methoxy-8-azabicyclo[3.2.1]octaneHCl

On Stock

187,00 € 250mg

AS57029

8-Boc-3-formyl-8-azabicyclo[3.2.1]octane

On Stock

279,00 € 100mg

AS57042

endo-8-Boc-8-azabicyclo[3.2.1]octane-3-carboxylic acid

On Stock

858,00 € 250mg

AS56147

exo-8-Boc-8-azabicyclo[3.2.1]octane-3-carboxylic acid

On Stock

240,00 € 250mg

AS17561

Page 28: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

Chemistry Services for Drug Discovery www.activate-scientifi c.com

28

Standard Pack Sizes: 1-5-10-25g • Call for 100-250-1000g pilot plant scale up

Bicyclic Rings [3.2.1]-[3.2.2]-[3.3.0]

Methyl 8-Azabicyclo[3.2.1]octane-3-carboxylate HCl

On Stock

293,00 € 250mg

AS17313

8-Boc-8-azabicyclo[3.2.1]oct-3-ene-3-boronic acid pinacol ester

On Stock

200,00 € 250mg

AS12095

endo-8-Boc-8-azabicyclo[3.2.1]octan-3-amine

On Stock

150,00 € 1g

AS12576

exo-8-Boc-8-azabicyclo[3.2.1]octan-3-amine

On Stock

285,00 € 1g

AS12577

exo-8-Boc-8-azabicyclo[3.2.1]octane-3-methanamine

On Stock

365,00 € 1g

AS17734

3-(Boc-amino)-8-azabicyclo[3.2.1]octane

CALL

586,00 € 1g

AS31229

exo-3-(Boc-amino)-8-azabicyclo[3.2.1]octane

On Stock

295,00 € 1g

AS12572

endo-3-(Boc-amino)-8-azabicyclo[3.2.1]octane

On Stock

260,00 € 250mg

AS12912

endo-8-Methyl-8-azabicyclo[3.2.1]octan-3-amine

On Stock

195,00 € 1g

AS12408

1,4-Diazabicyclo[3.2.1]octane diHCl

On Stock

284,00 € 250mg

AS56439

(1R,5R)-1,4-Diazabicyclo[3.2.1]octanediHCl

On Stock

457,00 € 100mg

AS56440

2-Boc-2,6-diazabicyclo[3.2.1]octane

CALL

1650,00 € 1g

AS3933

6-Boc-3,6-diazabicyclo[3.2.1]octane HCl

On Stock

308,00 € 100mg

AS55651

3,8-Diazabicyclo[3.2.1]octan-2-one

On Stock

288,00 € 100mg

AS56937

3-Boc-3,8-diazabicyclo[3.2.1]octane

On Stock

285,00 € 1g

AS33566

3-Benzyl-3,8-diazabicyclo[3.2.1]octane

On Stock

1235,00 € 1g

AS37503

8-Boc-3,8-diazabicyclo[3.2.1]octane

On Stock

254,00 € 250mg

AS37404

8-Benzyl-3,8-diazabicyclo[3.2.1]octanediHCl

On Stock

465,00 € 1g

AS37567-B

1,4-Diazabicyclo[3.2.2]nonane

On Stock

251,00 € 1g

AS39978

1,4-Diazabicyclo[3.2.2]nonan-3-one

On Stock

361,00 € 250mg

AS12099

6-Boc-3,6-diazabicyclo[3.2.2]nonane

On Stock

222,00 € 250mg

AS42767

3-Azabicyclo[3.3.0]octane HCl

On Stock

125,00 € 5g

AS20661

Bicyclo[3.3.1]nonane-3,7-dione

On Stock

356,00 € 1g

AS80237

1-Azabicyclo[3.3.1]nonan-4-one

On Stock

1265,00 € 1g

AS16054

Page 29: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

Activate Scientifi c · Am Mitterweg 12 · D-83209 Prien · Germany · Tel: +49 (0) 8051-965166021A The Maltings · Roydon Road · Stanstead Abbotts · Hertfordshire SG12 8HG · UK · Tel: +44 (0) 1279843244

www.activate-scientifi c.com · info@activate-scientifi c.com · info-uk@activate-scientifi c.com

29

Chemistry Services for Drug Discovery www.activate-scientifi c.com

Bicyclic Rings [3.3.1]

3-Azabicyclo[3.3.1]nonane HCl

On Stock

774,00 € 500mg

AS51926

3-Boc-3-azabicyclo[3.3.1]nonan-7-one

On Stock

478,00 € 250mg

AS56082

3-Boc-3-azabicyclo[3.3.1]nonan-9-amine

CALL

1835,00 € 1g

AS18545

3-Oxa-7-azabicyclo[3.3.1]nonane

On Stock

167,00 € 250mg

AS29191

9-Azabicyclo[3.3.1]nonan-3-one HCl

On Stock

195,00 € 1g

AS51927-B

9-Benzyl-9-azabicyclo[3.3.1]nonan-3-one

On Stock

105,00 € 1g

AS20049

9-Boc-9-azabicyclo[3.3.1]nonan-3-one

On Stock

94,00 € 1g

AS20050

9-Methyl-9-azabicyclo[3.3.1]nonan-3-one

On Stock

48,00 € 1g

AS20051

9-Azabicyclo[3.3.1]nonan-3-ol

On Stock

285,00 € 1g

AS12227

endo-9-Azabicyclo[3.3.1]nonan-3-ol HCl

On Stock

187,00 € 250mg

AS56959

Methyl 9-azabicyclo[3.3.1]nonane-3-carboxylate HCl

On Stock

260,00 € 100mg

AS18447

9-Methyl-7-oxa-9-azabicyclo[3.3.1]nonan-3-one

On Stock

243,00 € 250mg

AS23343

9-Boc-9-azabicyclo[3.3.1]non-2-ene-3-boronic acid pinacol ester

On Stock

612,00 € 1g

AS18410

exo-9-Boc-9-azabicyclo[3.3.1]nonan-3-amine

On Stock

395,00 € 250mg

AS17776

endo-9-Boc-3-amino-9-azabicyclo[3.3.1]nonane

On Stock

255,00 € 1g

AS20358

exo-3-(Boc-amino)-9-azabicyclo[3.3.1]nonane

On Stock

220,00 € 100mg

AS17702

endo-3-(Boc-amino)-9-azabicyclo[3.3.1]nonane

On Stock

264,00 € 250mg

AS12564

exo-9-Boc-9-azabicyclo[3.3.1]nonane-3-methanamine

On Stock

328,00 € 250mg

AS57808

3-Oxa-9-azabicyclo[3.3.1]nonan-7-one HCl

On Stock

284,00 € 250mg

AS14839-B

9-Benzyl-3-oxa-9-azabicyclo[3.3.1]nonan-7-one

On Stock

133,00 € 250mg

AS24657

endo-3-Oxa-9-azabicyclo[3.3.1]nonan-7-olHCl

On Stock

572,00 € 250mg

AS56144

endo-9-Boc-3-oxa-9-azabicyclo[3.3.1]nonan-7-amine

On Stock

295,00 € 100mg

AS17913

exo-7-(Boc-amino)-3-oxa-9-aza-bicyclo[3.3.1]nonane

On Stock

599,00 € 100mg

AS55828

endo-7-(Boc-amino)-3-oxa-9-aza-bicyclo[3.3.1]nonane

On Stock

599,00 € 100mg

AS55829

Page 30: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

Chemistry Services for Drug Discovery www.activate-scientifi c.com

30

Standard Pack Sizes: 1-5-10-25g • Call for 100-250-1000g pilot plant scale up

Bicyclic Rings [3.3.1]-[4.1.0]-[4.2.0]

9-Boc-3-oxa-9-azabicyclo[3.3.1]nonane-7-carboxylic acid

On Stock

712,00 € 250mg

AS18057

3-Boc-3,7-diazabicyclo[3.3.1]nonane HCl

On Stock

558,00 € 250mg

AS56534

cis-3,7-Diazabicyclo[3.3.0]octane

CALL

758,00 € 1g

AS27751-CIS

3-Boc-9-oxa-3,7-diazabicyclo[3.3.1]nonane HCl

On Stock

482,00 € 100mg

AS56513

3-Boc-7-benzyl-3,7-diazabicyclo[3.3.1]nonan-9-one

On Stock

296,00 € 1g

AS26656

3-Boc-7-(2,2,2-trifl uoroacetyl)-3,7-diazabicyclo[3.3.1]nonan-9-ol

On Stock

625,00 € 1g

AS14843

9-Boc-3,9-diazabicyclo[3.3.1]nonane

On Stock

365,00 € 250mg

AS57967

2-Boc-2-azabicyclo[4.1.0]heptane-2-carboxylic acid

On Stock

403,00 € 100mg

AS74719-RAC

3-Benzyl-7-oxa-3-azabicyclo[4.1.0]heptane

CALL

425,00 € 1g

AS17105-RAC

2-Oxa-5-azabicyclo[4.1.0]heptane HCl

On Stock

495,00 € 250mg

AS72030

Bicyclo[4.2.0]octa-1,3,5-triene

On Stock

254,00 € 1g

AS37796

7-Oxobicyclo[4.2.0]octa-1,3,5-triene

On Stock

469,00 € 1g

AS34761

(S)-1,4-Diazabicyclo[4.3.0]nonane

On Stock

424,00 € 1g

AS21097-A

(R)-1,4-Diazabicyclo[4.3.0]nonane

On Stock

437,00 € 1g

AS34413

2-Boc-2,7-diazabicyclo[4.2.0]octane

On Stock

732,00 € 100mg

AS56294

7-Boc-2,7-diazabicyclo[4.2.0]octane

On Stock

688,00 € 100mg

AS56295

3-Boc-3,7-diazabicyclo[4.2.0]octane

On Stock

1180,00 € 1g

AS24701-RAC

cis-3-Boc-3,7-diazabicyclo[4.2.0]octane

On Stock

384,00 € 250mg

AS24701-CIS

(1R,6S)-3-Boc-3,7-diazabicyclo[4.2.0]octane

CALL

494,00 € 250mg

AS24701-1R6S

(1S,6R)-3-Boc-3,7-diazabicyclo[4.2.0]octane

On Stock

530,00 € 250mg

AS24701-1S6R

cis-7-Boc-3,7-diazabicyclo[4.2.0]octane

CALL

554,00 € 250mg

AS25929-CIS

(1R,6R)-7-Boc-3,7-diazabicyclo[4.2.0]octane

On Stock

595,00 € 250mg

AS25929-1R6R

(1S,6S)-7-Boc-3,7-diazabicyclo[4.2.0]octane

CALL

533,00 € 250mg

AS25929-1S6S

cis-7-Cbz-3,7-diazabicyclo[4.2.0]octane

CALL

554,00 € 250mg

AS27156-CIS

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Bicyclic Rings [4.2.0]-[4.2.1]-[5.1.0]-[5.2.0]-[5.4.0]

(1R,6R)-7-Cbz-3,7-diazabicyclo[4.2.0]octane

CALL

565,00 € 250mg

AS27156-1R6R

cis-3-Methyl-3,7-diazabicyclo[4.2.0]octane

On Stock

1458,00 € 250mg

AS27158-CIS

(1R,6S)-3-Methyl-3,7-diazabicyclo[4.2.0]octane

CALL

1458,00 € 250mg

AS27158-1R6S

(1S,6R)-3-Methyl-3,7-diazabicyclo[4.2.0]octane

On Stock

1458,00 € 250mg

AS27158-1S6R

3-Boc-3,8-diazabicyclo[4.2.0]octane

On Stock

389,00 € 250mg

AS22114-RAC

cis-3-Boc-3,8-diazabicyclo[4.2.0]octane

On Stock

376,00 € 250mg

AS22114-CIS

(1S,6R)-3-Boc-3,8-diazabicyclo[4.2.0]octane

On Stock

554,00 € 250mg

AS22114-1S6R

(1R,6S)-3-Boc-3,8-diazabicyclo[4.2.0]octane

On Stock

554,00 € 250mg

AS22114-1R6S

8-Boc-3,8-diazabicyclo[4.2.0]octane

On Stock

528,00 € 250mg

AS23633-RAC

cis-8-Boc-3,8-diazabicyclo[4.2.0]octane

CALL

554,00 € 250mg

AS23633-CIS

(1S,6R)-8-Boc-3,8-diazabicyclo[4.2.0]octane

On Stock

565,00 € 250mg

AS23633-1S6R

cis-3-Methyl-3,8-diazabicyclo[4.2.0]octane

CALL

1360,00 € 250mg

AS25914-CIS

(1R,6S)-3-Methyl-3,8-diazabicyclo[4.2.0]octane

CALL

1458,00 € 250mg

AS25914-1R6S

(1S,6R)-3-Methyl-3,8-diazabicyclo[4.2.0]octane

CALL

1458,00 € 250mg

AS25914-1S6R

(1S,6R)-8-Cbz-3,8-diazabicyclo[4.2.0]octane

CALL

612,00 € 250mg

AS25912-1S6R

cis-3-Boc-6-methyl-3,8-diazabicyclo[4.2.0]octane

On Stock

985,00 € 100mg

AS56297-CIS

3-Boc-3,9-diazabicyclo[4.2.1]nonane

On Stock

300,00 € 100mg

AS17959

9-Boc-3,9-diazabicyclo[4.2.1]nonan-4-one

On Stock

280,00 € 100mg

AS56289

4-tosyl-4-Azabicyclo[5.1.0]octane-8-carboxylic acid

On Stock

960,00 € 1g

AS80613

Ethyl 4,4-dimethyl-3,5-dioxabicyclo[5.1.0]octane-8-carboxylate

On Stock

250,00 € 250mg

AS80301

4,4-Dimethyl-3,5,8-trioxabicyclo[5.1.0]octane

On Stock

295,00 € 5g

AS80114

cis, trans, trans-3,5-Dioxabicyclo[5.1.0]octane-8-carboxylic acid ethyl ester

On Stock

279,00 € 250mg

AS15155

4-Boc-4,8-diazabicyclo[5.2.0]nonane

On Stock

624,00 € 250mg

AS25314

1,8-Diazabicyclo[5.4.0]undec-7-ene

CALL

48,00 € 25g

AS33441

Page 32: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

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32

Standard Pack Sizes: 1-5-10-25g • Call for 100-250-1000g pilot plant scale up

Cyclopropanes

2-Bromo-1-cyclopropylethan-1-one

On Stock

48,00 € 1g

AS20275

3-(Cyclopropyl)-3-oxopropanenitrile

On Stock

98,00 € 1g

AS21368

Methyl 3-(cyclopropyl)-3-oxopropanoate

On Stock

108,00 € 5g

AS20022

Ethyl 3-(cyclopropyl)-3-oxopropanoate

On Stock

114,00 € 25g

AS21397

1-Fluorocyclopropane-1-carboxylic acid

On Stock

320,00 € 250mg

AS43504

1-(Trifl uoromethyl)cyclopropane-1-carboxylic acid

On Stock

145,00 € 1g

AS55439

1-(Trifl uoromethyl)cyclopropane-1-methanol

On Stock

824,00 € 250mg

AS55911

2-Fluorocyclopropane-1-carboxylic acid

On Stock

180,00 € 250mg

AS80256-RAC

trans-2-Fluorocyclopropane-1-carboxylicacid

On Stock

220,00 € 250mg

AS80256-TRANS

(1R,2R)-2-Fluorocyclopropane-1-carboxylic acid

On Stock

260,00 € 100mg

AS80256-1R2R

(1S,2S)-2-Fluorocyclopropane-1-carboxylic acid

On Stock

260,00 € 100mg

AS80256-1S2S

2-(Trifl uoromethyl)cyclopropane-1-carboxylic acid

On Stock

237,00 € 100mg

AS57209

2-Chloro-2-fl uorocyclopropane-1-carboxylic acid

On Stock

356,00 € 1g

AS80294

(Bromomethyl)cyclopropane

On Stock

36,00 € 5g

AS50203

(Bromoethynyl)cyclopropane

On Stock

452,00 € 5g

AS25120

2-Cyano-3-(cyclopropyl)acrylic acid

On Stock

614,00 € 1g

AS18407

Cyclopropane-1-boronic acid pinacol ester

On Stock

44,00 € 1g

AS33294

1-(Cyclopropylmethyl)1H-pyrazole-4-boronic acid pinacol ester

On Stock

208,00 € 250mg

AS37149

1-(Cyclopropyl)pyrazole-5-boronic acid pinacol ester

On Stock

945,00 € 1g

AS28218

Cyclopropylmethanethiol

On Stock

360,00 € 250mg

AS18566

Cyclopropanesulfonamide

On Stock

98,00 € 5g

AS21566

Cyclopropanesulfonylchloride

On Stock

65,00 € 5g

AS34200

1-Methylcyclopropane-1-sulfonyl chloride

On Stock

158,00 € 1g

AS16172

Cyclopropane-1-methanamine

On Stock

52,00 € 5g

AS20025

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Cyclopropanes

1-Methylcyclopropan-1-amine HCl

On Stock

166,00 € 250mg

AS16174

(Cyclopropylmethyl)hydrazine diHCl

On Stock

1026,00 € 5g

AS24036

N-(Cyclopropylmethyl)cyclopropanamine

On Stock

348,00 € 1g

AS27670

1-(Aminomethyl)cyclopropan-1-ol

On Stock

375,00 € 250mg

AS37267

1-(Aminomethyl)cyclopropane-1-carboxylicacid HCl

On Stock

215,00 € 1g

AS74522

1-(2-Aminoethyl)cyclopropane-1-carboxylicacid HCl

On Stock

365,00 € 250mg

AS57025

Methyl cis-2-(Boc-amino)cyclopropane-1-carboxylate

On Stock

187,00 € 250mg

AS57263-CIS

trans-(1R,2R)-2-((Boc-amino)methyl)cyclo-propane-1-carboxylic acid

On Stock

365,00 € 250mg

AS57265-TRANS

1-Methylcyclopropan-1-ol

On Stock

260,00 € 250mg

AS36706

Boc-cyclopropane

On Stock

96,00 € 1g

AS24892

1-Methylcyclopropane-1-carboxylic acid

On Stock

142,00 € 1g

AS21123

Ethyl 1-(hydroxymethyl)cyclopropane-1-carboxylate

On Stock

262,00 € 1g

AS42928

1-Methylcyclopropane-1-carbonyl chloride

On Stock

201,00 € 250mg

AS57069

trans-2-Cyanocyclopropane-1-carboxylicacid

On Stock

255,00 € 250mg

AS57075-TRANS

Ethyl cis-2-cyanocyclopropane-1-carboxylate

On Stock

730,00 € 1g

AS57306-CIS

2-Carbamoylcyclopropane-1-carboxylicacid

On Stock

187,00 € 250mg

AS57203

trans-2-(Methoxycarbonyl)cyclopropane-1-carboxylic acid

On Stock

187,00 € 250mg

AS57208-TRANS

N-Boc-N-(3-piperidyl)cyclopropylamine

On Stock

243,00 € 250mg

AS27074

2-(Cyclopropyl)pyrimidine-5-carboxylic acid

On Stock

246,00 € 1g

AS26983

3-(Cyclopropyl)azetidin-3-ol HCl

On Stock

285,00 € 1g

AS12879

1-(Cyclopropyl)piperidin-4-one

On Stock

48,00 € 1g

AS33862

1-(Cyclopropyl)1H-pyrazole

CALL

624,00 € 250mg

AS37602

5-(Cyclopropyl)1H-imidazole

On Stock

795,00 € 1g

AS56517

1-Cyclopropyl[1,4]diazepane

On Stock

499,00 € 1g

AS74663

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34

Standard Pack Sizes: 1-5-10-25g • Call for 100-250-1000g pilot plant scale up

Oxetanes

Oxetane-2-methanamine

On Stock

383,00 € 250mg

AS51902

Oxetane-2-methanol

On Stock

170,00 € 250mg

AS51903

Oxetane-2-carboxylic acid

On Stock

335,00 € 250mg

AS6115-A

2-(Iodomethyl)oxetane

On Stock

724,00 € 1g

AS72023

Oxetan-3-one

On Stock

24,00 € 1g

AS6000

Oxetane-3-boronic acid pinacolester

On Stock

380,00 € 500mg

AS80281

Potassium trifl uoro(oxetan-3-yl)borate

On Stock

420,00 € 500mg

AS80287

3-(Iodomethyl)oxetane

On Stock

295,00 € 250mg

AS17746

3-Bromooxetane

On Stock

190,00 € 1g

AS6101

Oxetan-3-amine

On Stock

87,00 € 1g

AS6082

Oxetane-3-methanamine

On Stock

200,00 € 500mg

AS6099

N-Methyloxetane-3-amine

On Stock

200,00 € 250mg

AS6100-A

N-(Cyclopropyl)oxetan-3-amine

On Stock

620,00 € 250mg

AS17948

3-(Methylaminomethyl)oxetane

On Stock

785,00 € 250mg

AS55650

Oxetane-3-carboxylic acid

On Stock

385,00 € 1g

AS51134

3-((Phenylsulfonyl)methylene)oxetane

On Stock

180,00 € 250mg

AS80217

1-(Oxetan-3-ylidene)propan-2-one

On Stock

300,00 € 250mg

AS80220

3-(Nitromethylene)oxetane

On Stock

624,00 € 1g

AS6096

2-(3-(Nitromethyl)oxetan-3-yl)acetic acid

On Stock

537,00 € 1g

AS6050

Ethyl 2-(oxetan-3-yloxy)acetate

On Stock

184,00 € 1g

AS6044

Ethyl 2-(3-aminooxetan-3-yl)acetate

On Stock

270,00 € 250mg

AS6017

2-(Oxetan-3-ylidene)acetonitrile

On Stock

295,00 € 500mg

AS6031

Ethyl 2-(oxetan-3-ylidene)acetate

On Stock

223,00 € 1g

AS6020

3-Phenyloxetane

CALL

647,00 € 1g

AS72043

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Oxetanes

3-(Trifl uoromethyl)oxetane-3-amine HCl

On Stock

1906,00 € 1g

AS9772

3-(4-Fluorophenyl)oxetan-3-amine HCl

On Stock

189,00 € 100mg

AS57714

3-Fluoro-3-(iodomethyl)oxetane

On Stock

353,00 € 100mg

AS56310

3-Fluoro-3-phenyloxetane

CALL

1709,00 € 1g

AS72041

3-Phenyloxetane-3-methanamine

On Stock

428,00 € 100mg

AS52011

3-(Boc-amino)-3-(3-bromophenyl)oxetane

On Stock

1533,00 € 1g

AS9586

3-Allyloxetan-3-ol

On Stock

457,00 € 1g

AS6070

3,3-Dimethoxyoxetane

CALL

585,00 € 1g

AS72035

3-(Aminomethyl)oxetan-3-ol

On Stock

220,00 € 100mg

AS17813

3-(Boc-amino)oxetane-3-methanol

On Stock

380,00 € 250mg

AS17816

3-Phenyloxetan-3-ol

On Stock

285,00 € 100mg

AS52010

3-Hydroxyoxetane-3-carboxylic acid

On Stock

366,00 € 250mg

AS6122

3-(Hydroxymethyl)oxetane-3-carboxylic acid

On Stock

344,00 € 250mg

AS25604

3-Aminooxetane-3-carboxylic acid

On Stock

226,00 € 250mg

AS6015

3-Methyloxetan-3-ethanone

On Stock

285,00 € 1g

AS12538

3-(3-Bromophenyl)-3-methyloxetane

On Stock

564,00 € 100mg

AS56602

3-Methyloxetane-3-methanamine

On Stock

92,00 € 1g

AS6098

3-Methyloxetane-3-carboxaldehyde

On Stock

129,00 € 1g

AS12149

3-Methyloxetane-3-carboxylic acid

On Stock

48,00 € 1g

AS13048

3-(Oxetan-3-yl)azetidine

On Stock

382,00 € 100mg

AS43675

1-(Oxetan-3-yl)azetidin-3-amine

On Stock

260,00 € 100mg

AS55534-A

4-Iodo-1-(oxetan-3-yl)-1H-pyrazole

On Stock

485,00 € 250mg

AS80333

(3R)-1-(Oxetan-3-yl)piperidin-3-amine

On Stock

430,00 € 250mg

AS56548

5-Bromo-N-(oxetan-3-yl)pyrimidin-2-amine

On Stock

485,00 € 1g

AS9671

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36

Standard Pack Sizes: 1-5-10-25g • Call for 100-250-1000g pilot plant scale up

Cyclobutanes

Cyclobutanol

On Stock

77,00 € 1g

AS21221

Cyclobutanone

On Stock

26,00 € 1g

AS20518

Cyclobutanemethanesulfonyl chloride

On Stock

565,00 € 1g

AS41434

Bromocyclobutane

On Stock

78,00 € 5g

AS57779

Cyclobutaneboronic acid

On Stock

202,00 € 1g

AS39699

Cyclobutanehydrazine HCl

On Stock

148,00 € 250mg

AS36298

(Aminomethyl)cyclobutane HCl

On Stock

85,00 € 1g

AS12136-B

1-Cyclobutylethan-1-amine HCl

On Stock

254,00 € 100mg

AS57060

Cyclobutanecarboxamidine HCl

On Stock

856,00 € 5g

AS27587-B

N-Methoxy-N-methylcyclobutane-1-carboxamide

On Stock

158,00 € 250mg

AS57785

Cyclobutanecarbonitrile

On Stock

87,00 € 1g

AS55361

Cyclobutanecarboxylic acid

On Stock

76,00 € 25g

AS20119

Ethyl cyclobutanecarboxylate

On Stock

145,00 € 25g

AS24310

1-Cyclobutylethan-1-one

On Stock

139,00 € 1g

AS57266

2-Cyclobutylideneacetic acid

On Stock

347,00 € 1g

AS55412

3-(Cyclobutyl)-3-oxopropionitrile

On Stock

195,00 € 1g

AS12613

2-Amino-2-cyclobutylacetic acid

On Stock

260,00 € 1g

AS56883-RAC

(2R)-2-Amino-2-cyclobutylacetic acid

On Stock

328,00 € 250mg

AS56883-2R

(2S)-2-Amino-2-cyclobutylacetic acid

On Stock

328,00 € 250mg

AS56883-2S

(S)-2-(Boc-amino)-2-(cyclobutyl)acetic acid

On Stock

485,00 € 1g

AS43660

2-(Boc-amino)cyclobutane-3-propanoic acid

On Stock

187,00 € 250mg

AS57584

Ethyl 3-(cyclobutyl)-3-oxopropanoate

On Stock

199,00 € 1g

AS21737

1-Cyclobutyl-1H-pyrazole-4 boronic acidpinacol ester

On Stock

166,00 € 250mg

AS33955

1-Cyclobutyl-1H-pyrazole-5-boronic acidpinacol ester

On Stock

254,00 € 100mg

AS56920

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Activate Scientifi c · Am Mitterweg 12 · D-83209 Prien · Germany · Tel: +49 (0) 8051-965166021A The Maltings · Roydon Road · Stanstead Abbotts · Hertfordshire SG12 8HG · UK · Tel: +44 (0) 1279843244

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Cyclobutanes

1-Aminocyclobutane-1-carbonitrile

On Stock

194,00 € 250mg

AS36294

1-Methylcyclobutane-1-methanamine HCl

On Stock

352,00 € 250mg

AS72000

1-(Aminomethyl)cyclobutan-1-ol

On Stock

266,00 € 250mg

AS37286

1-Fluorocyclobutane-1-methanamine HCl

On Stock

192,00 € 100mg

AS57384

1-Aminocyclobutane-1-carboxylic acid HCl

On Stock

105,00 € 5g

AS22527

1-(Aminomethyl)cyclobutane-1-carboxylicacid HCl

On Stock

215,00 € 1g

AS74520

1-(Boc-amino)cyclobutane-1-carboxylicacid

On Stock

107,00 € 1g

AS20421

1-[(Boc-amino)methyl]cyclobutane-1-carboxylic acid

On Stock

215,00 € 1g

AS74524

1-Methylcyclobutane-1-carboxylic acid

On Stock

235,00 € 1g

AS17006

1-Phenylcyclobutane-1-carboxylic acid

On Stock

114,00 € 250mg

AS20006

1-(4-Chlorophenyl)cyclobutane-1-carboxylic acid

On Stock

96,00 € 1g

AS34923

Methyl 1-amino-cyclobutane-1-carboxylate

On Stock

132,00 € 250mg

AS13066

Methyl 1-(aminomethyl)cyclobutane-1-carboxylate HCl

On Stock

389,00 € 250mg

AS40962

2-(Benzyloxy)cyclobutan-1-one

On Stock

254,00 € 100mg

AS55885-RAC

cis-2-(Benzyloxy)cyclobutan-1-ol

On Stock

493,00 € 100mg

AS55885-CIS

cis-2-Aminocyclobutane-1-carboxylicacid HCl

On Stock

223,00 € 100mg

AS56961-BCIS

cis-2-(Boc-amino)cyclobutane-1-carboxylic acid

On Stock

333,00 € 100mg

AS57526-CIS

cis-2-(Methoxycarbonyl)cyclobutane-1-carboxylic acid

On Stock

375,00 € 100mg

AS55901-CIS

Methyl cis-2-aminocyclobutane-1-carboxylate HCl

On Stock

250,00 € 100mg

AS55853-CIS

Methyl (1R,2S)-2-aminocyclobutane-1-carboxylate

On Stock

582,00 € 100mg

AS51676-1R2S

3-Hydroxycyclobutan-1-one

On Stock

320,00 € 250mg

AS56063

3-[[(1,1-Dimethylethyl)dimethylsilyl]oxy]cyclobutan-1-one

On Stock

420,00 € 500mg

AS17655

3-(Hydroxymethyl)cyclobutan-1-one

On Stock

289,00 € 1g

AS12896

3-(Aminomethyl)cyclobutan-1-one HCl

On Stock

190,00 € 250mg

AS17332-B

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Chemistry Services for Drug Discovery www.activate-scientifi c.com

38

Standard Pack Sizes: 1-5-10-25g • Call for 100-250-1000g pilot plant scale up

Cyclobutanes

3-Bromocyclobutan-1-one

On Stock

270,00 € 250mg

AS51924

3-(Bromomethyl)cyclobutan-1-one

On Stock

285,00 € 1g

AS17068

3-(4-Bromophenyl)cyclobutan-1-one

On Stock

197,00 € 250mg

AS25112

3-(Cyclopropyl)cyclobutan-1-one

On Stock

288,00 € 100mg

AS57044

3-Methylenecyclobutane-1-carbonitrile

On Stock

245,00 € 5g

AS31180

3-Oxocyclobutane-1-carbonitrile

On Stock

116,00 € 1g

AS15262

3-Oxocyclobutane-1-carboxylic acid

On Stock

41,00 € 5g

AS22937

Methyl 3-oxocyclobutane-1-carboxylate

On Stock

28,00 € 1g

AS15166

1-Boc-cyclobutan-3-one

On Stock

146,00 € 5g

AS57588

5,8-Dioxaspiro[3.4]octane-2-carboxylicacid

On Stock

274,00 € 1g

AS17049

3-Oxocyclobutyl acetate

On Stock

265,00 € 1g

AS17138

3-Fluorocyclobutan-1-ol

On Stock

460,00 € 100mg

AS56394-RAC

trans-3-Fluorocyclobutan-1-ol

On Stock

620,00 € 100mg

AS56394-TRANS

cis-3-Aminocyclobutan-1-ol HCl

On Stock

138,00 € 250mg

AS12789-BCIS

trans-3-Aminocyclobutan-1-ol HCl

On Stock

146,00 € 250mg

AS12789-BTRANS

cis-3-(Aminomethyl)cyclobutan-1-ol HCl

On Stock

270,00 € 250mg

AS12396-BCIS

trans-3-(Aminomethyl)cyclobutan-1-ol HCl

On Stock

200,00 € 250mg

AS12396-BTRANS

cis-3-(Boc-aminomethyl)cyclobutan-1-ol

On Stock

327,00 € 250mg

AS56358-CIS

trans-3-(Boc-aminomethyl)cyclobutan-1-ol

On Stock

415,00 € 250mg

AS56358-TRANS

3-(Methylamino)cyclobutan-1-ol

On Stock

322,00 € 250mg

AS55632-RAC

cis-3-(Methylamino)cyclobutan-1-ol HCl

On Stock

538,00 € 250mg

AS55632-BCIS

trans-3-(Methylamino)cyclobutan-1-ol HCl

On Stock

334,00 € 250mg

AS55632-BTRANS

cis-(N-Boc-N-methylamino)cyclobutan-3-ol

On Stock

352,00 € 250mg

AS17642-CIS

trans-(N-Boc-N-methylamino)cyclobutan-3-ol

On Stock

260,00 € 250mg

AS17642-TRANS

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Cyclobutanes

trans-3-Aminocyclobutanemethan-1-ol HCl

On Stock

360,00 € 250mg

AS12800-BTRANS

cis-1-(Boc-amino)cyclobutane-3-methanol

On Stock

275,00 € 1g

AS12797-CIS

trans-1-(Boc-amino)cyclobutan-3-methanol

On Stock

180,00 € 250mg

AS12797-TRANS

cis-3-[[(1,1-Dimethylethyl)dimethylsilyl]oxy]cyclobutan-1-ol

On Stock

478,00 € 250mg

AS56395-CIS

3-[[(1,1-Dimethylethyl)dimethylsilyl]oxy]cyclobutan-1-ol

On Stock

256,00 € 250mg

AS56395-RAC

trans-3-[[(1,1-Dimethylethyl)dimethylsilyl]oxy]cyclobutan-1-ol

On Stock

330,00 € 100mg

AS56395-TRANS

cis-3-[[(1,1-Dimethylethyl)dimethylsilyl]oxy]cyclobutane-1-methanol

On Stock

352,00 € 250mg

AS55778-CIS

trans-3-[[(1,1-Dimethylethyl)dimethylsilyl]oxy]cyclobutane-1-methanol

On Stock

394,00 € 250mg

AS55778-TRANS

3-Fluorocyclobutan-1-amine HCl

On Stock

226,00 € 250mg

AS55653-BRAC

cis-3-Fluorocyclobutan-1-amine HCl

On Stock

220,00 € 100mg

AS55653-BCIS

trans-3-Fluorocyclobutan-1-amine HCl

On Stock

550,00 € 100mg

AS55653-BTRANS

3-Fluorocyclobutane-1-methamine HCl

On Stock

290,00 € 100mg

AS17926

3-Methoxycyclobutan-1-amine HCl

On Stock

284,00 € 250mg

AS12790-BRAC

cis-3-Methoxycyclobutan-1-amine HCl

On Stock

230,00 € 100mg

AS12790-BCIS

cis-3-(Methoxymethyl)cyclobutan-1-amineHCl

On Stock

365,00 € 250mg

AS57272-BCIS

3-Methoxycyclobutane-1-methanamine

On Stock

206,00 € 100mg

AS57645

1-(Boc-amino)cyclobutan-3-amine

On Stock

420,00 € 250mg

AS12913-RAC

cis-1-(Boc-amino)cyclobutan-3-amine

On Stock

330,00 € 250mg

AS12913-CIS

trans-1-(Boc-amino)cyclobutan-3-amine

On Stock

230,00 € 250mg

AS12913-TRANS

1-(Boc-amino)cyclobutane-3-methanamine

On Stock

537,00 € 250mg

AS18105-RAC

trans-1-(Boc-amino)cyclobutane-3-methanamine

On Stock

420,00 € 250mg

AS18105-TRANS

cis-1-(Boc-amino)cyclobutane-3-methanamine

On Stock

380,00 € 250mg

AS18105-CIS

(N-Boc-N-methylamino)cyclobutan-3-amine

On Stock

457,00 € 100mg

AS56507-RAC

trans-(N-Boc-N-methylamino)cyclobutan-3-amine

On Stock

558,00 € 250mg

AS56507-TRANS

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40

Standard Pack Sizes: 1-5-10-25g • Call for 100-250-1000g pilot plant scale up

Cyclobutanes

trans-3-(Methylsulfonyl)cyclobutan-1-amine HCl

On Stock

395,00 € 100mg

AS18203-TRANS

cis-3-(Methylsulfonyl)cyclobutan-1-amineHCl

On Stock

446,00 € 100mg

AS18203-CIS

3-Methylcyclobutane-1-carboxylic acid

On Stock

252,00 € 1g

AS55366-RAC

cis-3-Methylcyclobutane-1-carboxylic acid

On Stock

298,00 € 100mg

AS55366-CIS

trans-3-Methylcyclobutane-1-carboxylicacid

On Stock

320,00 € 100mg

AS55366-TRANS

3-(Benzyloxy)cyclobutane-1-carboxylic acid

On Stock

78,00 € 1g

AS12024

3-Hydroxycyclobutane-1-carboxylic acid

On Stock

176,00 € 1g

AS17683-RAC

cis-3-Hydroxycyclobutane-1-carboxylicacid

On Stock

296,00 € 1g

AS17683-CIS

trans-3-Hydroxycyclobutane-1-carboxylicacid

On Stock

280,00 € 250mg

AS17683-TRANS

3-Methoxycyclobutane-1-carboxylic acid

On Stock

301,00 € 250mg

AS56423-RAC

cis-3-Methoxycyclobutane-1-carboxylicacid

On Stock

284,00 € 250mg

AS56423-CIS

trans-3-Methoxycyclobutane-1-carboxylicacid

On Stock

352,00 € 250mg

AS56423-TRANS

3-(Methoxycarbonyl)cyclobutane-1-carboxylic acid

On Stock

328,00 € 250mg

AS57377

3-Chlorocyclobutane-1-carboxylic acid

On Stock

119,00 € 250mg

AS57692

trans-3-Chlorocyclobutane-1-carboxylicacid

On Stock

219,00 € 250mg

AS57911-TRANS

3-Fluorocyclobutane-1-carboxylic acid

On Stock

260,00 € 250mg

AS12895

3-(Trifl uoromethyl)cyclobutane-1-carboxylic acid

On Stock

329,00 € 100mg

AS57055

3-Aminocyclobutane-1-carboxylic acid HCl

On Stock

206,00 € 250mg

AS31858-BRAC

cis-3-Aminocyclobutane-1-carboxylicacid HCl

On Stock

200,00 € 250mg

AS31858-BCIS

3-(Aminomethyl)cyclobutane-1-carboxylicacid HCl

On Stock

277,00 € 100mg

AS57708

3-(Dimethylamino)cyclobutane-1-carboxylic acid

On Stock

189,00 € 100mg

AS57493

cis-3-(Boc-amino)cyclobutane-1-carboxylic acid

On Stock

285,00 € 1g

AS12343-CIS

3-(Boc-amino)cyclobutane-1-carboxylicacid

On Stock

145,00 € 1g

AS12343-RAC

trans-3-(Boc-amino)cyclobutane-1-carboxylic acid

On Stock

195,00 € 1g

AS12343-TRANS

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Activate Scientifi c · Am Mitterweg 12 · D-83209 Prien · Germany · Tel: +49 (0) 8051-965166021A The Maltings · Roydon Road · Stanstead Abbotts · Hertfordshire SG12 8HG · UK · Tel: +44 (0) 1279843244

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Cyclobutanes

Methyl 3-hydroxycyclobutane-1-carboxylate

On Stock

82,00 € 1g

AS12170

Methyl trans-3-hydroxycyclobutane-1-carboxylate

On Stock

184,00 € 250mg

AS17129-TRANS

Methyl 3-chlorocyclobutane-1-carboxylate

On Stock

265,00 € 1g

AS17062

Methyl 3-bromocyclobutane-1-carboxylate

On Stock

352,00 € 250mg

AS55991-RAC

Methyl trans-3-bromocyclobutane-1-carboxylate

On Stock

298,00 € 100mg

AS55991-TRANS

Methyl 3-aminocyclobutane-1-carboxylateHCl

On Stock

219,00 € 250mg

AS17453-BRAC

Methyl cis-3-aminocyclobutane-1-carboxylate HCl

On Stock

444,00 € 1g

AS17453-BCIS

Methyl 3-(aminomethyl)cyclobutane-1-carboxylate HCl

On Stock

478,00 € 250mg

AS56574

Methyl cis-3-(Boc-amino)cyclobutane-1-carboxylate

On Stock

256,00 € 1g

AS17104-CIS

Methyl trans-3-(Boc-amino)cyclo-butane-1-carboxylate

On Stock

275,00 € 1g

AS17104-TRANS

(3-Aminocyclobutyl)acetic acid

On Stock

678,00 € 250mg

AS55645-ARAC

cis-(3-Aminocyclobutyl)acetic acid HCl

On Stock

385,00 € 100mg

AS55645-BCIS

cis-3-(Boc-amino)cyclobutan-1-acetic acid

On Stock

385,00 € 100mg

AS56926-CIS

1-Methyl-3-oxocyclobutane-1-carboxylicacid

On Stock

398,00 € 1g

AS55431

Methyl 3-oxo-1-methylcyclobutane-1-carboxylate

On Stock

325,00 € 1g

AS55563

1-(Boc-amino)-1-methylcyclobutan-3-one

On Stock

394,00 € 250mg

AS55898

cis-3-Amino-1-methylcyclobutane-1-carboxylic acid HCl

On Stock

865,00 € 250mg

AS18213-CIS

trans-3-Amino-1-methylcyclobutane-1-carboxylic acid HCl

On Stock

570,00 € 100mg

AS18213-TRANS

Methyl 2,2-dimethyl-3-oxocyclobutane-1-carboxylate

On Stock

478,00 € 250mg

AS56500

cis-3-Amino-2,2-dimethylcyclobutan-1-olHCl

On Stock

589,00 € 100mg

AS55880-BCIS

1-(Boc-amino)-2,2-dimethylcyclobutan-3-one

On Stock

323,00 € 100mg

AS56941

Methyl cis-3-amino-2,2-dimethylcyclo-butane-1-carboxylate HCl

On Stock

330,00 € 100mg

AS55626-BCIS

cis-3-(Boc-amino)-2,2-dimethylcyclo-butane-1-carboxylic acid

On Stock

330,00 € 100mg

AS55627-CIS

Methyl cis-2,2-dimethyl-3-hydroxycyclo-butane-1-carboxylate

On Stock

558,00 € 250mg

AS56503-CIS

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42

Standard Pack Sizes: 1-5-10-25g • Call for 100-250-1000g pilot plant scale up

Cyclobutanes

Methyl 2,2-dimethyl-3-hydroxycyclobutane-1-carboxylate

On Stock

478,00 € 250mg

AS56503-RAC

3,3-Dimethylcyclobutan-1-methanol

On Stock

187,00 € 250mg

AS56949

2-(3,3-Dimethoxycyclobutyl)ethan-1-ol

On Stock

189,00 € 100mg

AS57268

3,3-Dimethylcyclobutan-1-amine HCl

On Stock

365,00 € 250mg

AS57014

3,3-Dimethylcyclobutane-1-methanamine

On Stock

189,00 € 100mg

AS56948

3,3-Dimethylcyclobutane-1-carboxylic acid

On Stock

143,00 € 250mg

AS55565

Methyl 3,3-dimethylcyclobutane-1-carboxylate

On Stock

295,00 € 1g

AS55460

3-Hydroxymethyl-3-methylcyclobutan-1-one

On Stock

867,00 € 1g

AS55503

3-Fluoro-3-methylcyclobutane-1-carboxylic acid

On Stock

223,00 € 100mg

AS57492

3-Amino-3-methylcyclobutan-1-ol HCl

On Stock

558,00 € 250mg

AS55638-BRAC

cis-3-Amino-3-methylcyclobutan-1-ol HCl

On Stock

621,00 € 250mg

AS55638-BCIS

trans-3-Amino-3-methylcyclobutan-1-ol HCl

On Stock

358,00 € 100mg

AS55638-BTRANS

trans-3-Hydroxy-3-methylcyclobutan-1-amine HCl

On Stock

395,00 € 100mg

AS18146-TRANS

cis-1-(Boc-amino)3-methylcyclobutan-3-ol

On Stock

305,00 € 100mg

AS56247-CIS

trans-1-(Boc-amino)3-methylcyclobutan-3-ol

On Stock

671,00 € 100mg

AS56247-TRANS

cis-3-Hydroxy-3-methylcyclobutane-1-methamine

On Stock

858,00 € 250mg

AS56401-CIS

trans-3-Hydroxy-3-methylcyclobutane-1-methamine

On Stock

724,00 € 100mg

AS56401-TRANS

cis-1-(Boc-amino)-1-methylcyclobutan-3-amine

On Stock

767,00 € 250mg

AS56428-CIS

trans-1-(Boc-amino)-1-methylcyclobutan-3-amine

On Stock

708,00 € 250mg

AS56428-TRANS

cis-1-(Boc-amino)-3-methylcyclobutan-3-amine

On Stock

564,00 € 100mg

AS56429-CIS

trans-1-(Boc-amino)-3-methylcyclobutan-3-amine

On Stock

708,00 € 250mg

AS56429-TRANS

cis-3-Amino-1-(trifl uoromethyl)cyclobutan-1-ol HCl

On Stock

493,00 € 100mg

AS56483-BCIS

3-Amino-1-(trifl uoromethyl)cyclobutan-1-ol HCl

On Stock

595,00 € 1g

AS56483-BRAC

3-Hydroxy-3-(trifl uoromethyl)cyclobutane-1-carboxylic acid

On Stock

180,00 € 250mg

AS36950

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Activate Scientifi c · Am Mitterweg 12 · D-83209 Prien · Germany · Tel: +49 (0) 8051-965166021A The Maltings · Roydon Road · Stanstead Abbotts · Hertfordshire SG12 8HG · UK · Tel: +44 (0) 1279843244

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Cyclobutanes

Methyl 3-hydroxy-3-(trifl uoromethyl)-cyclobutane-1-carboxylate

On Stock

187,00 € 250mg

AS57691

3,3-Difl uorocyclobutan-1-one

On Stock

370,00 € 100mg

AS18081

3,3-Difl uorocyclobutan-1-ol

On Stock

350,00 € 250mg

AS17595

3,3-Difl uorocyclobutane-1-methanol

On Stock

285,00 € 1g

AS51105

3,3-Difl uorocyclobutan-1-ethanol

On Stock

254,00 € 100mg

AS56935

3,3-Difl uorocyclobutan-1-amine HCl

On Stock

111,00 € 1g

AS12139

3,3-Difl uorocyclobutane-1-methanamineHCl

On Stock

250,00 € 250mg

AS12138

(3,3-Difl uorocyclobutyl)-N-methyl-methanamine HCl

On Stock

218,00 € 100mg

AS55505

3,3-Difl uorocyclobutane-1-carboxylic acid

On Stock

96,00 € 1g

AS15329

Methyl 3,3-difl uorocyclobutane-1-carboxylate

On Stock

150,00 € 1g

AS12137

Methyl 2-(3,3-difl uorocyclobutyl)acetate

On Stock

321,00 € 100mg

AS56934

1-Amino-3,3-difl uorocyclobutane-1-methanol HCl

On Stock

220,00 € 100mg

AS17804

1-(Boc-amino)-3,3-difl uorocyclobutane-1-methanol

On Stock

189,00 € 100mg

AS57595

1-(Aminomethyl)-3,3-difl uorocyclobutane-1-methanol

On Stock

260,00 € 100mg

AS56311

1-Amino-3,3-difl uorocyclobutane-1-carboxylic acid

On Stock

250,00 € 100mg

AS17924

1-(Boc-amino)-3,3-difl uorocyclobutane-1-carboxylic acid

On Stock

200,00 € 100mg

AS17697

2-(3,3-Difl uorocyclobutyl)acetic acid

On Stock

446,00 € 100mg

AS55793

2-Amino-2-(3,3-difl uorocyclobutyl)-acetonitrile HCl

On Stock

430,00 € 100mg

AS51664

2-(Boc-amino)-3-(3,3-difl uorocyclobutyl)-propanoic acid

On Stock

329,00 € 100mg

AS57416

3,3-Difl uoro-1-methylcyclobutane-1-methanol

On Stock

290,00 € 100mg

AS56433

3,3-Difl uoro-1-methylcyclobutan-1-amineHCl

On Stock

478,00 € 250mg

AS18471

3,3-Difl uoro-1-methylcyclobutane-1-methamine HCl

On Stock

290,00 € 100mg

AS55624

3,3-Difl uoro-1-methylcyclobutane-1-carboxylic acid

On Stock

289,00 € 250mg

AS55502

Methyl 3,3-difl uoro-1-methylcyclobutane-1-carboxylate

On Stock

252,00 € 250mg

AS55909

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44

Standard Pack Sizes: 1-5-10-25g • Call for 100-250-1000g pilot plant scale up

Azetidines

Azetidine HCl

On Stock

90,00 € 5g

AS23056-B

4-[(1-Azetidinyl)methyl]phenylboronicacid pinacol ester

On Stock

765,00 € 1g

AS27084

(R)-Methyl 2-azetidinecarboxylate HCl

On Stock

295,00 € 1g

AS55430

(S)-1-Boc-2-(aminomethyl)azetidine

On Stock

284,00 € 250mg

AS17393

(2R)-2-(Methoxymethyl)azetidine

On Stock

352,00 € 250mg

AS56390

(S)-Methyl 1-(2-fl uoroethyl)azetidine-2-carboxylate

On Stock

189,00 € 100mg

AS57531

(2R)-2-(Boc-aminomethyl)azetidine HCl

On Stock

254,00 € 100mg

AS57385

(2S,3R)-3-Methylazetidine-2-carboxylicacid

On Stock

254,00 € 100mg

AS57528-2S3R

(2R)-4-Oxoazetidine-2-carboxylic acid

On Stock

200,00 € 100mg

AS56329

2-Azetidin-3-yl-propan-2-ol HCl

On Stock

275,00 € 1g

AS55424

3-[(tert-Butyldimethylsilanyl)oxy]azetidine

On Stock

286,00 € 1g

AS55407

3-Fluoroazetidine HCl

On Stock

86,00 € 1g

AS5040

3-Azetidinethiol HCl

On Stock

415,00 € 250mg

AS56302

3-(Oxetan-3-yl)azetidine

On Stock

382,00 € 100mg

AS43675

3-Phenoxyazetidine

On Stock

285,00 € 1g

AS55386

1-Boc-3-acetylazetidine

On Stock

295,00 € 1g

AS55453

1-Boc-3-allylazetidine

On Stock

430,00 € 250mg

AS56015

N-Boc-3-(2-oxoethylidene)azetidine

On Stock

675,00 € 1g

AS9720

1-Boc-3-(cyclopropan-1-amine)azetidine

On Stock

526,00 € 250mg

AS56304

3-(Difl uoromethyl)azetidine HCl

On Stock

189,00 € 100mg

AS57131

1-Boc-3-(iodoethyl)azetidine

On Stock

206,00 € 250mg

AS51972

3-Methyl 1-Boc-azetidine-3-carboxylate

On Stock

274,00 € 1g

AS51974

N-(Azetidin-3-yl)methanesulfonamide HCl

On Stock

326,00 € 1g

AS55406

1-(Methylsulfonyl)-3-azetidinecarboxylicacid

On Stock

243,00 € 250mg

AS26487

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Activate Scientifi c · Am Mitterweg 12 · D-83209 Prien · Germany · Tel: +49 (0) 8051-965166021A The Maltings · Roydon Road · Stanstead Abbotts · Hertfordshire SG12 8HG · UK · Tel: +44 (0) 1279843244

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Azetidines

3-Cyano-1-azetidinesulfonylchloride

On Stock

334,00 € 1g

AS17634

1-Boc-3-methanesulfonyloxyazetidine

On Stock

32,00 € 1g

AS12668

4-[(3-Hydroxy-1-azetidinyl)methyl]phenyl-boronic acid HCl

On Stock

310,00 € 250mg

AS27445

1-(Azetidin-3-yl)-3-fl uoroazetidine oxalate

On Stock

985,00 € 1g

AS55523

1-(Oxetan-3-yl)azetidin-3-amine

On Stock

260,00 € 100mg

AS55534-A

1-Boc-3-(2-Oxopyrrolidin-1-yl)azetidine

On Stock

865,00 € 1g

AS51940

(3R)-1-(Azetidin-3-yl)-3-fl uoropyrrolidinediHCl

On Stock

321,00 € 100mg

AS56886

1-(1-Boc-pyrrolidin-3-yl)azetidine-3-carboxylic acid

CALL

585,00 € 1g

AS62932

1-(1-Boc-3-azetidinyl)pyrazole-4-boronic acid pinacol ester

On Stock

284,00 € 250mg

AS56484

1-(2-Methylsulfanyl-pyrimidin-4-yl)azetidine-3-carboxylic acid

On Stock

459,00 € 500mg

AS60009

1-(5-Fluoropyrimidin-2-yl)azetidine-3-carboxylic acid

On Stock

459,00 € 500mg

AS60012

1-(6-Chloro-pyridazin-3-yl)-azetidine-3-carboxylic acid

On Stock

403,00 € 500mg

AS60018

3,3-Difl uoroazetidine HCl

On Stock

88,00 € 1g

AS32635

(3-Fluoroazetidin-3-yl)methanol

On Stock

572,00 € 250mg

AS56419

3-(Trifl uoromethyl)azetidin-3-ol HCl

On Stock

170,00 € 250mg

AS17537

3-Fluoro-3-methylazetidine HCl

On Stock

323,00 € 100mg

AS56418

1-Boc-3-cyano-3-fl uoroazetidine

On Stock

365,00 € 250mg

AS57509

1-Boc-3-fl uoroazetidine-3-methanamine

On Stock

360,00 € 100mg

AS18172

3-(Boc-aminomethyl)-3-fl uoroazetidineHCl

On Stock

329,00 € 100mg

AS56417-B

1-(Boc-amino)-2,2-difl uoroethylazetidine

On Stock

237,00 € 100mg

AS57515

1-Boc-3-fl uoroazetidine-3-carboxylic acid

On Stock

170,00 € 250mg

AS3601

3-Amino-1-Boc-azetidine-3-carboxylic acid

On Stock

365,00 € 250mg

AS57533

1-Boc-3-ethynylazetidin-3-ol

On Stock

291,00 € 250mg

AS56305

1-Boc-2-(3-Hydroxyazetidin-3-yl)piperidine

On Stock

284,00 € 250mg

AS56400

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46

Standard Pack Sizes: 1-5-10-25g • Call for 100-250-1000g pilot plant scale up

Cyclopentanes

Iodocyclopentane

On Stock

146,00 € 5g

AS57016

(Bromomethyl)cyclopentane

On Stock

88,00 € 1g

AS44458

Cyclopentanesulfonic acid

On Stock

189,00 € 100mg

AS57126

Cyclopentanesulfonyl Chloride

On Stock

356,00 € 5g

AS27115

3-(Cyclopentyl)prop-2-enenitrile

On Stock

120,00 € 1g

AS57447

Ethyl 3-cyclopentyl-3-oxopropanoate

On Stock

155,00 € 1g

AS21738

1-(Boc-amino)cyclopentane

On Stock

187,00 € 5g

AS74118

Ethyl 2-(cyclopentylamino)acetate HCl

On Stock

120,00 € 1g

AS74617

2-(Cyclopentylamino)acetamide HCl

On Stock

161,00 € 1g

AS74614

(3-Oxocyclopentyl)boronic acid pinacolester

On Stock

399,00 € 250mg

AS66100

3-Oxocyclopentane-1-carboxylic acid

On Stock

87,00 € 1g

AS32103

(1R)-3-Oxocyclopentane-1-carboxylic acid

On Stock

187,00 € 250mg

AS57699

Methyl (1S)-3-oxocyclopentane-1-carboxylate

On Stock

328,00 € 250mg

AS57654

3-(Cyclopentyl)-4-oxobutanenitrile

On Stock

540,00 € 250mg

AS80397

1-(Trifl uoromethyl)cyclopentan-1-amineHCl

On Stock

352,00 € 250mg

AS56576

3,3-Difl uorocyclopentan-1-ol

On Stock

359,00 € 100mg

AS57444

3,3-Difl uorocyclopentane-1-methanol

On Stock

284,00 € 250mg

AS56421

(1R)-3,3-Difl uorocyclopentane-1-methanol

On Stock

300,00 € 100mg

AS57657

3,3-Difl uorocyclopentan-1-amine HCl

On Stock

324,00 € 250mg

AS12524-B

(1R)-3,3-Difl uorocyclopentan-1-amine HCl

On Stock

493,00 € 100mg

AS56422

(1S)-3,3-Difl uorocyclopentane-1-carboxylic acid

On Stock

333,00 € 100mg

AS57656

1-(3,3-Difl uorocyclopentyl)ethanone

On Stock

AS57302

1-Aminocyclopentane-1-carboxamide

On Stock

75,00 € 10g

AS33462

1-(Boc-amino)cyclopentane-1-carboxylicacid

On Stock

39,00 € 1g

AS20418

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Activate Scientifi c · Am Mitterweg 12 · D-83209 Prien · Germany · Tel: +49 (0) 8051-965166021A The Maltings · Roydon Road · Stanstead Abbotts · Hertfordshire SG12 8HG · UK · Tel: +44 (0) 1279843244

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Chemistry Services for Drug Discovery www.activate-scientifi c.com

Cyclopentanes

1-(Boc-aminomethyl)cyclopentan-1-amine

On Stock

194,00 € 250mg

AS55776

(1S,2R)-2-Amino-1-(Boc-amino)cyclopentane

On Stock

243,00 € 250mg

AS27160-1S2R

(1R,2R)-2-Aminocyclopentan-1-ol HCl

On Stock

96,00 € 1g

AS18277

cis-(Boc-amino)cyclopentan-2-ol

On Stock

478,00 € 250mg

AS56584-CIS

trans-2-(Boc-amino)cyclopentane-1-carboxylic acid

CALL

237,00 € 250mg

AS16156-TRANS

(1S,2S)-2-(Boc-amino)cyclopentane-1-carboxylic acid

On Stock

490,00 € 1g

AS16156-1S2S

3-(Boc-amino)cyclopentan-1-one

On Stock

239,00 € 1g

AS25663

(3R)-3-(Boc-amino)cyclopentan-1-one

On Stock

352,00 € 250mg

AS55015

(1S,3S)-3-Aminocyclopentan-1-ol HCl

On Stock

306,00 € 250mg

AS57772-1S3S

Methyl (1R,3S)-3-aminocyclopentane-1-carboxylate HCl

On Stock

254,00 € 100mg

AS57653-1R3S

cis-3-(Boc-amino)cyclopentan-1-ol

On Stock

285,00 € 1g

AS17421-CIS

(1R,3S)-3-(Boc-amino)cyclopentan-1-ol

On Stock

465,00 € 1g

AS17421-1R3S

(1S,3R)-3-(Boc-amino)cyclopentan-1-ol

On Stock

265,00 € 1g

AS17421-1S3R

trans-3-(Boc-amino)cyclopentan-1-ol

On Stock

290,00 € 250mg

AS17597-TRANS

(1R,3R)-3-(Boc-amino)cyclopentan-1-ol

On Stock

489,00 € 250mg

AS17597-1R3R

(1R,3S)-3-Aminocyclopentane-1-carboxylic acid

On Stock

166,00 € 250mg

AS22265-1R3S

(1S,3R)-3-Aminocyclopentane-1-carboxylic acid

On Stock

385,00 € 1g

AS22265-1S3R

(1S,3S)-3-(Boc-amino)cyclopentan-1-ol

On Stock

189,00 € 100mg

AS57857-1S3S

(1S,3R)-3-(Boc-amino)cyclopentan-1-amine

On Stock

365,00 € 250mg

AS57781-1S3R

(1R,3R)-3-(Boc-amino)cyclopentan-1-amine

On Stock

323,00 € 100mg

AS57851-1R3R

(1R,3R)-N-Boc-1-aminocyclopentane-3-carboxylic acid

On Stock

476,00 € 250mg

AS18462-1R3R

Methyl cis-3-aminocyclopentane-1-carboxylate HCl

On Stock

364,00 € 250mg

AS28504-BCIS

1-(Cyclopentyl)-5-oxopyrrolidine-3-carboxylic acid

On Stock

176,00 € 1g

AS77011

5-(Cyclopentyl)-1H-pyrazol-3-amine

On Stock

187,00 € 250mg

AS57853

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Chemistry Services for Drug Discovery www.activate-scientifi c.com

48

Standard Pack Sizes: 1-5-10-25g • Call for 100-250-1000g pilot plant scale up

Pyrrolidines

(2R)-1-Boc-2-acetylpyrrolidine

On Stock

285,00 € 250mg

AS57823

(2S)-1-Boc-2-ethynylpyrrolidine

On Stock

228,00 € 100mg

AS57304

(2R)-2-(Fluoromethyl)pyrrolidine HCl

On Stock

625,00 € 1g

AS56799

5-[(2R)-Pyrrolidin-2-yl]-2H-1,2,3,4-tetrazole HCl

On Stock

223,00 € 100mg

AS57038

1-Boc-(2S)-2-(4-Bromo-1H-imidazol-2-yl)pyrrolidine

On Stock

119,00 € 250mg

AS57453

(3R)-3-Methylpyrrolidine HCl

On Stock

143,00 € 250mg

AS57739

(3S)-3-(Methoxymethyl)pyrrolidine HCl

On Stock

255,00 € 250mg

AS57639

N-Methyl-N-[(3S)-pyrrolidin-3-yl]methane-sulfonamide HCl

On Stock

219,00 € 250mg

AS56902

[1H-Pyrazol-4-boronic acid pinacol ester-1-yl]-(3R)-1-Boc-pyrrolidine

On Stock

255,00 € 250mg

AS57001

(S)-1-Acetyl-3-hydroxypyrrolidine

On Stock

123,00 € 1g

AS21636

(3R)-1-Methanesulfonylpyrrolidin-3-amine HCl

On Stock

119,00 € 250mg

AS57570

(S)-1-(Azetidin-3-yl)pyrrolidin-3-ol HCl

On Stock

595,00 € 250mg

AS56743

(3R)-1-(Azetidin-3-yl)-3-fl uoropyrrolidinediHCl

On Stock

321,00 € 100mg

AS56886

(3S)-1-(Oxetan-3-yl)pyrrolidin-3-amine

On Stock

206,00 € 100mg

AS57712

(4R)-4-Aminopyrrolidin-2-one HCl

On Stock

365,00 € 250mg

AS57004

(R)-4-(Aminomethyl)pyrrolidin-2-one

On Stock

320,00 € 100mg

AS56482

(R)-4-Mercaptopyrrolidin-2-one

On Stock

284,00 € 250mg

AS56796

4-(Trifl uoromethyl)pyrrolidin-2-one

On Stock

254,00 € 100mg

AS57849

2-Methyl trans-1-boc-4-fl uoropyrrolidine-2-carboxylate

On Stock

157,00 € 1g

AS56964-TRANS

(2R,4S)-1-Boc-4-amino-2-methyl-pyrrolidine

On Stock

365,00 € 250mg

AS57773-2R4S

1-Boc-(2S,4S)-4-amino-2-methyl-pyrrolidine

On Stock

AS57774-2S4S

(2R,4S)-4-(Boc-amino)pyrrolidine-2-carboxylic acid

On Stock

306,00 € 250mg

AS57524-2R4S

(2S,4R)-1-Boc-4-fl uoropyrrolidine-2-methanol

On Stock

328,00 € 250mg

AS56907-2S4R

1-Boc-(2S,4S)-4-fl uoropyrrolidine-2-methanamine

On Stock

187,00 € 250mg

AS56908-2S4S

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Activate Scientifi c · Am Mitterweg 12 · D-83209 Prien · Germany · Tel: +49 (0) 8051-965166021A The Maltings · Roydon Road · Stanstead Abbotts · Hertfordshire SG12 8HG · UK · Tel: +44 (0) 1279843244

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Pyrrolidines

(2R,4S)-4-Fluoropyrrolidine-2-carboxylicacid

On Stock

187,00 € 250mg

AS56985-2R4S

(2R,4R)-1-Boc-4-fl uoropyrrolidine-2-carboxylic acid

On Stock

189,00 € 100mg

AS56963-2R4R

2-Methyl (2R,4R)-1-boc-4-fl uoropyrrolidine-2-carboxylate

On Stock

328,00 € 250mg

AS56962-2R4R

(5S)-5-(Aminomethyl)pyrrolidin-2-one

On Stock

189,00 € 100mg

AS57720

1-Boc-4-(prop-2-en-1-yl)pyrrolidin-3-one

On Stock

158,00 € 250mg

AS57098

cis-1-Boc-3-bromo-4-fl uoropyrrolidine

On Stock

328,00 € 250mg

AS57831-CIS

(3-Boc-amino)-4-fl uoropyrrolidine

On Stock

557,00 € 250mg

AS55591-RAC

3-Fluoro-4-pyrrolidinobenzoic acid

On Stock

142,00 € 1g

AS22502

cis-(3-Boc-amino)-4-fl uoropyrrolidine

On Stock

280,00 € 250mg

AS55591-CIS

trans-(3-Boc-amino)-4-fl uoropyrrolidine

On Stock

400,00 € 250mg

AS55591-TRANS

(3R,4R)-1-Boc-dihydroxypyrrolidine

On Stock

194,00 € 250mg

AS55817-3R4R

(3R,4S)-1-Boc-dihydroxypyrrolidine

On Stock

210,00 € 250mg

AS55817-3R4S

(3S,4S)-1-Boc-dihydroxypyrrolidine

On Stock

194,00 € 250mg

AS55817-3S4S

1-Boc-(3S,4S)-3-amino-4-hydroxy-pyrrolidine

On Stock

119,00 € 250mg

AS57843-3S4S

1-Boc-(3R,4R)-3-amino-4-hydroxy-pyrrolidine

On Stock

169,00 € 250mg

AS57845-3R4R

3-Methyl 1-boc-3-fl uoropyrrolidine-3-carboxylate

On Stock

187,00 € 250mg

AS57620

3-(Boc-aminomethyl)-3-fl uoropyrrolidine

On Stock

328,00 € 250mg

AS57623

[(2S)-4,4-Difl uoropyrrolidin-2-yl]methanolHCl

On Stock

187,00 € 250mg

AS57612

[(2S)-4,4-Difl uoro-1-methylpyrrolidin-2-yl]methanol

On Stock

189,00 € 100mg

AS57678

(S)-1-Boc-2-(aminomethyl)-4,4-difl uoro-pyrrolidine

On Stock

284,00 € 250mg

AS56339

(2S)-(Boc-amino)-4,4-difl uoropyrrolidine

On Stock

333,00 € 100mg

AS57613

1-Boc-4,4-difl uoropyrrolidin-3-amine

On Stock

858,00 € 500mg

AS56388

Methyl (S)-4,4-difl uoropyrrolidine-2-carboxylate HCl

On Stock

158,00 € 250mg

AS56780

(2R)-1-Boc-4,4-difl uoro-2-methyl-pyrrolidine-2-carboxylic acid

CALL

558,00 € 250mg

AS56465

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Chemistry Services for Drug Discovery www.activate-scientifi c.com

50

Standard Pack Sizes: 1-5-10-25g • Call for 100-250-1000g pilot plant scale up

Tetrahydrofurans

2-Hydroxytetrahydrofuran

On Stock

239,00 € 1g

AS24695

Tetrahydrofuran-2-carbaldehyde

On Stock

686,00 € 1g

AS41760

(S)-Tetrahydrofuran-2-carboxylic acid

On Stock

132,00 € 25g

AS33910

2-Cyanotetrahydrofuran

On Stock

215,00 € 1g

AS23829

Ethyl 3-oxo-3-(2-tetrahydrofuryl)-propanoate

On Stock

332,00 € 1g

AS24426

3-Ethynyltetrahydrofuran

On Stock

678,00 € 250mg

AS56241

3-Iodotetrahydrofuran

On Stock

185,00 € 1g

AS12617

(R)-3-Iodotetrahydrofuran

On Stock

270,00 € 250mg

AS17263

3-Bromotetrahydrofuran

On Stock

135,00 € 1g

AS12618

3-(Bromomethyl)tetrahydrofuran

On Stock

324,00 € 1g

AS12656

(S)-3-Hydroxytetrahydrofuran

On Stock

49,00 € 1g

AS32492

(R)-3-Hydroxytetrahydrofuran

On Stock

64,00 € 1g

AS32493

(S)-Tetrahydrofuran-3-methanol

On Stock

360,00 € 500mg

AS12445

(R)-Tetrahydrofuran-3-methanol

On Stock

350,00 € 250mg

AS12926

(S)-Tetrahydrofuran-3-carboxylic acid

On Stock

308,00 € 250mg

AS12443

(R)-Tetrahydrofuran-3-carboxylic acid

On Stock

214,00 € 250mg

AS12444

3-Aminotetrahydrofuran

On Stock

155,00 € 1g

AS20740-A

(S)-3-Aminotetrahydrofuran HCl

On Stock

216,00 € 1g

AS18386-B

(R)-3-Aminotetrahydrofuran HCl

On Stock

139,00 € 1g

AS32238

N-Methyltetrahydrofuran-3-amine

CALL

485,00 € 1g

AS55689-A

Tetrahydrofuran-3-methanamine

On Stock

29,00 € 1g

AS2004-A

(R)-1-Tetrahydrofuran-3-methanamine

On Stock

230,00 € 100mg

AS12446-A

(S)-1-Tetrahydrofuran-3-methanamine

On Stock

352,00 € 250mg

AS12447-A

N-Methyl-N-(tetrahydrofuran-3-yl)azetidin-3-amine diHCl

On Stock

270,00 € 100mg

AS80356

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Activate Scientifi c · Am Mitterweg 12 · D-83209 Prien · Germany · Tel: +49 (0) 8051-965166021A The Maltings · Roydon Road · Stanstead Abbotts · Hertfordshire SG12 8HG · UK · Tel: +44 (0) 1279843244

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51

Chemistry Services for Drug Discovery www.activate-scientifi c.com

Tetrahydrofurans

Methyl tetrahydrofuran-3-carboxylate

On Stock

169,00 € 1g

AS55375

(R)-Methyl tetrahydrofuran-3-carboxylate

On Stock

201,00 € 250mg

AS55709

[1-(Tetrahydrofuran-3-yl)cyclopropyl]amine HCl

On Stock

592,00 € 1g

AS78412

1-Tetrahydrofuran-3-piperazinediTFA

On Stock

320,00 € 100mg

AS80371

Ethyl 2-methyltetrahydrofuran-2-carboxylate

CALL

685,00 € 5g

AS27925

2-Amino-2-(3-tetrahydrofuranyl)ethanol

On Stock

243,00 € 250mg

AS24520

(S)-N-Boc-3-aminotetrahydrofuran-2-one

On Stock

428,00 € 5g

AS29402

Ethyl 2-oxotetrahydrofuran-3-carboxylate

On Stock

299,00 € 250mg

AS44311

(S)-(+)-5-Oxo-2-tetrahydrofurancarboxylic acid

On Stock

199,00 € 5g

AS23155

Methyl 4-oxotetrahydrofuran-3-carboxylate

On Stock

325,00 € 1g

AS12150

cis-3-(Boc-amino)-4-hydroxytetra-hydrofuran

On Stock

478,00 € 250mg

AS56150-CIS

trans-3-(Boc-amino)-4-hydroxytetra-hydrofuran

On Stock

194,00 € 250mg

AS56150-TRANS

cis-4-(Aminomethyl)tetrahydrofuran-3-ol

On Stock

457,00 € 100mg

AS56149-ACIS

cis-Tetrahydrofuran-3,4-diamine diHCl

On Stock

336,00 € 1g

AS55581-BCIS

(3R,4R)-Tetrahydrofuran-3,4-diamine

On Stock

444,00 € 250mg

AS55581-3R4R

(3S,4S)-Tetrahydrofuran-3,4-diamine

On Stock

444,00 € 250mg

AS55581-3S4S

(3S)-3-(Boc-amino)-tetrahydrofuran-5-one

On Stock

148,00 € 1g

AS44157

2-Methyltetrahydrofuran-2-methanamine

On Stock

420,00 € 250mg

AS17656

2-Methyltetrahydrofuran-2-carboxylic acid

On Stock

240,00 € 1g

AS23719

Methyl 2-methyltetrahydrofuran-2-carboxylate

On Stock

223,00 € 1g

AS24091

3-Aminotetrahydrofuran-3-carboxylic acid

On Stock

275,00 € 1g

AS12638

Butyl (S)-3-aminotetrahydrofuran-3-carboxylate

CALL

218,00 € 1g

AS90440

3-Methyltetrahydrofuran-3-carboxylic acid

On Stock

394,00 € 250mg

AS56454

3-Methyltetrahydrofuran-3-methanamine

On Stock

206,00 € 250mg

AS56455

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52

Standard Pack Sizes: 1-5-10-25g • Call for 100-250-1000g pilot plant scale up

Cyclohexanes

2-Amino-1-(cyclohexyl)ethanone HCl

CALL

558,00 € 250mg

AS56155

Ethyl 3-(cyclohexyl)-3-oxopropanoate

On Stock

155,00 € 1g

AS21739

O-(Cyclohexylmethyl)hydroxylamine

On Stock

268,00 € 250mg

AS15326

Cyclohexylsulfamoyl chloride

On Stock

765,00 € 5g

AS25427

(2R)-2-Amino-2-(cyclohexyl)ethanol

CALL

372,00 € 1g

AS90266-A2R

(2S)-2-(Boc-amino)-2-(cyclohexyl)ethanol

CALL

300,00 € 5g

AS90270-2S

(2R)-2-(Boc-amino)-3-(cyclohexyl)propionic acid

On Stock

38,00 € 1g

AS90213-2R

(R)-1-(Boc-amino)cyclohexan-1-one

On Stock

166,00 € 250mg

AS28530-1R

(1S,2S)-2-(Benzylamino)cyclohexan-1-ol

On Stock

105,00 € 1g

AS27831-1S2S

(1S,2R)-2-Methylcyclohexan-1-amine HCl

On Stock

228,00 € 250mg

AS90095-1S2R

3-(Boc-amino)cyclohexan-1-one

On Stock

105,00 € 1g

AS33914

3-(Aminomethyl)cyclohexan-1-ol

On Stock

195,00 € 1g

AS25850

(1S,3R)-3-Aminocyclohexane-1-carboxylicacid HCl

On Stock

254,00 € 100mg

AS57861-1S3R

cis-3-Aminocyclohexane-1-carboxylic acidHCl

On Stock

120,00 € 1g

AS57861-CIS

(1S,3R)-1-(Boc-amino)cyclohexan-3-amine

On Stock

385,00 € 100mg

AS57947-1S3R

(1R,3S)-1-(Boc-amino)cyclohexan-3-amine

On Stock

385,00 € 100mg

AS57947-1R3S

4-Hydroxycyclohexan-1-one

On Stock

107,00 € 1g

AS22161

4-Oxocyclohexane-1-carboxylic acid

On Stock

58,00 € 1g

AS18022

4-Fluorocyclohexane-1-carboxylic acid

On Stock

365,00 € 250mg

AS57957

1-(Bromomethyl)-4-(trifl uoromethyl)cyclo-hexane

CALL

612,00 € 1g

AS27884

cis-4-(Aminomethyl)cyclohexan-1-ol HCl

On Stock

416,00 € 250mg

AS56735-CIS

trans-4-(Aminomethyl)cyclohexan-1-ol HCl

On Stock

416,00 € 250mg

AS56735-TRANS

4-(N-Boc-N-methylamino)cyclohexan-1-ol

On Stock

465,00 € 5g

AS55446-RAC

cis-4-(N-Boc-N-methylamino)cyclohexan-1-ol

On Stock

587,00 € 250mg

AS55446-CIS

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Activate Scientifi c · Am Mitterweg 12 · D-83209 Prien · Germany · Tel: +49 (0) 8051-965166021A The Maltings · Roydon Road · Stanstead Abbotts · Hertfordshire SG12 8HG · UK · Tel: +44 (0) 1279843244

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53

Chemistry Services for Drug Discovery www.activate-scientifi c.com

Cyclohexanes

trans-4-(N-Boc-N-methylamino)cyclo-hexan-1-ol

On Stock

411,00 € 1g

AS55446-TRANS

Methyl trans-4-(Boc-amino)cyclohexane-1-carboxylate

On Stock

168,00 € 1g

AS55335-TRANS

cis-4-(Boc-amino)cyclohexane-1-methanamine

On Stock

352,00 € 250mg

AS55830-CIS

trans-1-(Boc-amino)-4-ethenylcyclo-hexane

On Stock

285,00 € 250mg

AS57794-TRANS

1-(Trifl uoromethyl)cyclohexan-1-amineHCl

On Stock

415,00 € 250mg

AS56575

1-Aminocyclohexane-1-carboxylic acid

On Stock

183,00 € 100g

AS20415

1-(Boc-amino)cyclohexane-1-carboxylicacid

On Stock

105,00 € 1g

AS20420

1-(Boc-amino)-1-methylcyclohexan-4-one

On Stock

328,00 € 250mg

AS57918

Ethyl 1-methyl-4-oxocyclohexane-1-carboxylate

On Stock

165,00 € 250mg

AS28833

1-(3-Fluorophenyl)-4-oxocyclohexane-1-carboxylic acid

On Stock

765,00 € 5g

AS26059

4-Amino-1-(trifl uoromethyl)cyclohexan-1-ol HCl

On Stock

284,00 € 250mg

AS56445-BRAC

cis-4-Amino-1-(trifl uoromethyl)cyclohexan-1-ol

On Stock

441,00 € 100mg

AS56445-ACIS

trans-4-Amino-1-(trifl uoromethyl)cyclo-hexan-1-ol

On Stock

360,00 € 100mg

AS56445-ATRANS

trans-4-Amino-4-methylcyclohexan-1-olHCl

On Stock

572,00 € 250mg

AS56405-TRANS

cis-4-(Boc-amino)-4-methylcyclohexan-1-ol

On Stock

531,00 € 250mg

AS56406-CIS

cis-4-(Boc-amino)methylcyclohexan-1-ol

On Stock

426,00 € 250mg

AS55506-CIS

4,4-Difl uorocyclohexan-1-one

On Stock

46,00 € 1g

AS51104

4,4-Difl uorocyclohexane-1-carboxaldehyde

On Stock

351,00 € 1g

AS19123

4,4-Difl uorocyclohexane-1-boronicacid pinacol ester

On Stock

450,00 € 250mg

AS28002

4,4-Difl uorocyclohexan-1-amine HCl

On Stock

135,00 € 1g

AS51757

4,4-Difl uorocyclohexane-1-methanamineHCl

On Stock

252,00 € 250mg

AS51755

4,4-Difl uorocyclohexane-1-carboxylic acid

On Stock

58,00 € 1g

AS40375

4,4-Difl uoro-1-methylcyclohexan-1-methanamine

On Stock

332,00 € 100mg

AS57909

cis-5-(Boc-amino)-3,3-difl uorocyclo-hexane-1-carboxylic acid

On Stock

339,00 € 100mg

AS57391-CIS

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54

Standard Pack Sizes: 1-5-10-25g • Call for 100-250-1000g pilot plant scale up

Piperidines

(R)-3-Fluoropiperidine HCl

On Stock

328,00 € 100mg

AS18198

(R)-1-Boc-3-methylaminopiperidine

On Stock

245,00 € 1g

AS55452

(S)-3-(Boc-aminomethyl)piperidine

On Stock

125,00 € 1g

AS55026

(S)-Methyl 1-Boc-piperidine-3-carboxylate

On Stock

113,00 € 1g

AS55030

(3R)-1-(Oxetan-3-yl)piperidin-3-amine

On Stock

430,00 € 250mg

AS56548

(1-Pyridin-2-ylmethyl-piperidin-3-yl)-methanol

CALL

145,00 € 200mg

AS60892

Pyrazine-2-carboxylic acid piperidin-3-amide HCl

CALL

136,00 € 200mg

AS61101

4-Ethynylpiperidine HCl

On Stock

284,00 € 250mg

AS56225

4-(Difl uoromethoxy)piperidine HCl

CALL

394,00 € 250mg

AS56001

1-Boc-piperidine-4-boronic acid pinacolester

On Stock

105,00 € 1g

AS41816

1-Boc-piperidine-4-carboxaldehyde

On Stock

105,00 € 5g

AS20652

1-Boc-4-(1-(Ethoxycarbonyl)cyclopropyl)piperidine

On Stock

595,00 € 250mg

AS56797

1,1,1-Trifl uoro-2-(piperidin-4-yl)propan-2-ol

On Stock

254,00 € 100mg

AS57116

(1-(5-Fluoropyrimidin-2-yl)piperidin-4-yl)methanol

On Stock

403,00 € 500mg

AS61146

1-Methanesulfonylpiperidin-4-amine

On Stock

132,00 € 1g

AS21979

1-Methylpiperidine-4-sulfonamide

On Stock

223,00 € 100mg

AS57121

1-(2,2,2-Trifl uoroacetyl)piperidine-4-carboxylic acid

On Stock

124,00 € 1g

AS14696

(3S,4S)-3-Fluoropiperidin-4-ol HCl

On Stock

199,00 € 100mg

AS57913-3S4S

cis-1-Boc-3-fl uoropiperidine-4-methanol

On Stock

340,00 € 100mg

AS14679-CIS

trans-4-Fluoro-3-piperidinol

On Stock

287,00 € 100mg

AS55578-ATRANS

1-Boc-4-fl uoropiperidine-3-methanol

CALL

1052,00 € 250mg

AS14529

trans-1-Boc-4-fl uoropiperidin-3-amine

On Stock

288,00 € 100mg

AS14541-TRANS

3-(Boc-amino)-4-fl uoropiperidine

On Stock

446,00 € 100mg

AS56324

(3S,4R)-1-Boc-3-fl uoropiperidin-4-amine

On Stock

380,00 € 250mg

AS16050-3S4R

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Piperidines

(3S,4S)-4-(Boc-amino)-3-fl uoropiperidine

On Stock

254,00 € 100mg

AS56932-3S4S

1-Boc-3-fl uoropiperidine-4-carboxylic acid

On Stock

675,00 € 250mg

AS14600

1-Boc-3-fl uoro-piperidine-5-methanol

CALL

1245,00 € 1g

AS14788

(3S,5S)-3-(Boc-amino)-5-fl uoropiperidine

On Stock

AS57603-3S5S

cis-1-Boc-3-fl uoro-5,5-dimethylpiperidin-4-ol

On Stock

189,00 € 100mg

AS57946-CIS

1-Boc-3-(aminomethyl)-3-fl uoropiperidine

On Stock

439,00 € 250mg

AS14735

3-(N-Boc-aminomethyl)-3-fl uoropiperidine

On Stock

254,00 € 100mg

AS57958

4-Fluoropiperidine-4-methanol

On Stock

287,00 € 250mg

AS16119-A

4-(Fluoromethyl)piperidin-4-ol HCl

On Stock

295,00 € 250mg

AS17539

4-(Trifl uoromethyl)piperidin-4-ol

On Stock

187,00 € 250mg

AS56973

4-Fluoro-1-methylpiperidine-4-methanol

On Stock

310,00 € 250mg

AS24006

3,3-Difl uoropiperidin-4-one HCl

On Stock

320,00 € 250mg

AS55482

4-(Boc-amino)-3,3-difl uoropiperidine

On Stock

382,00 € 100mg

AS18125

1-Boc-3,3-difl uoro-4-methylenepiperidine

On Stock

425,00 € 250mg

AS14780

4-Ethyl 1-Boc-3,3-difl uoro-4-methyl-piperidine-4-carboxylate

On Stock

428,00 € 250mg

AS14535

1-Boc-3,3-difl uoropiperidin-5-ol

On Stock

380,00 € 100mg

AS14783

1-Boc-3,3-difl uoropiperidine-5-methanol

On Stock

543,00 € 250mg

AS14782

4,4-Difl uoro-2-methylpiperidine HCl

On Stock

234,00 € 250mg

AS17840

3-(Boc-amino)-4,4-difl uoropiperidine

On Stock

333,00 € 100mg

AS56307

1-Boc-4,4-difl uoropiperidine-3-methanol

On Stock

609,00 € 250mg

AS14801

5,5-Difl uoropiperidin-2-one

On Stock

223,00 € 100mg

AS57706

5,5-Difl uoropiperidine-2-carboxylic acid

On Stock

370,00 € 250mg

AS17674

5,5-Difl uoropiperidine-3-carboxylicacid HCl

On Stock

832,00 € 250mg

AS14749

3-(Boc-amino)-5,5-difl uoropiperidine

On Stock

250,00 € 100mg

AS56323

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Chemistry Services for Drug Discovery www.activate-scientifi c.com

56

Standard Pack Sizes: 1-5-10-25g • Call for 100-250-1000g pilot plant scale up

Tetrahydropyrans

Tetrahydropyran-2-carboxylic acid

On Stock

132,00 € 250mg

AS20728

Tetrahydropyran-2-methanamine

On Stock

239,00 € 1g

AS20726

2-(3-Bromopropoxy)tetrahydropyran

On Stock

167,00 € 5g

AS23675

2-[[(Tetrahydropyran-2-yl)oxy]methyl]benzaldehyde

CALL

166,00 € 250mg

AS27270

4-[(Tetrahydropyran-2-yl)oxy]phenyl-boronic acid

On Stock

157,00 € 25g

AS27447

2-[4-(Tetrahydropyran-2-yloxy)phenyl]ethylamine

CALL

536,00 € 1g

AS28227

6-Amino-9-(tetrahydropyran-2-yl)-9H-purine

CALL

536,00 € 1g

AS28496

3-Bromotetrahydropyran

On Stock

269,00 € 500mg

AS37105

(S)-3-Aminotetrahydropyran HCl

On Stock

243,00 € 250mg

AS26910

(R)-3-Aminotetrahydropyran HCl

On Stock

230,00 € 250mg

AS26911-B

4-Bromotetrahydropyran

On Stock

32,00 € 1g

AS20466

4-(Bromomethyl)tetrahydropyran

On Stock

47,00 € 1g

AS1354

Tetrahydropyran-4-methanol

On Stock

115,00 € 1g

AS20467

4-Aminotetrahydropyran

On Stock

86,00 € 1g

AS20459-A

4-[(Methylamino)methyl]tetrahydropyran

On Stock

862,00 € 1g

AS28758

Tetrahydropyran-4-carboxaldehyde

On Stock

85,00 € 1g

AS12601

Tetrahydropyran-4-carboxamidine HCl

On Stock

190,00 € 250mg

AS17155

Tetrahydropyranyl-4-acetic acid

On Stock

107,00 € 1g

AS12603

Ethyl 3-Oxo-3-(4-tetrahydropyranyl)propanoate

On Stock

166,00 € 250mg

AS24196

4-Tetrahydropyranylglycine

On Stock

224,00 € 1g

AS12758

Methyl 2-amino-2-(tetrahydropyran-4-yl)acetate HCl

On Stock

197,00 € 250mg

AS28856

4-(4-Bromophenyl)tetrahydropyran

On Stock

132,00 € 250mg

AS24948

4-(4-Tetrahydropyranyl)phenylboronic acidpinacol ester

On Stock

166,00 € 250mg

AS26394

1-[2-[(Tetrahydropyran-4-yl)oxy]phenyl]methylamine

CALL

452,00 € 1g

AS27205

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Tetrahydropyrans

6-(Tetrahydropyran-4-yloxy)pyridine-3-boronic acid pinacol ester

On Stock

176,00 € 250mg

AS32641

3-Chlorotetrahydropyran-4-one

CALL

685,00 € 5g

AS28705

trans-4-Aminotetrahydropyran-3-ol

On Stock

520,00 € 1g

AS17921-ATRANS

cis-4-Aminotetrahydropyran-3-ol HCl

On Stock

284,00 € 250mg

AS17921-BCIS

trans-3-Amino-4-hydroxytetrahydropyranHCl

On Stock

158,00 € 250mg

AS57895-TRANS

(3R,4R)-3-Amino-4-hydroxytetrahydro-pyran

On Stock

206,00 € 250mg

AS18162-3R4R

(3S,4S)-3-Amino-4-hydroxytetrahydro-pyran

On Stock

200,00 € 250mg

AS18162-3S4S

cis-4-Amino-3-(methoxy)tetrahydropyran

On Stock

420,00 € 250mg

AS55349-CIS

trans-4-amino-3-(methoxy)tetrahydropyran

On Stock

478,00 € 250mg

AS55349-TRANS

cis-3-Methyl-4-aminotetrahydropyran HCl

CALL

478,00 € 250mg

AS56332-BCIS

trans-3-Methyl-4-aminotetrahydropyranHCl

On Stock

284,00 € 250mg

AS56332-BTRANS

3-Fluoro-4,4-dihydroxytetrahydropyran

On Stock

725,00 € 1g

AS55488

4-Ethynyltetrahydropyran-4-ol

On Stock

284,00 € 250mg

AS56447

4-Aminotetrahydropyran-4-methanol

On Stock

484,00 € 1g

AS24734

4-Methyltetrahydropyran-4-carboxylic acid

On Stock

267,00 € 1g

AS23720

4-Aminotetrahydropyran-4-carboxylic acid

On Stock

140,00 € 1g

AS24760

4-(Boc-amino)tetrahydropyran-4-carboxylic acid

On Stock

442,00 € 1g

AS24258

Methyl 4-aminotetrahydropyran-4-carboxylate

On Stock

296,00 € 1g

AS26636

Methyl 4-fl uorotetrahydro-2H-pyran-4-carboxylate

On Stock

352,00 € 250mg

AS56357

2,2-Dimethyltetrahydropyran-4-ol

On Stock

195,00 € 1g

AS26900

2,2-Dimethyltetrahydropyran-4-carbaldehyde

On Stock

243,00 € 250mg

AS27258

(R)-2-Methyltetrahydropyran-4-one

On Stock

478,00 € 250mg

AS56242

(2S,5R)-5-(Boc-amino)tetrahydropyran-2-carboxylic acid

On Stock

635,00 € 100mg

AS56450-2S5R

1-(2-Tetrahydropyranyl)1H-pyrazole-4-boronic acid pinacol ester

On Stock

42,00 € 1g

AS12378

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58

Standard Pack Sizes: 1-5-10-25g • Call for 100-250-1000g pilot plant scale up

Piperazines

1N-Isopropylpiperazine

On Stock

48,00 € 5g

AS20368

1-(Cyclopropylmethyl)piperazine

On Stock

123,00 € 1g

AS20562

1-(Cyclopropylcarbonyl)piperazine

On Stock

259,00 € 5g

AS20528

1-(3-Fluorophenyl)piperazine

On Stock

120,00 € 1g

AS74245

1-(2-Trifl uoromethylphenyl)piperazine

On Stock

66,00 € 1g

AS74284

1-[2-(Methylsulphonyl)phenyl]piperazine

On Stock

170,00 € 1g

AS21340

1-[4-(2-Hydroxyethyl)-1-piperazinyl]ethanone

On Stock

105,00 € 5g

AS25932

1-Boc-4-(4-amino-2-trifl uoromethylphenyl)piperazine

On Stock

187,00 € 1g

AS30067

(2R)-1,2-Dimethylpiperazine

On Stock

352,00 € 250mg

AS55570

(2S)-1,2-Dimethylpiperazine

On Stock

485,00 € 1g

AS26835-A

(3R)-1,3-Dimethylpiperazine hemioxalate

On Stock

328,00 € 250mg

AS57800

(5R)-1,5-Dimethylpiperazin-2-one

On Stock

395,00 € 250mg

AS3041

(2S,5R)-1-Boc-2,5-dimethylpiperazine

On Stock

285,00 € 1g

AS3579-2S5R

(3S,5S)-1-Boc-3,5-dimethylpiperazine

On Stock

620,00 € 250mg

AS3215-3S5S

(3R,5R)-1-Boc-3,5-dimethylpiperazine

On Stock

620,00 € 250mg

AS3221-3R5R

(2R,6S)-2,6-Dimethylpiperazine

On Stock

37,00 € 5g

AS18036-CIS

(2S,6S)-1-Boc-2,6-dimethylpiperazine

On Stock

620,00 € 250mg

AS3216-2S6S

(2R,6R)-1-Boc-2,6-dimethylpiperazine

On Stock

620,00 € 250mg

AS3222-2R6R

cis-2-[2,6-Dimethylpiperazin-1-yl]acetamide

On Stock

545,00 € 250mg

AS80350-CIS

1-Boc-2,2-dimethylpiperazine HCl

On Stock

236,00 € 1g

AS12101

1-Boc-3,3-dimethylpiperazine

On Stock

185,00 € 1g

AS13361

1-Methanesulfonylpiperazine

On Stock

105,00 € 5g

AS20639

4-Methyl-1-piperazinecarbonyl chlorideHCl

CALL

98,00 € 25g

AS25305

3-Amino-1-(4-methylpiperazin-1-yl)-1-propanone diHCl

On Stock

172,00 € 1g

AS74027

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Activate Scientifi c · Am Mitterweg 12 · D-83209 Prien · Germany · Tel: +49 (0) 8051-965166021A The Maltings · Roydon Road · Stanstead Abbotts · Hertfordshire SG12 8HG · UK · Tel: +44 (0) 1279843244

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Chemistry Services for Drug Discovery www.activate-scientifi c.com

Piperazines

4-(4-Boc-piperazino)phenylboronic acidpinacol ester

On Stock

114,00 € 250mg

AS23073

4-(4-Methylpiperazin-1-yl)phenylboronicacid

On Stock

132,00 € 1g

AS21040

4-((4-Methylpiperazin-1-yl)methyl)phenyl-boronic acid pinacol ester

On Stock

113,00 € 1g

AS41747

2-Fluoro-4-(4-methylpiperazin-1-yl)benzoic acid

On Stock

199,00 € 1g

AS22486

3-Fluoro-4-(piperazin-1-yl)benzonitrile

On Stock

123,00 € 1g

AS20264

5-Fluoro-2-piperazinobenzoic acid

On Stock

199,00 € 1g

AS22474

1-Boc-4-(pyrrolidin-3-yl)piperazine

On Stock

488,00 € 1g

AS74440

1-[(2-Pyridyl)methyl]piperazine

On Stock

87,00 € 1g

AS20664

1-(3-Trifl uoromethylpyridin-2-yl)piperazine

On Stock

197,00 € 5g

AS74087

5-Bromo-2-(4-methylpiperazin-1-yl)-3-(trifl uoromethyl)pyridine HCl

CALL

782,00 € 5g

AS68507

2-[4-(6-Amino-2-methylpyrimidin-4-yl)piperazin-1-yl]ethanol

On Stock

338,00 € 1g

AS30440

5-Fluoro-2-(2-methylpiperazin-1-yl)pyrimidine HCl

CALL

403,00 € 500mg

AS62421

Cyclopropyl(6-piperazin-1-yl-pyrimidin-4-yl)amine HCl

On Stock

468,00 € 500mg

AS62477

1-Boc-piperazine-2-one

On Stock

141,00 € 250mg

AS26547

1-Methylpiperazin-2-one

On Stock

265,00 € 1g

AS3082-A

1-Ethylpiperazin-2-one

On Stock

399,00 € 1g

AS3083

1-Isopropylpiperazin-2-one

On Stock

912,00 € 5g

AS23374

1-(4-Aminophenyl)piperazin-2-one

On Stock

158,00 € 250mg

AS20455

1-(1,1-Dimethylethyl)piperazin-2-one

On Stock

450,00 € 250mg

AS80337

1-(Tetrahydro-2H-pyran-4-yl)piperazin-2-one HCl

On Stock

680,00 € 250mg

AS80367

(S)-Piperazine-2-carboxylic acid

On Stock

52,00 € 1g

AS55033

2-(4-Fluorophenyl)piperazine diHCl

On Stock

294,00 € 1g

AS30077

2-(4-Isopropylpiperazin-1-yl)ethylamine

On Stock

187,00 € 1g

AS74178

4-(4-Piperazine-2-phenyl)morpholine

On Stock

254,00 € 1g

AS30089

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60

Standard Pack Sizes: 1-5-10-25g • Call for 100-250-1000g pilot plant scale up

Morpholines-Thiomorpholines-Oxazepanes

(R)-2-Methylmorpholine HCl

On Stock

465,00 € 1g

AS16124

(S)-2-Methylmorpholine HCl

On Stock

276,00 € 250mg

AS31353-B

(R)-2-Ethylmorpholine

CALL

320,00 € 250mg

AS12234

(R)-2-Isopropylmorpholine

On Stock

350,00 € 250mg

AS3638

(S)-2-Isopropylmorpholine

On Stock

360,00 € 250mg

AS3639

(S)-2-Benzylmorpholine

On Stock

356,00 € 250mg

AS12236

(S)-N-Boc-morpholine-2-methanol

On Stock

154,00 € 1g

AS12059

(R)-2-(Methoxymethyl)morpholine HCl

On Stock

220,00 € 250mg

AS12245-B

(S)-2-(Methoxymethyl)morpholine HCl

On Stock

320,00 € 250mg

AS3631-B

(S)-N-Boc-morpholine-2-carbaldehyde

On Stock

360,00 € 250mg

AS12061

(R)-N-Boc-morpholine-2-carbaldehyde

On Stock

360,00 € 250mg

AS12062

(R)-N-Boc-morpholine-2-carboxylic acid

On Stock

295,00 € 1g

AS12063

Methyl (R)-morpholine-2-carboxylate HCl

On Stock

332,00 € 1g

AS12238

Morpholine-2-methanamine

On Stock

123,00 € 250mg

AS21856

N-Boc-morpholine-2-methanamine

On Stock

384,00 € 1g

AS22687

(R)-2-(Boc-aminomethyl)morpholine

On Stock

985,00 € 1g

AS55518

2-(3,4-Difl uorophenyl)morpholine HCl

On Stock

201,00 € 250mg

AS27032

2-(1H-Imidazol-2-yl)morpholine HCl

On Stock

430,00 € 250mg

AS56609

4-(4-Piperazine-2-phenyl)morpholine

On Stock

254,00 € 1g

AS30089

3-Ethylmorpholine

On Stock

444,00 € 1g

AS3435

(R)-3-Ethylmorpholine

On Stock

240,00 € 250mg

AS3434

(S)-3-Benzylmorpholine HCl

On Stock

737,00 € 1g

AS3421

(S)-3-(Methoxymethyl)morpholine HCl

On Stock

283,00 € 250mg

AS3451

N-Boc-morpholine-3-methanol

On Stock

159,00 € 250mg

AS25119

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Activate Scientifi c · Am Mitterweg 12 · D-83209 Prien · Germany · Tel: +49 (0) 8051-965166021A The Maltings · Roydon Road · Stanstead Abbotts · Hertfordshire SG12 8HG · UK · Tel: +44 (0) 1279843244

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61

Chemistry Services for Drug Discovery www.activate-scientifi c.com

Morpholines-Thiomorpholines-Oxazepanes

4-Boc-3-(aminomethyl)morpholine

On Stock

376,00 € 250mg

AS13087

(S)-3-(Boc-aminomethyl)morpholine

On Stock

865,00 € 1g

AS3658

4-Boc-3-morpholinecarboxylic acid

On Stock

200,00 € 1g

AS21171

Methyl 3-morpholinecarboxylate

On Stock

240,00 € 1g

AS21021

(R)-N-Boc-morpholine-3-nitrile

CALL

993,00 € 1g

AS3660

4-Methyl-morpholine-3-carbonitrile

On Stock

227,00 € 1g

AS74561

4-Boc-morpholine

On Stock

19,00 € 1g

AS38006

4-Morpholineacetic Acid

On Stock

42,00 € 1g

AS20714

4-(2-Bromoethyl)morpholine HBr

On Stock

105,00 € 1g

AS23354

4-(3-Chloropropyl)morpholine

On Stock

78,00 € 5g

AS22352-A

4-(3-Bromopropyl)morpholine HBr

CALL

267,00 € 1g

AS29556

4-(4-Amino-1-butyl)morpholine

On Stock

215,00 € 1g

AS74553

(S)-4-(2-Amino-propan-1-yl)morpholine

On Stock

699,00 € 1g

AS74646

4-[2-(2-Hydroxyethoxy)ethyl]morpholine

On Stock

239,00 € 1g

AS28853

Morpholine-4-sulfonyl chloride

On Stock

41,00 € 1g

AS41890

4-(Morpholine-4-carbonyl)phenylboronicacid pinacol ester

On Stock

271,00 € 5g

AS27430

4-(Azetidin-3-yl)-2,6-dimethylmorpholine

On Stock

223,00 € 100mg

AS56990

4-(3-Fluoro-4-nitrophenyl)morpholine

On Stock

296,00 € 1g

AS23232

4-(4-Bromo-2-fl uorophenyl)morpholine

On Stock

178,00 € 1g

AS23256

4-(Azetidin-3-yl)morpholine HCl

On Stock

325,00 € 1g

AS12877

4-(6-Bromopyrazin-2-yl)morpholine

On Stock

254,00 € 1g

AS30675

trans-2,5-Dimethylmorpholine

On Stock

785,00 € 1g

AS3440-ATRANS

(2S,5S)-2,5-Dimethylmorpholine HCl

On Stock

387,00 € 250mg

AS3440-2S5S

(2R,5R)-2,5-Dimethylmorpholine HCl

On Stock

323,00 € 250mg

AS3440-2R5R

Page 62: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

62

Standard Pack Sizes: 1-5-10-25g • Call for 100-250-1000g pilot plant scale up

www.activate-scientifi c.comChemistry Services for Drug Discovery

Morpholines-Thiomorpholines-Oxazepanes

cis-3,5-Dimethylmorpholine

On Stock

200,00 € 250mg

AS13436-ACIS

(3R,5R)-Dimethylmorpholine

On Stock

323,00 € 250mg

AS13436-A3R5R

trans-2,6-Dimethylmorpholine

On Stock

220,00 € 250mg

AS17516-TRANS

(2R,6R)-Dimethylmorpholine

On Stock

440,00 € 250mg

AS17516-2R6R

2,2-Dimethylmorpholine

On Stock

172,00 € 250mg

AS56638-A

Methyl 4-boc-2-methylmorpholine-2-carboxylate

On Stock

774,00 € 1g

AS90283

4-(Azetidin-3-yl)-2,2-dimethylmorpholinediTFA

On Stock

280,00 € 100mg

AS55981

2-Methylmorpholin-3-one

On Stock

152,00 € 250mg

AS29282

3,3-Dimethylmorpholine

On Stock

286,00 € 1g

AS3427

N-Boc-3-ethylmorpholine-3-carboxylic acid

On Stock

450,00 € 250mg

AS27073

3-Ethylmorpholine-3-carboxylic acid

On Stock

485,00 € 250mg

AS27388

4-Benzyl-5-oxomorpholine-3-carboxylicacid

On Stock

105,00 € 1g

AS21701

(S)-4-Benzyl-5-oxomorpholine-3-carboxylic acid

On Stock

132,00 € 1g

AS21712

Thiomorpholine-1-oxide HCl

On Stock

368,00 € 1g

AS51861

Thiomorpholine-1,1-dioxide HCl

On Stock

39,00 € 1g

AS15190

N-Boc-thiomorpholine-2-carboxylic acid

On Stock

149,00 € 250mg

AS24089

Ethyl thiomorpholine-2-carboxylate HCl

On Stock

252,00 € 1g

AS29275

N-Boc-thiomorpholine-3-carboxylic acid

On Stock

229,00 € 1g

AS25565

4-Azetidin-3-yl-thiomorpholine-1,1-dioxidediHCl

On Stock

350,00 € 250mg

AS51942-B

(1,4-Oxazepan-2-yl)methanol

On Stock

342,00 € 1g

AS23574-A

4-Boc-1,4-oxazepane-2-methanol

On Stock

233,00 € 1g

AS22631

4-Boc-1,4-oxazepane-2-carboxylic acid

On Stock

296,00 € 1g

AS21583

Methyl 1,4-oxazepane-2-carboxylate

CALL

324,00 € 250mg

AS21581

4-Boc-6-amino-1,4-oxazepane

On Stock

785,00 € 1g

AS44021

Page 63: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

Copyright © 2016 Activate Scientifi c GmbH

Page 64: TThe SPhe SP3--CollectionCollection · availability of region-isomers within related templates allows swift access to SAR and the inclusion of heteroatoms aids the modifi cation

The SP3-Collection